ATE473960T1 - Verfahren zur herstellung von 4,5-diamino- shikimisäure - Google Patents
Verfahren zur herstellung von 4,5-diamino- shikimisäureInfo
- Publication number
- ATE473960T1 ATE473960T1 AT05779453T AT05779453T ATE473960T1 AT E473960 T1 ATE473960 T1 AT E473960T1 AT 05779453 T AT05779453 T AT 05779453T AT 05779453 T AT05779453 T AT 05779453T AT E473960 T1 ATE473960 T1 AT E473960T1
- Authority
- AT
- Austria
- Prior art keywords
- shikimic acid
- diamino
- producing
- alkyl
- independent
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 150000003364 shikimic acids Chemical class 0.000 abstract 2
- 102000005348 Neuraminidase Human genes 0.000 abstract 1
- 108010006232 Neuraminidase Proteins 0.000 abstract 1
- 125000001589 carboacyl group Chemical group 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- VSZGPKBBMSAYNT-RRFJBIMHSA-N oseltamivir Chemical compound CCOC(=O)C1=C[C@@H](OC(CC)CC)[C@H](NC(C)=O)[C@@H](N)C1 VSZGPKBBMSAYNT-RRFJBIMHSA-N 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 230000003612 virological effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/04—Formation of amino groups in compounds containing carboxyl groups
- C07C227/10—Formation of amino groups in compounds containing carboxyl groups with simultaneously increasing the number of carbon atoms in the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
- C07C229/48—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
- C07C227/18—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions involving amino or carboxyl groups, e.g. hydrolysis of esters or amides, by formation of halides, salts or esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04104227 | 2004-09-02 | ||
| PCT/EP2005/009121 WO2006024436A1 (en) | 2004-09-02 | 2005-08-24 | Process for the preparation of 4,5-diamino shikimicacid |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE473960T1 true ATE473960T1 (de) | 2010-07-15 |
Family
ID=35542318
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT05779453T ATE473960T1 (de) | 2004-09-02 | 2005-08-24 | Verfahren zur herstellung von 4,5-diamino- shikimisäure |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US7514580B2 (de) |
| EP (1) | EP1791808B1 (de) |
| JP (1) | JP4682204B2 (de) |
| KR (1) | KR100859902B1 (de) |
| CN (1) | CN101010289B (de) |
| AT (1) | ATE473960T1 (de) |
| CA (1) | CA2577192C (de) |
| DE (1) | DE602005022326D1 (de) |
| DK (1) | DK1791808T3 (de) |
| ES (1) | ES2345778T3 (de) |
| IL (1) | IL181317A (de) |
| MX (1) | MX2007002316A (de) |
| TW (1) | TW200621683A (de) |
| WO (1) | WO2006024436A1 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101801914B (zh) * | 2007-09-18 | 2013-06-05 | 弗·哈夫曼-拉罗切有限公司 | 从莽草酸生成磷酸奥司他韦的方法 |
| JP5698128B2 (ja) | 2009-06-09 | 2015-04-08 | 国立大学法人 岡山大学 | ジヒドロキシヘキセン酸エステル及びその製造方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0920410B1 (de) * | 1996-08-23 | 2002-03-27 | Gilead Sciences, Inc. | Verfahren zur herstellung von cyclohexen-carboxylatderivate |
| EP1059283B1 (de) | 1999-06-11 | 2003-05-28 | F. Hoffmann-La Roche Ag | Verfahren zur Herstellung des Neuraminidase-Inhibitoren ro-64-0796 |
| US6462226B1 (en) * | 1999-12-03 | 2002-10-08 | Hoffmann-La Roche Inc. | Process for the preparation of 4,5-diamino shikimic acid derivatives |
| US6403824B2 (en) * | 2000-02-22 | 2002-06-11 | Hoffmann-La Roche Inc. | Process for the preparation for 4,5-diamino shikimic acid derivatives |
| US6518048B2 (en) * | 2000-04-10 | 2003-02-11 | Hoffmann-La Roche Inc. | Stereo-specific synthesis of shimikic acid derivatives with improved efficiency |
-
2005
- 2005-08-24 DK DK05779453.9T patent/DK1791808T3/da active
- 2005-08-24 CA CA2577192A patent/CA2577192C/en not_active Expired - Fee Related
- 2005-08-24 KR KR1020077004856A patent/KR100859902B1/ko not_active Expired - Fee Related
- 2005-08-24 AT AT05779453T patent/ATE473960T1/de active
- 2005-08-24 WO PCT/EP2005/009121 patent/WO2006024436A1/en not_active Ceased
- 2005-08-24 ES ES05779453T patent/ES2345778T3/es not_active Expired - Lifetime
- 2005-08-24 DE DE602005022326T patent/DE602005022326D1/de not_active Expired - Lifetime
- 2005-08-24 EP EP05779453A patent/EP1791808B1/de not_active Expired - Lifetime
- 2005-08-24 MX MX2007002316A patent/MX2007002316A/es active IP Right Grant
- 2005-08-24 JP JP2007528738A patent/JP4682204B2/ja not_active Expired - Fee Related
- 2005-08-24 CN CN2005800294860A patent/CN101010289B/zh not_active Expired - Fee Related
- 2005-08-30 TW TW094129673A patent/TW200621683A/zh unknown
- 2005-08-30 US US11/215,753 patent/US7514580B2/en not_active Expired - Fee Related
-
2007
- 2007-02-13 IL IL181317A patent/IL181317A/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| TW200621683A (en) | 2006-07-01 |
| DE602005022326D1 (de) | 2010-08-26 |
| DK1791808T3 (da) | 2010-08-09 |
| EP1791808B1 (de) | 2010-07-14 |
| IL181317A (en) | 2011-12-29 |
| JP2008511568A (ja) | 2008-04-17 |
| CN101010289A (zh) | 2007-08-01 |
| CA2577192A1 (en) | 2006-03-09 |
| US7514580B2 (en) | 2009-04-07 |
| US20060047002A1 (en) | 2006-03-02 |
| IL181317A0 (en) | 2007-07-04 |
| MX2007002316A (es) | 2007-04-17 |
| CA2577192C (en) | 2013-01-15 |
| EP1791808A1 (de) | 2007-06-06 |
| CN101010289B (zh) | 2011-05-25 |
| JP4682204B2 (ja) | 2011-05-11 |
| ES2345778T3 (es) | 2010-10-01 |
| KR100859902B1 (ko) | 2008-09-23 |
| KR20070039973A (ko) | 2007-04-13 |
| WO2006024436A1 (en) | 2006-03-09 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| WO2001028996A3 (en) | Pyrrolidine derivatives, their preparation and their use as inhibitors of neuraminidases | |
| MX2009003739A (es) | Derivados de hidrobenzamida como inhibidores de hsp90. | |
| ATE478084T1 (de) | Verfahren zur herstellung von 4'- azidocytidinderivaten | |
| MA29464B1 (fr) | Methode de preparation d'acides 1,6-dihydro-6-oxo-4-pyrimidinecarboxyliques eventuellement 2-substitues | |
| WO2004050620A3 (en) | Derivatives of succinic and glutaric acids and analogs thereof useful as inhibitors of phex | |
| MX2008010884A (es) | Acidos 4-fenil-tiazol-5-carboxilicos y amidas de acidos 4-fenil-tiazol-5-carboxilicos como inhibidores de la plk1. | |
| EA200900797A1 (ru) | Способ синтеза производных 3-аминотетрагидрофуран-3-карбоновой кислоты и их применение в качестве лекарственных средств | |
| WO2009037137A3 (en) | Process from shikimic acid to oseltamivir phosphate | |
| ATE261953T1 (de) | Verfahren zur herstellung von citalopram | |
| ATE441627T1 (de) | Verfahren zur herstellung von valsartan | |
| BR0010225A (pt) | Composto de amida, processo para prepará-lo, composição farmacêutica compreendendo dito composto, método de tratamento e uso | |
| DE602005022326D1 (de) | Verfahren zur herstellung von 4,5-diamino-shikimisäure | |
| ATE289583T1 (de) | Stereoisomere von propyl-isopropylacetamid, verfahren zu deren herstellung sowie diese enthaltende pharmazeutische zubereitungen | |
| EP1390343A4 (de) | Neue retinoidderivate und verfahren zur herstellung dieser verbindungen, sowie eine pharmazeutische anti-krebs-zusammensetzung, die diese verbindungen enthält | |
| BRPI0513299A (pt) | processo para preparação de ésteres de ácido 4, 4-difluoro-3-oxobutanóico | |
| BRPI0516192A (pt) | composto, e, método para a preparação de um composto | |
| AR019197A1 (es) | COMPUESTOS DERIVADOS DE PIPERIDINA ANTIHISTAMINICOS, COMPUESTOS INTERMEDIOS, PROCEDIMIENTO DE PREPARACIoN DE DERIVADOS DE PIPERIDINA Y PROCEDIMIENTOS DE PREPARACIoN DE INTERMEDIARIOS. | |
| ATE399757T1 (de) | Neues verfahren zur herstellung von nitrooxyderivaten von paracetamol | |
| ATE555093T1 (de) | Verfahren zur herstellung einer (s)-1-alkyl-2i,6i-pipecoloxylididverbindung | |
| DE602004008486D1 (de) | Verfahren zur herstellung von (1s,4r)-cis-4-ä2-amino-6-chlor-9h-purin-9-ylü-2-cyclopenten-1-methanol | |
| EA200500716A1 (ru) | Новые соединения 2,3-дигидро-4-(1h)-пиридона, способ их получения и фармацевтические композиции, которые их содержат | |
| DE602004020050D1 (de) | Verfahren zur herstellung substituierter imidazolderivate und in dem verfahren verwendete zwischenprodukte | |
| ATE439333T1 (de) | Verfahren zur herstellung optisch aktiver propoxyanilinderivate | |
| DE602004030091D1 (de) | Verfahren zur reduktiven deshalogenierung | |
| DK1112999T3 (da) | Reduktion af azider til aminer ved hjælp af phosphiner |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
Ref document number: 1791808 Country of ref document: EP |