ATE511512T1 - Olanzapinpamoat-dihydrat - Google Patents
Olanzapinpamoat-dihydratInfo
- Publication number
- ATE511512T1 ATE511512T1 AT05855335T AT05855335T ATE511512T1 AT E511512 T1 ATE511512 T1 AT E511512T1 AT 05855335 T AT05855335 T AT 05855335T AT 05855335 T AT05855335 T AT 05855335T AT E511512 T1 ATE511512 T1 AT E511512T1
- Authority
- AT
- Austria
- Prior art keywords
- olanzapin
- pamoate dihydrate
- dihydrate
- pamoate
- schizophrenia
- Prior art date
Links
- 150000004683 dihydrates Chemical class 0.000 title 1
- KVWDHTXUZHCGIO-UHFFFAOYSA-N olanzapine Chemical compound C1CN(C)CCN1C1=NC2=CC=CC=C2NC2=C1C=C(C)S2 KVWDHTXUZHCGIO-UHFFFAOYSA-N 0.000 title 1
- 229960001072 olanzapine pamoate Drugs 0.000 abstract 1
- -1 olanzapine pamoate dihydrate Chemical class 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 208000020016 psychiatric disease Diseases 0.000 abstract 1
- 201000000980 schizophrenia Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US64169305P | 2005-01-05 | 2005-01-05 | |
| PCT/US2005/046752 WO2006073886A1 (en) | 2005-01-05 | 2005-12-22 | Olanzapine pamoate dihydrate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE511512T1 true ATE511512T1 (de) | 2011-06-15 |
Family
ID=36024754
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT05855335T ATE511512T1 (de) | 2005-01-05 | 2005-12-22 | Olanzapinpamoat-dihydrat |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US7932249B2 (de) |
| EP (1) | EP1838716B1 (de) |
| JP (1) | JP4940152B2 (de) |
| AT (1) | ATE511512T1 (de) |
| CY (1) | CY1111762T1 (de) |
| DK (1) | DK1838716T3 (de) |
| ES (1) | ES2363364T3 (de) |
| PL (1) | PL1838716T3 (de) |
| PT (1) | PT1838716E (de) |
| SI (1) | SI1838716T1 (de) |
| WO (1) | WO2006073886A1 (de) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6617321B2 (en) | 1997-09-30 | 2003-09-09 | Eli Lilly And Company | 2-methyl-thieno-benzodiazepine formulation |
| SI1838716T1 (sl) | 2005-01-05 | 2011-10-28 | Lilly Co Eli | Olanzapin pamoat dihidrat |
| WO2011091142A2 (en) * | 2010-01-20 | 2011-07-28 | Teva Pharmaceutical Industries Ltd. | Crystalline and amorphous forms of olanzapine pamoate |
| US9132136B2 (en) * | 2010-08-02 | 2015-09-15 | Hoffmann-La Roche Inc. | Pharmaceutical combination |
| EP2629775A4 (de) | 2010-10-18 | 2014-06-11 | Dainippon Sumitomo Pharma Co | Injizierbare formulierung mit verzögerter freisetzung |
| US20140206667A1 (en) | 2012-11-14 | 2014-07-24 | Michela Gallagher | Methods and compositions for treating schizophrenia |
| BR112020013750A8 (pt) | 2018-01-05 | 2022-10-18 | Impel Neuropharma Inc | Dispensação intranasal de olanzapina por dispositivo olfativo de precisão |
| TWI756536B (zh) * | 2019-04-12 | 2022-03-01 | 佳勝科技股份有限公司 | 改質液晶高分子的製作方法、液晶高分子組合物及改變液晶高分子之熔點的方法 |
Family Cites Families (47)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3354036A (en) | 1963-11-19 | 1967-11-21 | Du Pont | Method of producing depression |
| GB1343936A (en) | 1970-07-21 | 1974-01-16 | Endo Lab | Narcotic antagonist compositions having prolonged activity |
| US3676557A (en) | 1971-03-02 | 1972-07-11 | Endo Lab | Long-acting narcotic antagonist formulations |
| ES410734A1 (es) | 1973-01-18 | 1976-01-01 | Rocador Sa | Procedimiento para la obtencion del pamoato de butacaina. |
| US3895111A (en) | 1973-06-27 | 1975-07-15 | American Cyanamid Co | Asthma treatment by inhalation of micronized N,N-diethyl-4-methyl-1-piperazinecarboxamide pamoate |
| US4016273A (en) | 1975-07-16 | 1977-04-05 | American Cyanamid Company | Sustained release forms of certain oxazepines for parenteral administration |
| US4076942A (en) | 1975-10-01 | 1978-02-28 | Merck & Co., Inc. | Crystalline dipilocarpinium pamoate |
| GB1539277A (en) | 1977-09-16 | 1979-01-31 | Wyeth John & Brother Ltd | Hexahydro-1h-azepines |
| US4320124A (en) | 1980-10-17 | 1982-03-16 | Pfizer Inc. | Composition for enhancing binding of a benzodiazepine to central benzodiazepine receptors and use thereof |
| US4675189A (en) | 1980-11-18 | 1987-06-23 | Syntex (U.S.A.) Inc. | Microencapsulation of water soluble active polypeptides |
| US4906474A (en) | 1983-03-22 | 1990-03-06 | Massachusetts Institute Of Technology | Bioerodible polyanhydrides for controlled drug delivery |
| DE3324192A1 (de) | 1983-07-05 | 1985-01-17 | Troponwerke Gmbh & Co Kg | Depot-antiphlogistika |
| US4816247A (en) | 1985-09-11 | 1989-03-28 | American Cyanamid Company | Emulsion compositions for administration of sparingly water soluble ionizable hydrophobic drugs |
| US4784845A (en) | 1985-09-16 | 1988-11-15 | American Cyanamid Company | Emulsion compostions for the parenteral administration of sparingly water soluble ionizable hydrophobic drugs |
| GB2209937B (en) | 1987-09-21 | 1991-07-03 | Depiopharm S A | Water insoluble polypeptides |
| US5292760A (en) | 1987-12-07 | 1994-03-08 | Hoechst-Roussel Pharmaceuticals Inc. | 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines |
| JPH01284333A (ja) | 1988-05-11 | 1989-11-15 | T Hasegawa Co Ltd | 乳化液組成物 |
| GB8819059D0 (en) | 1988-08-11 | 1988-09-14 | Lilly Industries Ltd | Benzodiazepine compounds & their use as pharmaceuticals |
| PH30995A (en) | 1989-07-07 | 1997-12-23 | Novartis Inc | Sustained release formulations of water soluble peptides. |
| US5439688A (en) | 1989-07-28 | 1995-08-08 | Debio Recherche Pharmaceutique S.A. | Process for preparing a pharmaceutical composition |
| GB9009229D0 (en) | 1990-04-25 | 1990-06-20 | Lilly Industries Ltd | Pharmaceutical compounds |
| US5229382A (en) | 1990-04-25 | 1993-07-20 | Lilly Industries Limited | 2-methyl-thieno-benzodiazepine |
| FR2663224B1 (fr) | 1990-06-14 | 1995-01-20 | Applicationes Farmaceuticas Sa | Forme galenique parenterale. |
| US5605897A (en) | 1991-04-23 | 1997-02-25 | Eli Lilly And Company | 2-methyl-thieno-benzodiazepine |
| EP0569096A1 (de) | 1992-05-08 | 1993-11-10 | Akzo Nobel N.V. | Depotpräparat |
| DE69327542T2 (de) | 1992-11-17 | 2000-07-06 | Yoshitomi Pharmaceutical Industries, Ltd. | Ein antipsychotikum enthaltende mikrokugel zur verzögerten freisetzung und verfahren für ihre herstellung |
| TW376319B (en) | 1993-04-28 | 1999-12-11 | Janssen Pharmaceutica Nv | Pharmaceutical composition containing risperidone pamoate and having a long acting activity for treating psychoses induced by the release of dopamine |
| CA2178592C (en) | 1993-12-09 | 2009-07-28 | Zentaris Gmbh | Long-acting injection suspensions and a process for their preparation |
| JP3701693B2 (ja) | 1993-12-28 | 2005-10-05 | 日本製薬株式会社 | 鎮痛薬含有注射用徐放性脂肪乳剤 |
| US6333021B1 (en) | 1994-11-22 | 2001-12-25 | Bracco Research S.A. | Microcapsules, method of making and their use |
| EG23659A (en) | 1995-03-24 | 2007-03-26 | Lilly Co Eli | Process and crystal forms of methyl-thieno-benzodiazepine |
| EG24221A (en) | 1995-03-24 | 2008-11-10 | Lilly Co Eli | Process for preparing olanzapine |
| CR5278A (es) | 1995-03-24 | 1996-07-04 | Lilly Co Eli | Formulacion oral de 2-metil-tieno-benzodiacepina |
| US5776928A (en) | 1995-04-21 | 1998-07-07 | Eli Lilly And Company | Method for treating dyskinesias with olanzapine |
| JPH11506096A (ja) | 1995-05-30 | 1999-06-02 | イーライ・リリー・アンド・カンパニー | 認識機能不全を処置する方法 |
| AU5872596A (en) | 1995-06-01 | 1996-12-18 | Eli Lilly And Company | Method for treating anorexia |
| US5693336A (en) | 1995-06-07 | 1997-12-02 | Nexstar Pharmaceuticals, Inc. | Blood stable liposomal cyclosporin formulations |
| US5891461A (en) | 1995-09-14 | 1999-04-06 | Cygnus, Inc. | Transdermal administration of olanzapine |
| US5736152A (en) | 1995-10-27 | 1998-04-07 | Atrix Laboratories, Inc. | Non-polymeric sustained release delivery system |
| JPH09157159A (ja) | 1995-12-11 | 1997-06-17 | Lion Corp | カロチノイド含有組成物 |
| JP2001500878A (ja) | 1996-09-23 | 2001-01-23 | イーライ・リリー・アンド・カンパニー | オランザピン二水和物d |
| US6617321B2 (en) | 1997-09-30 | 2003-09-09 | Eli Lilly And Company | 2-methyl-thieno-benzodiazepine formulation |
| US6169084B1 (en) * | 1997-09-30 | 2001-01-02 | Eli Lilly And Company | 2-methyl-thieno-benzodiazepine formulation |
| HK1041199B (en) * | 1998-09-30 | 2005-03-18 | Eli Lilly & Company | 2-Methyl-thiophenone-benzodiazine formula |
| SK2502003A3 (en) * | 2000-08-31 | 2004-03-02 | Reddys Lab Ltd Dr | Process for preparation of hydrates of olanzapine and their conversion into crystalline forms of olanzapine |
| CA2464306A1 (en) * | 2001-10-29 | 2003-05-08 | Dr. Reddy's Laboratories Ltd. | Olanzapine dihydrate-ii a process for its preparation and use thereof |
| SI1838716T1 (sl) | 2005-01-05 | 2011-10-28 | Lilly Co Eli | Olanzapin pamoat dihidrat |
-
2005
- 2005-12-22 SI SI200531351T patent/SI1838716T1/sl unknown
- 2005-12-22 EP EP05855335A patent/EP1838716B1/de not_active Expired - Lifetime
- 2005-12-22 AT AT05855335T patent/ATE511512T1/de active
- 2005-12-22 JP JP2007549505A patent/JP4940152B2/ja not_active Expired - Fee Related
- 2005-12-22 PL PL05855335T patent/PL1838716T3/pl unknown
- 2005-12-22 ES ES05855335T patent/ES2363364T3/es not_active Expired - Lifetime
- 2005-12-22 US US11/722,228 patent/US7932249B2/en active Active
- 2005-12-22 PT PT05855335T patent/PT1838716E/pt unknown
- 2005-12-22 WO PCT/US2005/046752 patent/WO2006073886A1/en not_active Ceased
- 2005-12-22 DK DK05855335.5T patent/DK1838716T3/da active
-
2011
- 2011-08-18 CY CY20111100789T patent/CY1111762T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1838716B1 (de) | 2011-06-01 |
| EP1838716A1 (de) | 2007-10-03 |
| PT1838716E (pt) | 2011-07-15 |
| ES2363364T3 (es) | 2011-08-02 |
| JP2008526748A (ja) | 2008-07-24 |
| CY1111762T1 (el) | 2015-10-07 |
| SI1838716T1 (sl) | 2011-10-28 |
| US20080096871A1 (en) | 2008-04-24 |
| JP4940152B2 (ja) | 2012-05-30 |
| DK1838716T3 (da) | 2011-07-25 |
| WO2006073886A1 (en) | 2006-07-13 |
| US7932249B2 (en) | 2011-04-26 |
| PL1838716T3 (pl) | 2011-09-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
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