AU2001237447A1 - Method for preparing pyrimidone derivatives with antifungal activity - Google Patents

Method for preparing pyrimidone derivatives with antifungal activity

Info

Publication number
AU2001237447A1
AU2001237447A1 AU2001237447A AU3744701A AU2001237447A1 AU 2001237447 A1 AU2001237447 A1 AU 2001237447A1 AU 2001237447 A AU2001237447 A AU 2001237447A AU 3744701 A AU3744701 A AU 3744701A AU 2001237447 A1 AU2001237447 A1 AU 2001237447A1
Authority
AU
Australia
Prior art keywords
antifungal activity
pyrimidone derivatives
preparing
preparing pyrimidone
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001237447A
Other languages
English (en)
Inventor
Manuel Anguita Lopez
Javier Bartroli Orpi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Noucor Health SA
Original Assignee
J Uriach y Cia SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by J Uriach y Cia SA filed Critical J Uriach y Cia SA
Publication of AU2001237447A1 publication Critical patent/AU2001237447A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2001237447A 2000-03-07 2001-03-05 Method for preparing pyrimidone derivatives with antifungal activity Abandoned AU2001237447A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ES200000625A ES2159488B1 (es) 2000-03-07 2000-03-07 Procedimiento para la preparacion de derivados de pirimidona con actividad antifungica.
ES200000625 2000-03-07
PCT/ES2001/000081 WO2001066519A2 (fr) 2000-03-07 2001-03-05 Procede de preparation de derives de pyrimidone a activite antifongique

Publications (1)

Publication Number Publication Date
AU2001237447A1 true AU2001237447A1 (en) 2001-09-17

Family

ID=8492714

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001237447A Abandoned AU2001237447A1 (en) 2000-03-07 2001-03-05 Method for preparing pyrimidone derivatives with antifungal activity

Country Status (17)

Country Link
US (1) US6653475B2 (fr)
EP (1) EP1282084B9 (fr)
JP (1) JP4772248B2 (fr)
KR (1) KR100735583B1 (fr)
AR (1) AR027607A1 (fr)
AT (1) ATE250256T1 (fr)
AU (1) AU2001237447A1 (fr)
BR (1) BRPI0108990B8 (fr)
CA (1) CA2402390C (fr)
DE (1) DE60100810T2 (fr)
DK (1) DK1282084T3 (fr)
ES (2) ES2159488B1 (fr)
HK (1) HK1052244B (fr)
MX (1) MXPA02008556A (fr)
NO (1) NO323314B1 (fr)
PT (1) PT1282084E (fr)
WO (1) WO2001066519A2 (fr)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7230000B1 (en) 1999-10-27 2007-06-12 Cytokinetics, Incorporated Methods and compositions utilizing quinazolinones
US6545004B1 (en) 1999-10-27 2003-04-08 Cytokinetics, Inc. Methods and compositions utilizing quinazolinones
EP1477481B1 (fr) * 2002-01-28 2009-07-22 Ube Industries, Ltd. Procede de production de derive de quinazolin-4-one
US7009049B2 (en) 2002-02-15 2006-03-07 Cytokinetics, Inc. Syntheses of quinazolinones
AU2003270015A1 (en) 2002-05-09 2003-12-02 Cytokinetics, Inc. Compounds, compositions, and methods
US7166595B2 (en) 2002-05-09 2007-01-23 Cytokinetics, Inc. Compounds, methods and compositions
WO2003103575A2 (fr) 2002-05-23 2003-12-18 Cytokinetics, Inc. Composes, compositions et procedes
CA2489367A1 (fr) 2002-06-14 2003-12-24 Cytokinetics, Inc. Composes, compositions et procedes
WO2004009036A2 (fr) 2002-07-23 2004-01-29 Cytokinetics, Inc. Composes, compositions et procedes
WO2004034972A2 (fr) 2002-09-30 2004-04-29 Cytokinetics, Inc. Composes, compositions, et procedes
EP1692112A4 (fr) 2003-12-08 2008-09-24 Cytokinetics Inc Composes, compositions, et methodes associees
JP5055263B2 (ja) 2005-03-30 2012-10-24 ダエウン ファーマシューティカル カンパニー リミテッド 抗真菌性トリアゾール誘導体
EP2049504A4 (fr) * 2006-08-07 2010-09-22 Stiefel Laboratories Composés cristallins antifongiques
EP2009009A1 (fr) * 2007-06-26 2008-12-31 Palau Pharma, S.A. Composés antifongiques cristallins
EP1887004A1 (fr) * 2006-08-07 2008-02-13 Palau Pharma, S.A. Formes cristallines de (1R,2R)-7-Chloro-3-[2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]quinazolin-4(3H)-one
TWI395728B (zh) 2006-12-06 2013-05-11 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
TWI415827B (zh) 2006-12-21 2013-11-21 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
EP2257555B1 (fr) 2008-03-03 2012-07-04 National Chemical Laboratory Composés de thiéno[2,3-d]-pyrimidin-4(3h)-one dotés de propriétés antifongiques et procédé associé
SE532624C2 (sv) * 2008-06-19 2010-03-09 Andritz Technology And Asset Management Gmbh Kylning av en cellulosamassabana
WO2012123952A1 (fr) * 2011-03-15 2012-09-20 Fdc Limited Énantiomères d'analogues de fluconazole contenant une fraction thiéno-[2,3-d]pyrimidin-4(3h)-one en tant qu'agents antifongiques
CN106588889B (zh) * 2016-11-25 2019-01-22 江苏恒盛药业有限公司 一种伏立康唑的制备方法
CN111018839B (zh) * 2019-12-02 2022-12-23 中国人民解放军第二军医大学 三氮唑醇类衍生物及其制备方法和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8819308D0 (en) * 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents
TW218017B (fr) * 1992-04-28 1993-12-21 Takeda Pharm Industry Co Ltd
MX9702382A (es) * 1995-08-02 1998-02-28 Uriach & Cia Sa J Nuevos derivados de pirimidona con actividad antifungica.

Also Published As

Publication number Publication date
HK1052244A1 (en) 2003-09-05
KR100735583B1 (ko) 2007-07-04
US6653475B2 (en) 2003-11-25
EP1282084B9 (fr) 2005-03-02
ATE250256T1 (de) 2003-10-15
AR027607A1 (es) 2003-04-02
CA2402390A1 (fr) 2001-09-13
NO20024256D0 (no) 2002-09-06
WO2001066519A2 (fr) 2001-09-13
BR0108990B1 (pt) 2014-03-25
EP1282084B1 (fr) 2003-09-17
CA2402390C (fr) 2009-09-15
DK1282084T3 (da) 2004-02-02
ES2207605T3 (es) 2004-06-01
NO323314B1 (no) 2007-03-12
DE60100810D1 (de) 2003-10-23
DE60100810T2 (de) 2004-07-01
ES2159488A1 (es) 2001-10-01
BR0108990A (pt) 2003-12-30
JP2004500391A (ja) 2004-01-08
WO2001066519A3 (fr) 2002-01-31
EP1282084A2 (fr) 2003-02-05
JP4772248B2 (ja) 2011-09-14
BRPI0108990B8 (pt) 2021-05-25
ES2159488B1 (es) 2002-04-16
KR20020075809A (ko) 2002-10-05
NO20024256L (no) 2002-09-06
PT1282084E (pt) 2004-02-27
HK1052244B (en) 2003-12-19
US20030064986A1 (en) 2003-04-03
MXPA02008556A (es) 2003-02-24

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