AU2014352875B2 - Gastrin antagonists (eg YF476, netazepide) for treatment and prevention of osteoporosis - Google Patents

Gastrin antagonists (eg YF476, netazepide) for treatment and prevention of osteoporosis Download PDF

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Publication number
AU2014352875B2
AU2014352875B2 AU2014352875A AU2014352875A AU2014352875B2 AU 2014352875 B2 AU2014352875 B2 AU 2014352875B2 AU 2014352875 A AU2014352875 A AU 2014352875A AU 2014352875 A AU2014352875 A AU 2014352875A AU 2014352875 B2 AU2014352875 B2 AU 2014352875B2
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gastrin
bone
animals
ovx
ovariectomy
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AU2014352875A8 (en
AU2014352875A1 (en
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Mark Kidd
Irvin Mark MODLIN
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CL Biosciences LLC
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CL Biosciences LLC
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2014352875A 2013-11-22 2014-11-21 Gastrin antagonists (eg YF476, netazepide) for treatment and prevention of osteoporosis Active AU2014352875B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361907980P 2013-11-22 2013-11-22
US61/907,980 2013-11-22
PCT/US2014/066832 WO2015077572A1 (en) 2013-11-22 2014-11-21 Gastrin antagonists (eg yf476, netazepide) for treatment and prevention of osteoporosis

Publications (3)

Publication Number Publication Date
AU2014352875A1 AU2014352875A1 (en) 2016-05-26
AU2014352875A8 AU2014352875A8 (en) 2016-06-30
AU2014352875B2 true AU2014352875B2 (en) 2019-10-24

Family

ID=52118000

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2014352875A Active AU2014352875B2 (en) 2013-11-22 2014-11-21 Gastrin antagonists (eg YF476, netazepide) for treatment and prevention of osteoporosis

Country Status (14)

Country Link
US (1) US10709714B2 (2)
EP (1) EP3071206B1 (2)
JP (1) JP6502939B2 (2)
KR (1) KR102254957B1 (2)
CN (1) CN106163527A (2)
AU (1) AU2014352875B2 (2)
BR (1) BR112016011727A2 (2)
CA (1) CA2929858C (2)
DK (1) DK3071206T3 (2)
ES (1) ES2870538T3 (2)
MX (1) MX2016006657A (2)
PL (1) PL3071206T3 (2)
RU (1) RU2693484C1 (2)
WO (1) WO2015077572A1 (2)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10881667B2 (en) 2018-10-30 2021-01-05 City University Of Hong Kong Method and composition for treating epilepsy
US11285161B2 (en) 2019-04-26 2022-03-29 City University Of Hong Kong Method and composition for treating mental disorder and pain associated with nerve damage
CN110935005A (zh) * 2019-11-19 2020-03-31 宁波大学 一种丙谷二肽的新用途
CN115770266B (zh) * 2023-01-30 2023-05-09 云南中医药大学 一种用于治疗绝经后骨质疏松的药物组合物

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WO2005007107A2 (en) * 2003-07-11 2005-01-27 University Of Massachusetts Histamine and cck2/gastrin receptor blockade in the treatment of acid-peptic disease and cancer

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Also Published As

Publication number Publication date
BR112016011727A2 (pt) 2017-08-08
JP2016538295A (ja) 2016-12-08
EP3071206A1 (en) 2016-09-28
RU2016124538A (ru) 2017-12-27
CA2929858A1 (en) 2015-05-28
KR102254957B1 (ko) 2021-05-25
WO2015077572A1 (en) 2015-05-28
JP6502939B2 (ja) 2019-04-17
EP3071206B1 (en) 2021-02-17
US20150148339A1 (en) 2015-05-28
RU2693484C1 (ru) 2019-07-03
DK3071206T3 (da) 2021-05-25
AU2014352875A8 (en) 2016-06-30
US10709714B2 (en) 2020-07-14
PL3071206T3 (pl) 2022-01-17
CA2929858C (en) 2022-03-29
AU2014352875A1 (en) 2016-05-26
ES2870538T3 (es) 2021-10-27
KR20160088891A (ko) 2016-07-26
CN106163527A (zh) 2016-11-23
MX2016006657A (es) 2016-10-12

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