BE775610Q - Derives amides d'acides halogeno et nitro benzoiques et leur preparation - Google Patents

Derives amides d'acides halogeno et nitro benzoiques et leur preparation

Info

Publication number
BE775610Q
BE775610Q BE775610A BE775610A BE775610Q BE 775610 Q BE775610 Q BE 775610Q BE 775610 A BE775610 A BE 775610A BE 775610 A BE775610 A BE 775610A BE 775610 Q BE775610 Q BE 775610Q
Authority
BE
Belgium
Prior art keywords
emi
benzamidoalkylpiperazine
derivs
halogen
acid chloride
Prior art date
Application number
BE775610A
Other languages
English (en)
Inventor
R Eche
J De Antoni
Original Assignee
Bruneau & Cie Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bruneau & Cie Lab filed Critical Bruneau & Cie Lab
Application granted granted Critical
Publication of BE775610Q publication Critical patent/BE775610Q/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Description


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 <EMI ID=4.1>   <EMI ID=5.1> 
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dans laquelle 

  
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nant pas plus de trois atones de carbone ou un

  
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du sulfate de sodium., le chloroforme est ensuite évaporé sous -

  
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 <EMI ID=28.1>  <EMI ID=29.1>  <EMI ID=30.1> 
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 <EMI ID=32.1> 
 Les exemples suivants., non limitatifs, illutrent ces préparations. 

  
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nutes, avec agitation, une solution de 15,8 g de chlorure d'aci-

  
 <EMI ID=34.1> 

  
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agite pendant 15 heures à la température ambiante , le produit

  
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posé basique en solution dans l'Sthanol par un équivalent d'acide chlorhydrique en solution dans le même alcool. Son point de

  
 <EMI ID=39.1> 

  
Procédé b 

  
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,Les composes correspondants sont consignes dans le tableau suivent : 

  
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dans les mêmes conditions que sous a). Les. constantes du pro-  duit obtenu sont les suivantes : 

  
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Claims (1)

  1. <EMI ID=65.1>
    <EMI ID=66.1>
    <EMI ID=67.1>
    <EMI ID=68.1>
    chlore, et peut exister.. plusieurs fois sur le
    <EMI ID=69.1>
    <EMI ID=70.1>
    <EMI ID=71.1> <EMI ID=72.1> <EMI ID=73.1>
    <EMI ID=74.1> <EMI ID=75.1>
    <EMI ID=76.1>
    <EMI ID=77.1>
    <EMI ID=78.1>
    <EMI ID=79.1>
BE775610A 1967-07-19 1971-11-19 Derives amides d'acides halogeno et nitro benzoiques et leur preparation BE775610Q (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR114791A FR1537901A (fr) 1967-07-19 1967-07-19 Dérivés amidés d'acides halogéno et nitro benzoïques et leur préparation
FR135764A FR93884E (fr) 1967-07-19 1968-01-12 Dérivés amidés d'acides halogéno et nitro benzoiques et leur préparation.

Publications (1)

Publication Number Publication Date
BE775610Q true BE775610Q (fr) 1972-03-16

Family

ID=32929144

Family Applications (1)

Application Number Title Priority Date Filing Date
BE775610A BE775610Q (fr) 1967-07-19 1971-11-19 Derives amides d'acides halogeno et nitro benzoiques et leur preparation

Country Status (2)

Country Link
BE (1) BE775610Q (fr)
FR (2) FR1537901A (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0104614A1 (fr) * 1982-09-24 1984-04-04 Chugai Seiyaku Kabushiki Kaisha Dérivés du phénylpipérazine et leur procédé de préparation

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3846430A (en) * 1968-01-12 1974-11-05 Bruneau & Cie Lab 1-(2-methoxy-phenyl)-4-{8 2-(4-fluoro-benzamido)-ethyl{9 -piperazine
IE911774A1 (en) * 1990-06-11 1991-12-18 Akzo Nv Pyridinylpiperazine derivatives
SE9201138D0 (sv) * 1992-04-09 1992-04-09 Astra Ab Novel phthalimidoalkylpiperazines
IT1266582B1 (it) * 1993-07-30 1997-01-09 Recordati Chem Pharm Derivati (di)azacicloesanici e diazacicloeptanici
US5659033A (en) * 1995-09-13 1997-08-19 Neurogen Corporation N-aminoalkylfluorenecarboxamides; a new class of dopamine receptor subtype specific ligands

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0104614A1 (fr) * 1982-09-24 1984-04-04 Chugai Seiyaku Kabushiki Kaisha Dérivés du phénylpipérazine et leur procédé de préparation

Also Published As

Publication number Publication date
FR1537901A (fr) 1968-08-30
FR93884E (fr) 1969-05-30

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