BE827451A - Indoles substitues et procede pour les preparer - Google Patents

Indoles substitues et procede pour les preparer

Info

Publication number
BE827451A
BE827451A BE1006567A BE1006567A BE827451A BE 827451 A BE827451 A BE 827451A BE 1006567 A BE1006567 A BE 1006567A BE 1006567 A BE1006567 A BE 1006567A BE 827451 A BE827451 A BE 827451A
Authority
BE
Belgium
Prior art keywords
indoles
substitutes
preparing
substitutes indoles
Prior art date
Application number
BE1006567A
Other languages
English (en)
Inventor
J J Plattner
C A Harbert
J R Tretter
W M Welch
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE827451A publication Critical patent/BE827451A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE1006567A 1974-04-01 1975-04-01 Indoles substitues et procede pour les preparer BE827451A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US45664074A 1974-04-01 1974-04-01

Publications (1)

Publication Number Publication Date
BE827451A true BE827451A (fr) 1975-10-01

Family

ID=23813560

Family Applications (1)

Application Number Title Priority Date Filing Date
BE1006567A BE827451A (fr) 1974-04-01 1975-04-01 Indoles substitues et procede pour les preparer

Country Status (6)

Country Link
JP (3) JPS5874683A (fr)
BE (1) BE827451A (fr)
CA (1) CA1056381A (fr)
GB (1) GB1476087A (fr)
IE (1) IE41352B1 (fr)
ZA (1) ZA751990B (fr)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2004063818A (ja) 2002-07-30 2004-02-26 Oki Electric Ind Co Ltd フレキシブルチューブを利用した半導体装置の製造方法
EP2560676B8 (fr) 2010-04-22 2016-10-12 Intra-Cellular Therapies, Inc. Composés organiques
WO2013155504A1 (fr) 2012-04-14 2013-10-17 Intra-Cellular Therapies, Inc. Nouveaux procédés
HUE053159T2 (hu) 2013-03-15 2021-06-28 Intra Cellular Therapies Inc Szerves vegyületek
IL305990B2 (en) 2013-12-03 2025-12-01 Intra Cellular Therapies Inc Long-acting injectable composition comprising polymeric microspheres of heterocycle fused gamma-carboline compounds or a pharmaceutical composition for sustained or delayed release comprising the compounds and their use in the treatment of bipolar disorder i and/or bipolar ii disorder
MX365969B (es) 2014-04-04 2019-06-21 Intra Cellular Therapies Inc Gamma-carbolinas fusionadas con heterociclos sustituidas con deuterio.
RU2016143091A (ru) 2014-04-04 2018-05-08 Интра-Селлулар Терапиз, Инк. Органические соединения
CN108883111B (zh) 2016-01-26 2021-10-08 细胞内治疗公司 有机化合物
PL3407889T3 (pl) 2016-03-25 2021-11-22 Intra-Cellular Therapies, Inc. Związki organiczne i ich zastosowanie w leczeniu lub zapobieganiu zaburzeniom ośrodkowego układu nerwowego
EP3436083A4 (fr) 2016-03-28 2019-11-27 Intra-Cellular Therapies, Inc. Nouvelles compositions et méthodes
US11331316B2 (en) 2016-10-12 2022-05-17 Intra-Cellular Therapies, Inc. Amorphous solid dispersions
US10906906B2 (en) 2016-12-29 2021-02-02 Intra-Cellular Therapies, Inc. Organic compounds
US10961245B2 (en) 2016-12-29 2021-03-30 Intra-Cellular Therapies, Inc. Substituted heterocycle fused gamma-carbolines for treatment of central nervous system disorders
IL268970B2 (en) 2017-03-24 2023-12-01 Intra Cellular Therapies Inc Oral transmucosal formulations of substituted heterocycle fused gamma carbolines
JP7224333B2 (ja) 2017-07-26 2023-02-17 イントラ-セルラー・セラピーズ・インコーポレイテッド 有機化合物
JP7223742B2 (ja) 2017-07-26 2023-02-16 イントラ-セルラー・セラピーズ・インコーポレイテッド 有機化合物
WO2019178484A1 (fr) 2018-03-16 2019-09-19 Intra-Cellular Therapies, Inc. Nouveaux procédés
AU2019240226B2 (en) 2018-03-23 2024-11-28 Intra-Cellular Therapies, Inc. Organic compounds
WO2019237037A1 (fr) 2018-06-08 2019-12-12 Intra-Cellular Therapies, Inc. Nouvelles méthodes
CA3106447A1 (fr) 2018-06-11 2019-12-19 Intra-Cellular Therapies, Inc. Synthese de gamma-carbolines fusionnees a heterocycles substitues
EP3843729A4 (fr) 2018-08-29 2022-06-01 Intra-Cellular Therapies, Inc. Nouvelles compositions et méthodes
CA3108558A1 (fr) 2018-08-31 2020-03-05 Intra-Cellular Therapies, Inc. Nouvelles methodes
CN112584837A (zh) 2018-08-31 2021-03-30 细胞内治疗公司 新方法
IL283963B2 (en) 2018-12-17 2025-01-01 Intra Cellular Therapies Inc Synthesis of condensed gamma-carbolines and converted heterocycles
EP3898580A4 (fr) 2018-12-17 2022-08-10 Intra-Cellular Therapies, Inc. Synthèse de gamma-carbolines fusionnées à hétérocycles substitués
US12195463B2 (en) 2018-12-21 2025-01-14 Intra-Cellular Therapies, Inc. Organic compounds
JP7673040B2 (ja) 2019-07-07 2025-05-08 イントラ-セルラー・セラピーズ・インコーポレイテッド 新規方法
US12414948B2 (en) 2022-05-18 2025-09-16 Intra-Cellular Therapies, Inc. Methods
CN116425670A (zh) * 2022-07-15 2023-07-14 英矽智能科技(上海)有限公司 作为tead抑制剂的新型杂环化合物

Also Published As

Publication number Publication date
GB1476087A (en) 1977-06-10
JPS5874681A (ja) 1983-05-06
JPS5915911B2 (ja) 1984-04-12
CA1056381A (fr) 1979-06-12
IE41352L (en) 1975-10-01
JPS5874682A (ja) 1983-05-06
ZA751990B (en) 1976-02-25
JPS5874683A (ja) 1983-05-06
IE41352B1 (en) 1979-12-19

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: PFIZER INC.

Effective date: 19840401