BE836528A - Nouveaux derives d'acide 3-amino- indazolecarboxylique - Google Patents

Nouveaux derives d'acide 3-amino- indazolecarboxylique

Info

Publication number
BE836528A
BE836528A BE162651A BE162651A BE836528A BE 836528 A BE836528 A BE 836528A BE 162651 A BE162651 A BE 162651A BE 162651 A BE162651 A BE 162651A BE 836528 A BE836528 A BE 836528A
Authority
BE
Belgium
Prior art keywords
amino
new derivatives
indazolecarboxylic acid
indazolecarboxylic
acid
Prior art date
Application number
BE162651A
Other languages
English (en)
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE836528A publication Critical patent/BE836528A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
BE162651A 1974-12-13 1975-12-11 Nouveaux derives d'acide 3-amino- indazolecarboxylique BE836528A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
BE836528A true BE836528A (fr) 1976-06-11

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
BE162651A BE836528A (fr) 1974-12-13 1975-12-11 Nouveaux derives d'acide 3-amino- indazolecarboxylique

Country Status (27)

Country Link
US (1) US4051252A (2)
JP (1) JPS5182266A (2)
AT (1) AT343653B (2)
BE (1) BE836528A (2)
CA (1) CA1059523A (2)
CH (1) CH622250A5 (2)
CS (1) CS189731B2 (2)
DD (1) DD125484A5 (2)
DE (1) DE2458965C3 (2)
DK (1) DK137082C (2)
ES (1) ES443429A1 (2)
FI (1) FI753493A7 (2)
FR (1) FR2293928A1 (2)
GB (1) GB1490306A (2)
HK (1) HK52580A (2)
HU (1) HU173557B (2)
IE (1) IE42208B1 (2)
IL (1) IL48642A (2)
KE (1) KE3078A (2)
LU (1) LU73993A1 (2)
NL (1) NL7514521A (2)
NO (1) NO145382C (2)
PL (1) PL99858B1 (2)
SE (1) SE419645B (2)
SU (1) SU604487A3 (2)
YU (1) YU315275A (2)
ZA (1) ZA757777B (2)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
CN1926132B (zh) * 2000-09-15 2010-12-29 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的吡唑化合物
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
EP1317450B1 (en) * 2000-09-15 2006-11-22 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
NZ526472A (en) 2000-12-21 2004-04-30 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
WO2003028720A1 (en) 2001-09-26 2003-04-10 Pharmacia Italia S.P.A. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
EP1472245A2 (en) * 2002-02-06 2004-11-03 Vertex Pharmaceuticals Incorporated Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
AU2003218215A1 (en) 2002-03-15 2003-09-29 Vertex Pharmaceuticals, Inc. Azolylaminoazines as inhibitors of protein kinases
JP4751063B2 (ja) 2002-05-17 2011-08-17 ファイザー イタリア ソシエタ ア レスポンサビリタ リミタータ キナーゼ阻害剤として活性のアミノインダゾール誘導体、それらの調製方法、及びそれらを含む薬学的組成物
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
DK1532145T3 (da) 2002-08-02 2007-01-15 Vertex Pharma Pyrazolpræparater der er anvendelige som inhibitorer af GSK-3
JP2006512313A (ja) * 2002-10-31 2006-04-13 アムジェン インコーポレイテッド 抗炎症剤
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
AU2004297235A1 (en) * 2003-12-04 2005-06-23 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
AU2006279376B2 (en) 2005-08-18 2011-04-14 Vertex Pharmaceuticals Incoporated Pyrazine kinase inhibitors
EP1954277B1 (en) * 2005-11-03 2017-01-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
BRPI0709963A2 (pt) * 2006-04-14 2011-08-02 Abbott Lab processo para a preparação de indazolil uréias que inibem receptores de subtipo 1 de vanilóide (vr1)
MX2009004807A (es) 2006-11-02 2009-06-15 Vertex Pharma Aminopiridinas y aminopirimidinas utiles como inhibidores de proteina cinasa.
NZ577768A (en) 2006-12-19 2012-01-12 Vertex Pharma Aminopyrimidines useful as inhibitors of protein kinases
ATE526328T1 (de) 2007-03-09 2011-10-15 Vertex Pharma Als inhibitoren von proteinkinasen geeignete aminopyrimidine
MX2009009592A (es) 2007-03-09 2009-11-10 Vertex Pharma Aminopiridinas utiles como inhibidores de proteinas cinasas.
MX2009009590A (es) 2007-03-09 2009-11-10 Vertex Pharma Aminopirimidinas utiles como inhibidores de proteinas cinasas.
AU2008240313A1 (en) 2007-04-13 2008-10-23 Aj Park Aminopyrimidines useful as kinase inhibitors
JP5389786B2 (ja) 2007-05-02 2014-01-15 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害として有用なアミノピリミジン
CN101679387A (zh) * 2007-05-02 2010-03-24 沃泰克斯药物股份有限公司 可用作激酶抑制剂的氨基嘧啶类化合物
AU2008247592A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
MX2009012719A (es) * 2007-05-24 2010-02-04 Vertex Pharma Tiazoles y pirazoles utiles como inhibidores de cinasa.
CN101790532B (zh) * 2007-07-31 2013-11-20 沃泰克斯药物股份有限公司 5-氟-1H-吡唑并[3,4-b]吡啶-3-胺及其衍生物的制备方法
WO2010027921A1 (en) * 2008-09-03 2010-03-11 Vertex Pharmaceuticals Incorporated Co-crystals and pharmaceutical formulations comprising the same
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
WO2014017936A2 (en) 2012-07-24 2014-01-30 Bial- Portela & Ca, S.A. Urea compounds and their use as enzyme inhibitors
WO2014017938A2 (en) * 2012-07-27 2014-01-30 BIAL - PORTELA & Cª, S.A. Process for the synthesis of substituted urea compounds
AU2014293731B2 (en) 2013-07-24 2018-03-08 Bial - Portela & Ca, S.A. Imidazolecarboxamides and their use as FAAH inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (2) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
DE2458965A1 (de) 1976-06-16
KE3078A (en) 1980-10-03
AT343653B (de) 1978-06-12
SE419645B (sv) 1981-08-17
FR2293928B1 (2) 1979-09-21
PL99858B1 (pl) 1978-08-31
JPS5182266A (en) 1976-07-19
DE2458965C3 (de) 1979-10-11
GB1490306A (en) 1977-11-02
FR2293928A1 (fr) 1976-07-09
ATA939775A (de) 1977-10-15
IL48642A0 (en) 1976-02-29
ZA757777B (en) 1976-11-24
AU8717075A (en) 1977-06-09
SU604487A3 (ru) 1978-04-25
HU173557B (hu) 1979-06-28
YU315275A (en) 1982-02-28
CA1059523A (en) 1979-07-31
FI753493A7 (2) 1976-06-14
DE2458965B2 (de) 1979-02-22
DK137082C (da) 1978-06-19
DK137082B (da) 1978-01-16
IE42208L (en) 1976-06-13
ES443429A1 (es) 1977-04-16
HK52580A (en) 1980-09-26
LU73993A1 (2) 1976-11-11
CH622250A5 (2) 1981-03-31
US4051252A (en) 1977-09-27
NO754024L (2) 1976-06-15
SE7513990L (sv) 1976-06-14
DK567275A (da) 1976-06-14
NO145382C (no) 1982-03-10
DD125484A5 (2) 1977-04-20
NL7514521A (nl) 1976-06-15
NO145382B (no) 1981-11-30
IL48642A (en) 1979-12-30
CS189731B2 (en) 1979-04-30
IE42208B1 (en) 1980-06-18

Similar Documents

Publication Publication Date Title
BE836528A (fr) Nouveaux derives d'acide 3-amino- indazolecarboxylique
BE851306A (fr) Nouveaux derives de l'acide 3-quinoleine carboxylique
FR2316942A1 (fr) Derives halo-substitues d'acide 1-(alcoyl) inferieur -5-aroylpyrrole-2-acetique
BE827255A (fr) Nouveaux derives de l'amino-3 dihydrothiophenone-2
BE782366A (fr) Nouveaux derives de l'acide cephalosporanique
BE835268A (fr) Derives de l'acide furannehydroxyamique
BE819640A (fr) Nouveaux derives de l'acide phenylbenzoique
BE859846A (fr) Nouveaux derives d'acide alpha-thio-alcanoique
BE809903A (fr) Nouveaux esters o-ethyl-s-n-propyl-o-vinyliques d'acide thionothiolphosphorique
BE822729A (fr) Nouveaux derives de l'acide lysergique
BE821557A (fr) Nouveaux derives de l'acide indane-5-acetique
FR2273806A1 (fr) Derives d'acide barbiturique
BE848023A (fr) Nouveaux derives de l'acide phosphorique,
FR2281101A1 (fr) Derives de l'acide prostanoique
BE828186A (fr) Derives de l'acide prostanoique
BE811209A (fr) Nouveaux derives de l'acide phenylacetique
BE852313A (fr) Nouveaux derives d'acide 4,5-dichlorimidazole-2-carboxylique
FR2305175A1 (fr) Nouveaux derives d'acide prostenoique
BE816343A (fr) Nouveaux derives de l'acide phenyl acetique
BE808969A (fr) Nouveaux derives de l'acide prostanoique
BE852172A (fr) Nouveaux derives de l'acide pyridil-phosphorique
BE782149A (fr) Nouveaux derives de l'acide thiohydroximique
BE823372A (fr) Nouveaux derives de l'acide isonicotinique
FR2100777A1 (fr) Nouveaux derives d'acide benzoique
BE824012A (fr) Derives d'acide butanoique