BG103180A - Метод за лечение на сърдечна недостатъчност - Google Patents

Метод за лечение на сърдечна недостатъчност Download PDF

Info

Publication number: BG103180A
Authority: BG; Bulgaria
Prior art keywords: dimethyl; phenoxy; trimethyl; ethyl; propoxy
Prior art date: 1998-02-17

Application number

BG103180A

Other languages

Bulgarian (bg)

English (en)

Inventor

Yuhpyng Chen

Anthony FOSSA

Original Assignee

Pfizer Products Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-02-17

Filing date

1999-02-16

Publication date

1999-09-30

1999-02-16 Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.

1999-09-30 Publication of BG103180A publication Critical patent/BG103180A/bg

Links

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QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
229960000281 trometamol Drugs 0.000 description 1
231100000397 ulcer Toxicity 0.000 description 1
230000002861 ventricular Effects 0.000 description 1
238000010792 warming Methods 0.000 description 1
238000005303 weighing Methods 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Life Sciences & Earth Sciences (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

BG103180A 1998-02-17 1999-02-16 Метод за лечение на сърдечна недостатъчност BG103180A (bg)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US7493498P	1998-02-17	1998-02-17

Publications (1)

Publication Number	Publication Date
BG103180A true BG103180A (bg)	1999-09-30

Family

ID=22122537

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG103180A BG103180A (bg)	1998-02-17	1999-02-16	Метод за лечение на сърдечна недостатъчност

Country Status (28)

Country	Link
US (1)	US6043260A (id)
EP (1)	EP0951906A1 (id)
JP (1)	JPH11292766A (id)
KR (1)	KR19990072616A (id)
CN (1)	CN1231176A (id)
AP (1)	AP9901464A0 (id)
AR (1)	AR017723A1 (id)
AU (1)	AU1732999A (id)
BG (1)	BG103180A (id)
BR (1)	BR9900653A (id)
CA (1)	CA2262252C (id)
EA (1)	EA199900124A3 (id)
GT (1)	GT199900015A (id)
HR (1)	HRP990054A2 (id)
HU (1)	HUP9900386A3 (id)
ID (1)	ID23218A (id)
IL (1)	IL128531A0 (id)
IS (1)	IS4975A (id)
MA (1)	MA26608A1 (id)
NO (1)	NO990722L (id)
OA (1)	OA10976A (id)
PA (1)	PA8467401A1 (id)
PE (1)	PE20000266A1 (id)
PL (1)	PL331507A1 (id)
SG (1)	SG81261A1 (id)
TN (1)	TNSN99024A1 (id)
TR (1)	TR199900328A2 (id)
ZA (1)	ZA991220B (id)

Families Citing this family (23)

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US6403599B1 (en)	1995-11-08	2002-06-11	Pfizer Inc	Corticotropin releasing factor antagonists
US7125880B1 (en)	1995-06-06	2006-10-24	Pfizer Inc.	Corticotropin releasing factor antagonists
US6956047B1 (en)	1995-06-06	2005-10-18	Pfizer Inc.	Corticotropin releasing factor antagonists
US6387894B1 (en) *	1999-06-11	2002-05-14	Pfizer Inc.	Use of CRF antagonists and renin-angiotensin system inhibitors
JP2003509478A (ja) *	1999-09-21	2003-03-11	エモリー・ユニバーシティ	血小板関連障害を処置する方法および組成物
CA2397633A1 (en) *	2000-01-18	2001-07-26	Pfizer Products Inc.	Corticotropin releasing factor antagonists
GB0027410D0 (en) *	2000-11-09	2000-12-27	Pfizer Ltd	Mutual prodrug of amlodipine and atorvastatin
US6737430B2 (en)	2000-11-09	2004-05-18	Pfizer, Inc.	Mutual prodrug of amlodipine and atorvastatin
US6992087B2 (en)	2001-11-21	2006-01-31	Pfizer Inc	Substituted aryl 1,4-pyrazine derivatives
WO2003072107A1 (en)	2002-02-22	2003-09-04	Pharmacia & Upjohn Company	Substituted pyrimidinones and pyrimidinthiones
AU2003220190A1 (en) *	2002-03-13	2003-09-29	Pharmacia & Upjohn Company Llc	Pyrazolo(1,5-a)pyridine derivatives as neurotransmitter modulators
BR0309551A (pt) *	2002-04-26	2005-02-09	Upjohn Co	Derivados substituìdos de pirazina
EP1539736A1 (en) *	2002-09-12	2005-06-15	Pharmacia & Upjohn Company LLC	Substituted 1,4-pyrazine derivatives
AR041470A1 (es) *	2002-10-17	2005-05-18	Upjohn Co	Compuestos de pirrolo (1,2 - b) piridazina y sus usos
AU2003278542A1 (en) *	2002-11-21	2004-06-15	Pharmacia & Upjohn Company Llc	Pyrazine compounds as crf modulators
MXPA05011387A (es) *	2003-04-23	2005-12-01	Pharmacia & Upjohn Co Llc	Pirimidinonas y pirimidinotionas sustituidas.
JP2006525309A (ja) *	2003-05-07	2006-11-09	ファルマシア・アンド・アップジョン・カンパニー・エルエルシー	ピロロ（１，２−ｂ）ピリダジン化合物、ならびにＣＲＦ−１受容体拮抗薬としてのその使用
EP1625115A1 (en) *	2003-05-09	2006-02-15	Pharmacia & Upjohn Company LLC	Substituted pyrimidine derivatives
CA2525195A1 (en) *	2003-05-09	2004-11-18	Pharmacia & Upjohn Company Llc	Pyrazinones as crf1 receptor antagonists for the treatment of cns disorders
MXPA05012082A (es) *	2003-05-09	2006-02-22	Pharmacia & Upjohn Co Llc	Compuestos como antagonistas del receptor crf1.
WO2005089639A2 (en) *	2004-03-16	2005-09-29	Talarico M D Matthew T	Method for vascular dysregulation
US20060211710A1 (en) *	2005-03-17	2006-09-21	Pfizer Inc	Substituted aryl 1,4-pyrazine derivatives
US8338441B2 (en) *	2009-05-15	2012-12-25	Gilead Sciences, Inc.	Inhibitors of human immunodeficiency virus replication

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW574214B (en) *	1994-06-08	2004-02-01	Pfizer	Corticotropin releasing factor antagonists
US6403599B1 (en) *	1995-11-08	2002-06-11	Pfizer Inc	Corticotropin releasing factor antagonists
EP0795327A1 (en) *	1996-03-13	1997-09-17	Pfizer Inc.	Use of Amlodipine for the treatment and prophylaxis of congestive cardiac failure of non-ischaemic origin

1999
- 1999-01-18 PA PA19998467401A patent/PA8467401A1/es unknown
- 1999-02-02 GT GT199900015A patent/GT199900015A/es unknown
- 1999-02-10 US US09/248,073 patent/US6043260A/en not_active Expired - Fee Related
- 1999-02-10 SG SG9900526A patent/SG81261A1/en unknown
- 1999-02-11 AP APAP/P/1999/001464A patent/AP9901464A0/en unknown
- 1999-02-11 EP EP99301006A patent/EP0951906A1/en not_active Withdrawn
- 1999-02-11 IS IS4975A patent/IS4975A/is unknown
- 1999-02-11 CN CN99102122A patent/CN1231176A/zh active Pending
- 1999-02-12 KR KR1019990004934A patent/KR19990072616A/ko not_active Ceased
- 1999-02-12 BR BR9900653-7A patent/BR9900653A/pt not_active Application Discontinuation
- 1999-02-12 PE PE1999000127A patent/PE20000266A1/es not_active Application Discontinuation
- 1999-02-15 IL IL12853199A patent/IL128531A0/xx unknown
- 1999-02-15 CA CA002262252A patent/CA2262252C/en not_active Expired - Fee Related
- 1999-02-15 ID IDP990113D patent/ID23218A/id unknown
- 1999-02-16 AU AU17329/99A patent/AU1732999A/en not_active Abandoned
- 1999-02-16 MA MA25465A patent/MA26608A1/fr unknown
- 1999-02-16 AR ARP990100619A patent/AR017723A1/es unknown
- 1999-02-16 JP JP11037464A patent/JPH11292766A/ja active Pending
- 1999-02-16 ZA ZA9901220A patent/ZA991220B/xx unknown
- 1999-02-16 BG BG103180A patent/BG103180A/bg unknown
- 1999-02-16 NO NO990722A patent/NO990722L/no unknown
- 1999-02-16 OA OA9900034A patent/OA10976A/en unknown
- 1999-02-16 EA EA199900124A patent/EA199900124A3/ru unknown
- 1999-02-16 TN TNTNSN99024A patent/TNSN99024A1/fr unknown
- 1999-02-16 HU HU9900386A patent/HUP9900386A3/hu unknown
- 1999-02-16 TR TR1999/00328A patent/TR199900328A2/xx unknown
- 1999-02-17 PL PL99331507A patent/PL331507A1/xx unknown
- 1999-02-17 HR HR60/074,934A patent/HRP990054A2/hr not_active Application Discontinuation

Also Published As

Publication number	Publication date
IL128531A0 (en)	2000-01-31
BR9900653A (pt)	2000-10-17
OA10976A (en)	2001-11-05
AP9901464A0 (en)	1999-03-31
PL331507A1 (en)	1999-08-30
HUP9900386A3 (en)	1999-12-28
US6043260A (en)	2000-03-28
SG81261A1 (en)	2001-06-19
IS4975A (is)	1999-08-18
MA26608A1 (fr)	2004-12-20
NO990722D0 (no)	1999-02-16
AU1732999A (en)	1999-09-02
GT199900015A (es)	2000-07-26
CN1231176A (zh)	1999-10-13
CA2262252A1 (en)	1999-08-17
ZA991220B (en)	2000-08-16
EA199900124A2 (ru)	1999-08-26
TNSN99024A1 (fr)	2005-11-10
NO990722L (no)	1999-08-18
HUP9900386A2 (hu)	1999-11-29
HU9900386D0 (en)	1999-04-28
PE20000266A1 (es)	2000-04-07
JPH11292766A (ja)	1999-10-26
ID23218A (id)	2000-03-30
AR017723A1 (es)	2001-09-12
EA199900124A3 (ru)	1999-12-29
CA2262252C (en)	2006-01-10
TR199900328A2 (xx)	1999-10-21
EP0951906A1 (en)	1999-10-27
KR19990072616A (ko)	1999-09-27
PA8467401A1 (es)	2000-09-29
HRP990054A2 (en)	2000-02-29

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US6043260A (en)	2000-03-28	Method of treating heart failure
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EP0908456A1 (de)	1999-04-14	Pyrazol-Derivate, ihre Herstellung und ihre Verwendung in Arzneimitteln
US5693674A (en)	1997-12-02	Method of using triaryl-ethylene derivatives in the treatment and prevention of osteoporosis
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JP3962110B2 (ja)	2007-08-22	置換されたベンジルオキシカルボニルグアニジン、それらの製造法、医薬または診断剤としてのそれらの使用およびそれらを含有する医薬
EP1176144B1 (de)	2003-07-09	Neue N-Triazolylmethyl-Piperazinderivate als Neurokininrezeptor-Antagonisten
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JPS63297358A (ja)	1988-12-05	ジアリールアルキル置換アルキルアミン
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JPH11100382A (ja)	1999-04-13	スルホンアミド置換化合物、その製法、医薬または診断薬としての使用およびそれを含有する医薬
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