BG103180A - Метод за лечение на сърдечна недостатъчност - Google Patents

Метод за лечение на сърдечна недостатъчност Download PDF

Info

Publication number: BG103180A
Authority: BG; Bulgaria
Prior art keywords: dimethyl; phenoxy; trimethyl; ethyl; propoxy
Prior art date: 1998-02-17

Application number

BG103180A

Other languages

Bulgarian (bg)

English (en)

Inventor

Yuhpyng Chen

Anthony FOSSA

Original Assignee

Pfizer Products Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-02-17

Filing date

1999-02-16

Publication date

1999-09-30

1999-02-16 Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.

1999-09-30 Publication of BG103180A publication Critical patent/BG103180A/bg

Links

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QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
229960000281 trometamol Drugs 0.000 description 1
231100000397 ulcer Toxicity 0.000 description 1
230000002861 ventricular Effects 0.000 description 1
238000010792 warming Methods 0.000 description 1
238000005303 weighing Methods 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

BG103180A 1998-02-17 1999-02-16 Метод за лечение на сърдечна недостатъчност BG103180A (bg)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US7493498P	1998-02-17	1998-02-17

Publications (1)

Publication Number	Publication Date
BG103180A true BG103180A (bg)	1999-09-30

Family

ID=22122537

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG103180A BG103180A (bg)	1998-02-17	1999-02-16	Метод за лечение на сърдечна недостатъчност

Country Status (28)

Country	Link
US (1)	US6043260A (is)
EP (1)	EP0951906A1 (is)
JP (1)	JPH11292766A (is)
KR (1)	KR19990072616A (is)
CN (1)	CN1231176A (is)
AP (1)	AP9901464A0 (is)
AR (1)	AR017723A1 (is)
AU (1)	AU1732999A (is)
BG (1)	BG103180A (is)
BR (1)	BR9900653A (is)
CA (1)	CA2262252C (is)
EA (1)	EA199900124A3 (is)
GT (1)	GT199900015A (is)
HR (1)	HRP990054A2 (is)
HU (1)	HUP9900386A3 (is)
ID (1)	ID23218A (is)
IL (1)	IL128531A0 (is)
IS (1)	IS4975A (is)
MA (1)	MA26608A1 (is)
NO (1)	NO990722L (is)
OA (1)	OA10976A (is)
PA (1)	PA8467401A1 (is)
PE (1)	PE20000266A1 (is)
PL (1)	PL331507A1 (is)
SG (1)	SG81261A1 (is)
TN (1)	TNSN99024A1 (is)
TR (1)	TR199900328A2 (is)
ZA (1)	ZA991220B (is)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
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US7067664B1 (en)	1995-06-06	2006-06-27	Pfizer Inc.	Corticotropin releasing factor antagonists
US6403599B1 (en)	1995-11-08	2002-06-11	Pfizer Inc	Corticotropin releasing factor antagonists
US6956047B1 (en)	1995-06-06	2005-10-18	Pfizer Inc.	Corticotropin releasing factor antagonists
US6387894B1 (en) *	1999-06-11	2002-05-14	Pfizer Inc.	Use of CRF antagonists and renin-angiotensin system inhibitors
EP1216037A2 (en)	1999-09-21	2002-06-26	Emory University	Methods and compositions for treating platelet-related disorders using mpl pathway inhibitory agents
MXPA02007047A (es) *	2000-01-18	2002-12-13	Pfizer Prod Inc	Antagonista del factor liberador de corticotropina.
GB0027410D0 (en) *	2000-11-09	2000-12-27	Pfizer Ltd	Mutual prodrug of amlodipine and atorvastatin
US6737430B2 (en)	2000-11-09	2004-05-18	Pfizer, Inc.	Mutual prodrug of amlodipine and atorvastatin
US6992087B2 (en)	2001-11-21	2006-01-31	Pfizer Inc	Substituted aryl 1,4-pyrazine derivatives
EP1476165A1 (en)	2002-02-22	2004-11-17	PHARMACIA & UPJOHN COMPANY	Substituted pyrimidinones and pyrimidinthiones
CA2478715A1 (en) *	2002-03-13	2003-09-25	Pharmacia & Upjohn Company	Novel pyrazolo [1,5-a]pyridine derivatives and their use as neurotransmitter modulators
AU2003223475A1 (en) *	2002-04-26	2003-11-10	Pharmacia And Upjohn Company	Substituted pyrazine derivatives
EP1539736A1 (en) *	2002-09-12	2005-06-15	Pharmacia & Upjohn Company LLC	Substituted 1,4-pyrazine derivatives
AR041470A1 (es) *	2002-10-17	2005-05-18	Upjohn Co	Compuestos de pirrolo (1,2 - b) piridazina y sus usos
WO2004046136A1 (en) *	2002-11-21	2004-06-03	Pharmacia & Upjohn Company Llc	Pyrazine compounds as crf modulators
BRPI0409649A (pt) *	2003-04-23	2006-04-25	Pharmacia & Upjohn Co Llc	pirimidinonas e pirimidinotionas substituìdas como antagonistas de crf
MXPA05011993A (es) *	2003-05-07	2006-02-02	Pharmacia & Upjohn Co Llc	Compuestos de pirrolo[1,2-b]piridazina.
CA2524519A1 (en) *	2003-05-09	2004-11-18	Pharmacia & Upjohn Company Llc	Compounds as crf1 receptor antagonists
MXPA05012081A (es) *	2003-05-09	2006-02-22	Pharmacia & Upjohn Co Llc	Derivados de pirimidina sustituidos.
EP1626965A1 (en) *	2003-05-09	2006-02-22	Pharmacia & Upjohn Company LLC	Pyrazinones as crf1 receptor antagonists for the treatment of cns disorders
WO2005089639A2 (en) *	2004-03-16	2005-09-29	Talarico M D Matthew T	Method for vascular dysregulation
US20060211710A1 (en) *	2005-03-17	2006-09-21	Pfizer Inc	Substituted aryl 1,4-pyrazine derivatives
US8338441B2 (en) *	2009-05-15	2012-12-25	Gilead Sciences, Inc.	Inhibitors of human immunodeficiency virus replication

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW574214B (en) *	1994-06-08	2004-02-01	Pfizer	Corticotropin releasing factor antagonists
US6403599B1 (en) *	1995-11-08	2002-06-11	Pfizer Inc	Corticotropin releasing factor antagonists
EP0795327A1 (en) *	1996-03-13	1997-09-17	Pfizer Inc.	Use of Amlodipine for the treatment and prophylaxis of congestive cardiac failure of non-ischaemic origin

1999
- 1999-01-18 PA PA19998467401A patent/PA8467401A1/es unknown
- 1999-02-02 GT GT199900015A patent/GT199900015A/es unknown
- 1999-02-10 SG SG9900526A patent/SG81261A1/en unknown
- 1999-02-10 US US09/248,073 patent/US6043260A/en not_active Expired - Fee Related
- 1999-02-11 CN CN99102122A patent/CN1231176A/zh active Pending
- 1999-02-11 EP EP99301006A patent/EP0951906A1/en not_active Withdrawn
- 1999-02-11 IS IS4975A patent/IS4975A/is unknown
- 1999-02-11 AP APAP/P/1999/001464A patent/AP9901464A0/en unknown
- 1999-02-12 BR BR9900653-7A patent/BR9900653A/pt not_active Application Discontinuation
- 1999-02-12 KR KR1019990004934A patent/KR19990072616A/ko not_active Ceased
- 1999-02-12 PE PE1999000127A patent/PE20000266A1/es not_active Application Discontinuation
- 1999-02-15 CA CA002262252A patent/CA2262252C/en not_active Expired - Fee Related
- 1999-02-15 IL IL12853199A patent/IL128531A0/xx unknown
- 1999-02-15 ID IDP990113D patent/ID23218A/id unknown
- 1999-02-16 JP JP11037464A patent/JPH11292766A/ja active Pending
- 1999-02-16 ZA ZA9901220A patent/ZA991220B/xx unknown
- 1999-02-16 EA EA199900124A patent/EA199900124A3/ru unknown
- 1999-02-16 TN TNTNSN99024A patent/TNSN99024A1/fr unknown
- 1999-02-16 MA MA25465A patent/MA26608A1/fr unknown
- 1999-02-16 TR TR1999/00328A patent/TR199900328A2/xx unknown
- 1999-02-16 HU HU9900386A patent/HUP9900386A3/hu unknown
- 1999-02-16 AU AU17329/99A patent/AU1732999A/en not_active Abandoned
- 1999-02-16 AR ARP990100619A patent/AR017723A1/es unknown
- 1999-02-16 NO NO990722A patent/NO990722L/no unknown
- 1999-02-16 OA OA9900034A patent/OA10976A/en unknown
- 1999-02-16 BG BG103180A patent/BG103180A/bg unknown
- 1999-02-17 PL PL99331507A patent/PL331507A1/xx unknown
- 1999-02-17 HR HR60/074,934A patent/HRP990054A2/hr not_active Application Discontinuation

Also Published As

Publication number	Publication date
CA2262252A1 (en)	1999-08-17
HUP9900386A2 (hu)	1999-11-29
EP0951906A1 (en)	1999-10-27
CA2262252C (en)	2006-01-10
AU1732999A (en)	1999-09-02
SG81261A1 (en)	2001-06-19
HUP9900386A3 (en)	1999-12-28
AR017723A1 (es)	2001-09-12
OA10976A (en)	2001-11-05
MA26608A1 (fr)	2004-12-20
NO990722D0 (no)	1999-02-16
HRP990054A2 (en)	2000-02-29
EA199900124A3 (ru)	1999-12-29
KR19990072616A (ko)	1999-09-27
IL128531A0 (en)	2000-01-31
ZA991220B (en)	2000-08-16
ID23218A (id)	2000-03-30
AP9901464A0 (en)	1999-03-31
US6043260A (en)	2000-03-28
NO990722L (no)	1999-08-18
PA8467401A1 (es)	2000-09-29
EA199900124A2 (ru)	1999-08-26
CN1231176A (zh)	1999-10-13
PE20000266A1 (es)	2000-04-07
GT199900015A (es)	2000-07-26
TR199900328A2 (xx)	1999-10-21
IS4975A (is)	1999-08-18
JPH11292766A (ja)	1999-10-26
HU9900386D0 (en)	1999-04-28
TNSN99024A1 (fr)	2005-11-10
PL331507A1 (en)	1999-08-30
BR9900653A (pt)	2000-10-17

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JPH11100382A (ja)	1999-04-13	スルホンアミド置換化合物、その製法、医薬または診断薬としての使用およびそれを含有する医薬
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