BG103432A - Derivatives of 1,4-diazabicyclo[2.2.2]oct-2-ylmethylbenzoate, method for their preparation and application in therapy - Google Patents
Derivatives of 1,4-diazabicyclo[2.2.2]oct-2-ylmethylbenzoate, method for their preparation and application in therapyInfo
- Publication number
- BG103432A BG103432A BG103432A BG10343299A BG103432A BG 103432 A BG103432 A BG 103432A BG 103432 A BG103432 A BG 103432A BG 10343299 A BG10343299 A BG 10343299A BG 103432 A BG103432 A BG 103432A
- Authority
- BG
- Bulgaria
- Prior art keywords
- ylmethylbenzoate
- diazabicyclo
- oct
- therapy
- derivatives
- Prior art date
Links
- NAIHEECEPHODMQ-UHFFFAOYSA-N 1,4-diazabicyclo[2.2.2]octan-3-ylmethyl benzoate Chemical class C1N(CC2)CCN2C1COC(=O)C1=CC=CC=C1 NAIHEECEPHODMQ-UHFFFAOYSA-N 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 238000002560 therapeutic procedure Methods 0.000 title 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000003277 amino group Chemical group 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 239000003446 ligand Substances 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 239000000387 serotonin 5-HT4 receptor agonist Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Otolaryngology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9614847A FR2756563B1 (fr) | 1996-12-04 | 1996-12-04 | Derives de benzoate de 1,4-diazabicyclo[2.2.2]oct-2-yl- methyle, leur preparation et leur application en therapeutique |
| PCT/FR1997/002174 WO1998024790A1 (fr) | 1996-12-04 | 1997-12-02 | Derives de benzoate de 1,4-diazabicyclo[2.2.2]oct-2-ylmethyle, leur preparation et leur application en therapeutique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG103432A true BG103432A (en) | 2000-06-30 |
Family
ID=9498306
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG103432A BG103432A (en) | 1996-12-04 | 1999-05-26 | Derivatives of 1,4-diazabicyclo[2.2.2]oct-2-ylmethylbenzoate, method for their preparation and application in therapy |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US6057321A (fr) |
| EP (1) | EP0942910A1 (fr) |
| JP (1) | JP2001504855A (fr) |
| KR (1) | KR20000069283A (fr) |
| CN (1) | CN1239962A (fr) |
| AU (1) | AU7624598A (fr) |
| BG (1) | BG103432A (fr) |
| BR (1) | BR9714215A (fr) |
| CA (1) | CA2271072A1 (fr) |
| CZ (1) | CZ193799A3 (fr) |
| EE (1) | EE9900218A (fr) |
| FR (1) | FR2756563B1 (fr) |
| HU (1) | HUP9904206A3 (fr) |
| IL (1) | IL129927A0 (fr) |
| NO (1) | NO992676L (fr) |
| NZ (1) | NZ336044A (fr) |
| SK (1) | SK74199A3 (fr) |
| TR (1) | TR199901068T2 (fr) |
| WO (1) | WO1998024790A1 (fr) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2223588C (fr) | 1995-06-07 | 2004-01-06 | Noven Pharmaceuticals, Inc. | Compositions transdermiques contenant des medicaments de faible poids moleculaire liquides a temperature ambiante |
| WO2004090030A1 (fr) * | 2003-04-08 | 2004-10-21 | Ciba Specialty Chemicals Holding Inc. | Dispersants polymeres photostabilisants dans des dispersions de pigments |
| US7880683B2 (en) * | 2004-08-18 | 2011-02-01 | Ruckus Wireless, Inc. | Antennas with polarization diversity |
| US8198386B2 (en) | 2007-04-16 | 2012-06-12 | Daikin Industries, Ltd. | Fluorine-containing elastomer composition and sealing material made of same |
| CN101842375A (zh) * | 2007-09-03 | 2010-09-22 | 巴斯夫欧洲公司 | 制备teda衍生物的方法 |
| CN102046629A (zh) * | 2008-05-30 | 2011-05-04 | 东曹株式会社 | 羟基烷基三亚乙基二胺类化合物的制造方法以及使用该化合物的用于制造聚氨酯树脂的催化剂组合物 |
| US20110077376A1 (en) * | 2008-05-30 | 2011-03-31 | Katsumi Tokumoto | Process for producing hydroxyalkyltriethylenediamine, and catalyst composition for the production of polyurethane resin using it |
| CN101671336B (zh) * | 2009-09-23 | 2013-11-13 | 辽宁利锋科技开发有限公司 | 芳杂环并嘧啶衍生物和类似物及其制备方法和用途 |
| JP5504835B2 (ja) * | 2009-11-13 | 2014-05-28 | 東ソー株式会社 | ヒドロキシアルキルピペラジン類及び／又はヒドロキシメチルトリエチレンジアミン類の製造方法 |
| JP5549847B2 (ja) * | 2009-11-16 | 2014-07-16 | 東ソー株式会社 | Ｎ−（２−アルコキシメチル）トリエチレンジアミン類の製造法 |
| JP5707912B2 (ja) * | 2010-12-08 | 2015-04-30 | 東ソー株式会社 | Ｎ−（ジヒドロキシアルキル）ジエチレントリアミン類の組成物、及びそれを用いた２−ヒドロキシ（アルキル）トリエチレンジアミン類の製造方 |
| JP6393959B2 (ja) | 2012-05-31 | 2018-09-26 | 東ソー株式会社 | ポリウレタン樹脂製造用触媒組成物及びそれを用いたポリウレタン樹脂の製造方法 |
| JP6252152B2 (ja) * | 2013-12-11 | 2017-12-27 | 東ソー株式会社 | 二環式アミン化合物の製造方法 |
| KR20220055152A (ko) | 2020-10-26 | 2022-05-03 | 인하대학교 산학협력단 | 급성 융모양막염 진단용 조성물 및 이를 이용한 급성 융모양막염 진단방법 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4772459A (en) * | 1986-09-09 | 1988-09-20 | Erbamont, Inc. | Method for controlling emesis caused by chemotherapeutic agents and antiemetic agents useful therein |
| TW282460B (fr) * | 1993-12-28 | 1996-08-01 | Yamanouchi Pharma Co Ltd | |
| FR2735475B1 (fr) * | 1995-06-13 | 1997-07-11 | Synthelabo | Derives de n-((1,4-diazabicyclo(2.2.2)oct-2-yl)methyl) benzamide, leur preparation et leur application en therapeutique |
-
1996
- 1996-12-04 FR FR9614847A patent/FR2756563B1/fr not_active Expired - Fee Related
-
1997
- 1997-12-02 KR KR1019997004915A patent/KR20000069283A/ko not_active Withdrawn
- 1997-12-02 TR TR1999/01068T patent/TR199901068T2/xx unknown
- 1997-12-02 NZ NZ336044A patent/NZ336044A/xx unknown
- 1997-12-02 AU AU76245/98A patent/AU7624598A/en not_active Abandoned
- 1997-12-02 WO PCT/FR1997/002174 patent/WO1998024790A1/fr not_active Ceased
- 1997-12-02 CA CA002271072A patent/CA2271072A1/fr not_active Abandoned
- 1997-12-02 IL IL12992797A patent/IL129927A0/xx unknown
- 1997-12-02 US US09/319,413 patent/US6057321A/en not_active Expired - Fee Related
- 1997-12-02 BR BR9714215-8A patent/BR9714215A/pt not_active Application Discontinuation
- 1997-12-02 HU HU9904206A patent/HUP9904206A3/hu unknown
- 1997-12-02 JP JP52527298A patent/JP2001504855A/ja active Pending
- 1997-12-02 SK SK741-99A patent/SK74199A3/sk unknown
- 1997-12-02 EP EP97948976A patent/EP0942910A1/fr not_active Withdrawn
- 1997-12-02 CN CN97180353A patent/CN1239962A/zh active Pending
- 1997-12-02 CZ CZ991937A patent/CZ193799A3/cs unknown
- 1997-12-02 EE EEP199900218A patent/EE9900218A/xx unknown
-
1999
- 1999-05-26 BG BG103432A patent/BG103432A/xx unknown
- 1999-06-02 NO NO992676A patent/NO992676L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CZ193799A3 (cs) | 1999-09-15 |
| FR2756563A1 (fr) | 1998-06-05 |
| NO992676L (no) | 1999-07-29 |
| SK74199A3 (en) | 2000-02-14 |
| EP0942910A1 (fr) | 1999-09-22 |
| TR199901068T2 (xx) | 1999-07-21 |
| HUP9904206A2 (hu) | 2000-06-28 |
| EE9900218A (et) | 1999-12-15 |
| HUP9904206A3 (en) | 2000-07-28 |
| CN1239962A (zh) | 1999-12-29 |
| KR20000069283A (ko) | 2000-11-25 |
| US6057321A (en) | 2000-05-02 |
| NO992676D0 (no) | 1999-06-02 |
| CA2271072A1 (fr) | 1998-06-11 |
| JP2001504855A (ja) | 2001-04-10 |
| BR9714215A (pt) | 2000-04-18 |
| NZ336044A (en) | 2000-03-27 |
| AU7624598A (en) | 1998-06-29 |
| WO1998024790A1 (fr) | 1998-06-11 |
| FR2756563B1 (fr) | 1998-12-24 |
| IL129927A0 (en) | 2000-02-29 |
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