NO992676L - 1,4-diazabicyklo[2,2,2]okt-2-ylmetylderivater, deres fremstilling og terapeutiske anvendelse - Google Patents
1,4-diazabicyklo[2,2,2]okt-2-ylmetylderivater, deres fremstilling og terapeutiske anvendelseInfo
- Publication number
- NO992676L NO992676L NO992676A NO992676A NO992676L NO 992676 L NO992676 L NO 992676L NO 992676 A NO992676 A NO 992676A NO 992676 A NO992676 A NO 992676A NO 992676 L NO992676 L NO 992676L
- Authority
- NO
- Norway
- Prior art keywords
- diazabicyclo
- oct
- preparation
- therapeutic use
- ylmethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Oppfinnelsen vedrører forbindelser med generell formel (I) hvor RI representerer en metylgruppe, Xx representerer et hydrogenatom eller ORX og Xx danner sammen en gruppe med formel -O(CH2)2-, -O(CH2)3-, -O(CH2)20- eller -O(CH2)3O-, X2 representerer et hydrogenatom eller en aminogruppe og X3 representerer et halogenatom. Forbindelsene er ligander av serotoninergiske reseptorer av typene 5-HT3 og/eller '5-HT4, og virker som 5-HT4 agonister og/eller 5-HT3 antagonister.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9614847A FR2756563B1 (fr) | 1996-12-04 | 1996-12-04 | Derives de benzoate de 1,4-diazabicyclo[2.2.2]oct-2-yl- methyle, leur preparation et leur application en therapeutique |
| PCT/FR1997/002174 WO1998024790A1 (fr) | 1996-12-04 | 1997-12-02 | Derives de benzoate de 1,4-diazabicyclo[2.2.2]oct-2-ylmethyle, leur preparation et leur application en therapeutique |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO992676D0 NO992676D0 (no) | 1999-06-02 |
| NO992676L true NO992676L (no) | 1999-07-29 |
Family
ID=9498306
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO992676A NO992676L (no) | 1996-12-04 | 1999-06-02 | 1,4-diazabicyklo[2,2,2]okt-2-ylmetylderivater, deres fremstilling og terapeutiske anvendelse |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US6057321A (no) |
| EP (1) | EP0942910A1 (no) |
| JP (1) | JP2001504855A (no) |
| KR (1) | KR20000069283A (no) |
| CN (1) | CN1239962A (no) |
| AU (1) | AU7624598A (no) |
| BG (1) | BG103432A (no) |
| BR (1) | BR9714215A (no) |
| CA (1) | CA2271072A1 (no) |
| CZ (1) | CZ193799A3 (no) |
| EE (1) | EE9900218A (no) |
| FR (1) | FR2756563B1 (no) |
| HU (1) | HUP9904206A3 (no) |
| IL (1) | IL129927A0 (no) |
| NO (1) | NO992676L (no) |
| NZ (1) | NZ336044A (no) |
| SK (1) | SK74199A3 (no) |
| TR (1) | TR199901068T2 (no) |
| WO (1) | WO1998024790A1 (no) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2223588C (en) | 1995-06-07 | 2004-01-06 | Noven Pharmaceuticals, Inc. | Transdermal compositions containing low molecular weight drugs which are liquid at room temperatures |
| CN1802409A (zh) * | 2003-04-08 | 2006-07-12 | 西巴特殊化学品控股有限公司 | 颜料分散体中的光稳定聚合物分散剂 |
| US7880683B2 (en) * | 2004-08-18 | 2011-02-01 | Ruckus Wireless, Inc. | Antennas with polarization diversity |
| US8198386B2 (en) | 2007-04-16 | 2012-06-12 | Daikin Industries, Ltd. | Fluorine-containing elastomer composition and sealing material made of same |
| CN101842375A (zh) * | 2007-09-03 | 2010-09-22 | 巴斯夫欧洲公司 | 制备teda衍生物的方法 |
| US20110077376A1 (en) * | 2008-05-30 | 2011-03-31 | Katsumi Tokumoto | Process for producing hydroxyalkyltriethylenediamine, and catalyst composition for the production of polyurethane resin using it |
| PL2295438T5 (pl) | 2008-05-30 | 2025-07-07 | Tosoh Corporation | Sposób wytwarzania kompozycji zawierającej hydroksyalkilotrietylenodiaminę i kompozycja katalizatora do wytwarzania żywicy poliuretanowej z zastosowaniem kompozycji hydroksyalkilotrietylenodiaminy |
| CN101671336B (zh) * | 2009-09-23 | 2013-11-13 | 辽宁利锋科技开发有限公司 | 芳杂环并嘧啶衍生物和类似物及其制备方法和用途 |
| JP5504835B2 (ja) * | 2009-11-13 | 2014-05-28 | 東ソー株式会社 | ヒドロキシアルキルピペラジン類及び／又はヒドロキシメチルトリエチレンジアミン類の製造方法 |
| JP5549847B2 (ja) * | 2009-11-16 | 2014-07-16 | 東ソー株式会社 | Ｎ−（２−アルコキシメチル）トリエチレンジアミン類の製造法 |
| JP5707912B2 (ja) * | 2010-12-08 | 2015-04-30 | 東ソー株式会社 | Ｎ−（ジヒドロキシアルキル）ジエチレントリアミン類の組成物、及びそれを用いた２−ヒドロキシ（アルキル）トリエチレンジアミン類の製造方 |
| JP6393959B2 (ja) | 2012-05-31 | 2018-09-26 | 東ソー株式会社 | ポリウレタン樹脂製造用触媒組成物及びそれを用いたポリウレタン樹脂の製造方法 |
| JP6252152B2 (ja) * | 2013-12-11 | 2017-12-27 | 東ソー株式会社 | 二環式アミン化合物の製造方法 |
| KR20220055152A (ko) | 2020-10-26 | 2022-05-03 | 인하대학교 산학협력단 | 급성 융모양막염 진단용 조성물 및 이를 이용한 급성 융모양막염 진단방법 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4772459A (en) * | 1986-09-09 | 1988-09-20 | Erbamont, Inc. | Method for controlling emesis caused by chemotherapeutic agents and antiemetic agents useful therein |
| TW282460B (no) * | 1993-12-28 | 1996-08-01 | Yamanouchi Pharma Co Ltd | |
| FR2735475B1 (fr) * | 1995-06-13 | 1997-07-11 | Synthelabo | Derives de n-((1,4-diazabicyclo(2.2.2)oct-2-yl)methyl) benzamide, leur preparation et leur application en therapeutique |
-
1996
- 1996-12-04 FR FR9614847A patent/FR2756563B1/fr not_active Expired - Fee Related
-
1997
- 1997-12-02 CN CN97180353A patent/CN1239962A/zh active Pending
- 1997-12-02 SK SK741-99A patent/SK74199A3/sk unknown
- 1997-12-02 US US09/319,413 patent/US6057321A/en not_active Expired - Fee Related
- 1997-12-02 TR TR1999/01068T patent/TR199901068T2/xx unknown
- 1997-12-02 IL IL12992797A patent/IL129927A0/xx unknown
- 1997-12-02 NZ NZ336044A patent/NZ336044A/xx unknown
- 1997-12-02 BR BR9714215-8A patent/BR9714215A/pt not_active Application Discontinuation
- 1997-12-02 AU AU76245/98A patent/AU7624598A/en not_active Abandoned
- 1997-12-02 HU HU9904206A patent/HUP9904206A3/hu unknown
- 1997-12-02 CZ CZ991937A patent/CZ193799A3/cs unknown
- 1997-12-02 WO PCT/FR1997/002174 patent/WO1998024790A1/fr not_active Ceased
- 1997-12-02 EE EEP199900218A patent/EE9900218A/xx unknown
- 1997-12-02 EP EP97948976A patent/EP0942910A1/fr not_active Withdrawn
- 1997-12-02 KR KR1019997004915A patent/KR20000069283A/ko not_active Withdrawn
- 1997-12-02 JP JP52527298A patent/JP2001504855A/ja active Pending
- 1997-12-02 CA CA002271072A patent/CA2271072A1/fr not_active Abandoned
-
1999
- 1999-05-26 BG BG103432A patent/BG103432A/xx unknown
- 1999-06-02 NO NO992676A patent/NO992676L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| SK74199A3 (en) | 2000-02-14 |
| TR199901068T2 (xx) | 1999-07-21 |
| NZ336044A (en) | 2000-03-27 |
| AU7624598A (en) | 1998-06-29 |
| KR20000069283A (ko) | 2000-11-25 |
| EE9900218A (et) | 1999-12-15 |
| CZ193799A3 (cs) | 1999-09-15 |
| EP0942910A1 (fr) | 1999-09-22 |
| HUP9904206A3 (en) | 2000-07-28 |
| FR2756563B1 (fr) | 1998-12-24 |
| CA2271072A1 (fr) | 1998-06-11 |
| WO1998024790A1 (fr) | 1998-06-11 |
| US6057321A (en) | 2000-05-02 |
| NO992676D0 (no) | 1999-06-02 |
| IL129927A0 (en) | 2000-02-29 |
| HUP9904206A2 (hu) | 2000-06-28 |
| FR2756563A1 (fr) | 1998-06-05 |
| CN1239962A (zh) | 1999-12-29 |
| BR9714215A (pt) | 2000-04-18 |
| JP2001504855A (ja) | 2001-04-10 |
| BG103432A (en) | 2000-06-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |