BG105519A - 3-(benzo(ox/thi)azol-7-yl)-1h-pyrimidine-2,4-diones - Google Patents
3-(benzo(ox/thi)azol-7-yl)-1h-pyrimidine-2,4-dionesInfo
- Publication number
- BG105519A BG105519A BG105519A BG10551901A BG105519A BG 105519 A BG105519 A BG 105519A BG 105519 A BG105519 A BG 105519A BG 10551901 A BG10551901 A BG 10551901A BG 105519 A BG105519 A BG 105519A
- Authority
- BG
- Bulgaria
- Prior art keywords
- alkyl
- halogen
- oxygen
- azol
- diones
- Prior art date
Links
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 6
- 229910052736 halogen Inorganic materials 0.000 abstract 4
- 150000002367 halogens Chemical class 0.000 abstract 4
- 229910052760 oxygen Inorganic materials 0.000 abstract 4
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 3
- 239000001301 oxygen Substances 0.000 abstract 3
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 2
- 239000005864 Sulphur Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 abstract 1
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 abstract 1
- MDFFNEOEWAXZRQ-UHFFFAOYSA-N aminyl Chemical compound [NH2] MDFFNEOEWAXZRQ-UHFFFAOYSA-N 0.000 abstract 1
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000004820 halides Chemical class 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 125000004434 sulfur atom Chemical group 0.000 abstract 1
- 125000002813 thiocarbonyl group Chemical group *C(*)=S 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
- A01N43/76—1,3-Oxazoles; Hydrogenated 1,3-oxazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
- A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/40—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
- C07C271/42—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/54—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C275/30—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by halogen atoms, or by nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19852802 | 1998-11-16 | ||
| PCT/EP1999/008514 WO2000028822A2 (fr) | 1998-11-16 | 1999-11-06 | 3-[benz(ox/thi)azol-7-yl]-1h-pyrimidin-2,4-diones |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG105519A true BG105519A (en) | 2002-01-31 |
Family
ID=7887962
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG105519A BG105519A (en) | 1998-11-16 | 2001-05-17 | 3-(benzo(ox/thi)azol-7-yl)-1h-pyrimidine-2,4-diones |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US6624119B1 (fr) |
| EP (1) | EP1131319B1 (fr) |
| JP (1) | JP2002529481A (fr) |
| KR (1) | KR20010104299A (fr) |
| CN (1) | CN1330649A (fr) |
| AR (1) | AR031062A1 (fr) |
| AT (1) | ATE248834T1 (fr) |
| AU (1) | AU1965500A (fr) |
| BG (1) | BG105519A (fr) |
| BR (1) | BR9915370A (fr) |
| CA (1) | CA2351564A1 (fr) |
| CZ (1) | CZ20011711A3 (fr) |
| DE (1) | DE59906902D1 (fr) |
| EA (1) | EA200100523A1 (fr) |
| HU (1) | HUP0105063A2 (fr) |
| ID (1) | ID28945A (fr) |
| IL (1) | IL142912A0 (fr) |
| MA (1) | MA25264A1 (fr) |
| NO (1) | NO20012386L (fr) |
| PL (1) | PL348187A1 (fr) |
| SK (1) | SK6722001A3 (fr) |
| TR (1) | TR200101359T2 (fr) |
| WO (1) | WO2000028822A2 (fr) |
| ZA (1) | ZA200104913B (fr) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001012625A2 (fr) * | 1999-08-12 | 2001-02-22 | Basf Aktiengesellschaft | Benzoxazoles substitues |
| GB2467670B (en) | 2007-10-04 | 2012-08-01 | Intellikine Inc | Chemical entities and therapeutic uses thereof |
| US8993580B2 (en) | 2008-03-14 | 2015-03-31 | Intellikine Llc | Benzothiazole kinase inhibitors and methods of use |
| JP5547099B2 (ja) | 2008-03-14 | 2014-07-09 | インテリカイン， エルエルシー | キナーゼ阻害剤および使用方法 |
| AU2009268611B2 (en) | 2008-07-08 | 2015-04-09 | Intellikine, Llc | Kinase inhibitors and methods of use |
| US8476282B2 (en) | 2008-11-03 | 2013-07-02 | Intellikine Llc | Benzoxazole kinase inhibitors and methods of use |
| MY162604A (en) | 2009-08-17 | 2017-06-30 | Intellikine Llc | Heterocyclic compounds and uses thereof |
| JP6130305B2 (ja) | 2011-02-23 | 2017-05-17 | インテリカイン， エルエルシー | キナーゼ阻害剤の組み合わせおよびそれらの使用 |
| UA120278C2 (uk) * | 2011-11-25 | 2019-11-11 | Адверіо Фарма Гмбх | Заміщені 5-фтор-1н-піразолопіридини в кристалічній формі |
| WO2014153509A1 (fr) | 2013-03-22 | 2014-09-25 | Millennium Pharmaceuticals, Inc. | Combinaison d'inhibiteurs catalytiques de mtorc1/2 et inhibiteurs sélectifs de la kinase aurora a |
| CN103288683B (zh) * | 2013-06-20 | 2015-09-16 | 郑州福源动物药业有限公司 | 一种“一锅法”制备尼卡巴嗪的方法 |
| CN113194752A (zh) | 2018-06-01 | 2021-07-30 | 康奈尔大学 | Pi3k相关疾病或病症的组合疗法 |
| CN117263927B (zh) * | 2023-09-28 | 2025-09-19 | 西北农林科技大学 | 杂环取代的n-吡啶基苯并噻唑类化合物及制备方法与应用 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK366887A (da) * | 1986-07-31 | 1988-05-13 | Hoffmann La Roche | Pyrimidinderivater |
| ATE111901T1 (de) * | 1990-01-18 | 1994-10-15 | Nissan Chemical Ind Ltd | Uracilderivate und pestizide, die diese als wirksame stoffe enthalten. |
| JPH0525143A (ja) | 1991-07-15 | 1993-02-02 | Nissan Chem Ind Ltd | ３−フエニルウラシル誘導体および除草剤 |
| US5169430A (en) | 1991-08-09 | 1992-12-08 | Uniroyal Chemical Company, Inc. | Benzenesulfonamide derivatives and methods for their production |
| WO1995017096A1 (fr) | 1993-12-22 | 1995-06-29 | Fmc Corporation | Haloalkyluraciles herbicides |
| US5753595A (en) | 1995-08-31 | 1998-05-19 | Fmc Corporation | Herbicidal 3-(substituted benzoxazol-7-yl) and 3-(Substituted benzothiazol-7-yl)-1-substituted-6-trifluoromethyl-2 4-(1h 3h)pyrimidinediones |
| DE19532048A1 (de) | 1995-08-31 | 1997-03-06 | Basf Ag | Substituierte Benzthiazole als Pflanzenschutzmittel |
| US6080702A (en) | 1995-10-04 | 2000-06-27 | Fmc Corporation | Herbicidal heterocyclic benzisoxazoles and benzisoxazolidinones |
| AU7257096A (en) | 1995-10-04 | 1997-04-28 | Fmc Corporation | Herbicidal 6-heterocyclic indazole derivatives |
| JP2001511140A (ja) | 1997-02-04 | 2001-08-07 | ビーエーエスエフ アクチェンゲゼルシャフト | ２−（２，４（１ｈ，３ｈ）−ピリミジンジオン−３−イル）ベンゾチアゾールの置換体 |
| US6077812A (en) | 1997-02-26 | 2000-06-20 | Fmc Corporation | Cycloimido-substituted benzofused heterocyclic herbicides |
| JPH10330359A (ja) | 1997-03-31 | 1998-12-15 | Nippon Bayeragrochem Kk | フエニルアセチレン誘導体及び除草剤 |
| DE19755926A1 (de) * | 1997-12-17 | 1999-06-24 | Basf Ag | Herbizide 3-(Benzazol-4-yl)pyrimidindion-Derivate |
-
1999
- 1999-11-06 WO PCT/EP1999/008514 patent/WO2000028822A2/fr not_active Ceased
- 1999-11-06 SK SK672-2001A patent/SK6722001A3/sk unknown
- 1999-11-06 AT AT99963288T patent/ATE248834T1/de not_active IP Right Cessation
- 1999-11-06 EA EA200100523A patent/EA200100523A1/ru unknown
- 1999-11-06 US US09/830,961 patent/US6624119B1/en not_active Expired - Fee Related
- 1999-11-06 TR TR2001/01359T patent/TR200101359T2/xx unknown
- 1999-11-06 BR BR9915370-0A patent/BR9915370A/pt not_active IP Right Cessation
- 1999-11-06 CA CA002351564A patent/CA2351564A1/fr not_active Abandoned
- 1999-11-06 PL PL99348187A patent/PL348187A1/xx not_active Application Discontinuation
- 1999-11-06 KR KR1020017006112A patent/KR20010104299A/ko not_active Withdrawn
- 1999-11-06 EP EP99963288A patent/EP1131319B1/fr not_active Expired - Lifetime
- 1999-11-06 CN CN99814526A patent/CN1330649A/zh active Pending
- 1999-11-06 DE DE59906902T patent/DE59906902D1/de not_active Expired - Fee Related
- 1999-11-06 JP JP2000581887A patent/JP2002529481A/ja not_active Withdrawn
- 1999-11-06 AU AU19655/00A patent/AU1965500A/en not_active Abandoned
- 1999-11-06 IL IL14291299A patent/IL142912A0/xx unknown
- 1999-11-06 CZ CZ20011711A patent/CZ20011711A3/cs unknown
- 1999-11-06 HU HU0105063A patent/HUP0105063A2/hu unknown
- 1999-11-06 ID IDW00200101285A patent/ID28945A/id unknown
- 1999-11-16 AR ARP990105816A patent/AR031062A1/es not_active Application Discontinuation
-
2001
- 2001-05-09 MA MA26187A patent/MA25264A1/fr unknown
- 2001-05-15 NO NO20012386A patent/NO20012386L/no not_active Application Discontinuation
- 2001-05-17 BG BG105519A patent/BG105519A/xx unknown
- 2001-06-15 ZA ZA200104913A patent/ZA200104913B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BR9915370A (pt) | 2001-08-14 |
| WO2000028822A3 (fr) | 2000-11-16 |
| NO20012386D0 (no) | 2001-05-15 |
| CA2351564A1 (fr) | 2000-05-25 |
| WO2000028822A2 (fr) | 2000-05-25 |
| AU1965500A (en) | 2000-06-05 |
| US6624119B1 (en) | 2003-09-23 |
| ZA200104913B (en) | 2002-08-28 |
| NO20012386L (no) | 2001-05-15 |
| KR20010104299A (ko) | 2001-11-24 |
| MA25264A1 (fr) | 2001-10-01 |
| EA200100523A1 (ru) | 2001-10-22 |
| AR031062A1 (es) | 2003-09-10 |
| PL348187A1 (en) | 2002-05-06 |
| EP1131319A2 (fr) | 2001-09-12 |
| ATE248834T1 (de) | 2003-09-15 |
| JP2002529481A (ja) | 2002-09-10 |
| TR200101359T2 (tr) | 2001-11-21 |
| EP1131319B1 (fr) | 2003-09-03 |
| CZ20011711A3 (cs) | 2002-02-13 |
| SK6722001A3 (en) | 2001-12-03 |
| DE59906902D1 (de) | 2003-10-09 |
| IL142912A0 (en) | 2002-04-21 |
| ID28945A (id) | 2001-07-19 |
| CN1330649A (zh) | 2002-01-09 |
| HUP0105063A2 (hu) | 2002-04-29 |
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