BG35042A3 - Method for preparing benzodiazepinic compounds - Google Patents

Method for preparing benzodiazepinic compounds

Info

Publication number: BG35042A3
Authority: BG; Bulgaria
Prior art keywords: benzodiazepinic; preparing; compounds; formulated; demonstrated
Prior art date: 1979-10-16

Application number

BG057344A

Other languages

Bulgarian (bg)

English (en)

Inventor

Jiban Chakrabarti

Terrence Hotten

Original Assignee

Lilly Industries Limited

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-10-16

Filing date

1980-10-15

Publication date

1983-01-16

1980-10-15 Application filed by Lilly Industries Limited filed Critical Lilly Industries Limited

1983-01-16 Publication of BG35042A3 publication Critical patent/BG35042A3/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Anesthesiology (AREA)
Psychiatry (AREA)
Hospice & Palliative Care (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Plural Heterocyclic Compounds (AREA)

BG057344A 1979-10-16 1980-10-15 Method for preparing benzodiazepinic compounds BG35042A3 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB7935846		1979-10-16

Publications (1)

Publication Number	Publication Date
BG35042A3 true BG35042A3 (en)	1983-01-16

Family

ID=10508540

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
BG057344A BG35042A3 (en)	1979-10-16	1980-10-15	Method for preparing benzodiazepinic compounds
BG049366A BG34907A3 (en)	1979-10-16	1980-10-15	Method for preparing benzodiazepine compounds

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
BG049366A BG34907A3 (en)	1979-10-16	1980-10-15	Method for preparing benzodiazepine compounds

Country Status (33)

Country	Link
US (3)	US4404137A (fr)
EP (1)	EP0027390B1 (fr)
JP (1)	JPS5663987A (fr)
KR (2)	KR850000471B1 (fr)
AR (2)	AR228041A1 (fr)
AT (1)	AT373889B (fr)
AU (1)	AU538500B2 (fr)
BE (1)	BE885729A (fr)
BG (2)	BG35042A3 (fr)
CA (1)	CA1159056A (fr)
CH (1)	CH646700A5 (fr)
CS (1)	CS244409B2 (fr)
DD (1)	DD153692A5 (fr)
DE (1)	DE3068706D1 (fr)
DK (1)	DK437480A (fr)
ES (1)	ES8106905A1 (fr)
FI (1)	FI67550C (fr)
FR (1)	FR2467851A1 (fr)
GB (1)	GB8327127D0 (fr)
GR (1)	GR70720B (fr)
HU (1)	HU182213B (fr)
IE (1)	IE50358B1 (fr)
IL (1)	IL61264A (fr)
IT (1)	IT1143047B (fr)
LU (1)	LU82853A1 (fr)
MX (1)	MX6233E (fr)
NZ (1)	NZ195248A (fr)
PH (2)	PH16288A (fr)
PL (2)	PL126824B1 (fr)
PT (1)	PT71913B (fr)
RO (2)	RO85822B (fr)
YU (1)	YU261580A (fr)
ZA (1)	ZA806342B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4404137A (en) *	1979-10-16	1983-09-13	Lilly Industries Limited	Pyrazolo [3,4-b][1,5]benzodiazepine compounds
US4431589A (en) *	1980-12-11	1984-02-14	Lilly House	Benzodiazepine compounds and their use as pharmaceuticals
US4596799A (en) *	1985-01-29	1986-06-24	Ciba-Geigy Corporation	9H-pyrrolo[2,1-c]-1,2,4-triazolo[4,3-a][1,4]benzodiazepines
TW219896B (fr) *	1988-07-07	1994-02-01	Duphar Int Res
GB8819059D0 (en) *	1988-08-11	1988-09-14	Lilly Industries Ltd	Benzodiazepine compounds & their use as pharmaceuticals
US5631250A (en) *	1995-03-24	1997-05-20	Eli Lilly And Company	Process and solvate of 2-methyl-thieno-benzodiazepine
US5637584A (en) *	1995-03-24	1997-06-10	Eli Lilly And Company	Solvate of olanzapine
US20050250767A1 (en) *	2003-01-23	2005-11-10	Weiner David M	Use of N-desmethylclozapine to treat human neuropsychiatric disease
WO2004064753A2 (fr) *	2003-01-23	2004-08-05	Acadia Pharmaceuticals Inc	Utilisation de la n-desmethylclozapine pour le traitement de maladies neuropsychiatriques chez l'homme
US20050085463A1 (en) *	2003-01-23	2005-04-21	Weiner David M.	Use of N-desmethylclozapine to treat human neuropsychiatric disease
BRPI0417749A (pt) *	2003-12-22	2007-04-10	Acadia Pharm Inc	composto, método de sintese de composto, bibliotecas combinatórias, composições farmacêuticas e métodos de tratamento de disfunções neuropsiquiátricas
BRPI0509524A (pt) *	2004-04-01	2007-09-18	Acadia Pharm Inc	formas cristalinas de n-desmetilclozapina
WO2007053618A1 (fr) *	2005-10-31	2007-05-10	Acadia Pharmaceuticals Inc.	Promédicaments d'agonistes muscariniques et méthodes de traitement de troubles neuropsychiatriques
JP5438482B2 (ja) *	2009-12-03	2014-03-12	Ｊｕｋｉ株式会社	ミシン、ミシンの縫製データ編集装置及びミシンの縫製データ編集プログラム

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3450694A (en) *	1966-02-23	1969-06-17	Abbott Lab	Substituted benzoxazepines and benzothiazepines
US3758479A (en) *	1967-03-22	1973-09-11	Sandoz Ag	Nitro and sulphamoyl substituted dibenzodiazepines
DE1795183B1 (de) *	1968-08-20	1972-07-20	Thomae Gmbh Dr K	5,11-Dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-on-derivate und Arzneimittel
CA918659A (en) *	1969-07-31	1973-01-09	Yoshitomi Pharmaceutical Industries	11-(4-substituted-1-piperazinyl)-dibenzo (b,f) (1,4) thiazepines
US4115568A (en) *	1974-11-26	1978-09-19	Lilly Industries Limited	Thieno[3,2-b]-[1,5]benzodiazepines
US4172831A (en) *	1974-11-26	1979-10-30	Lilly Industries Limited	Thieno-benzodiazepines
US3953430A (en) *	1975-02-24	1976-04-27	American Cyanamid Company	Substituted benzodiazepin-10-ones and method of use
US3951981A (en) *	1975-02-24	1976-04-20	American Cyanamid Company	Substituted benzodiazepines and method of use
DE2707269A1 (de) *	1977-02-19	1978-08-24	Hoechst Ag	Heterocyclische stickstoffverbindungen und verfahren zu ihrer herstellung
DE2707270A1 (de) *	1977-02-19	1978-08-24	Hoechst Ag	Pyrazolo-diazepine und verfahren zu ihrer herstellung
US4097597A (en) *	1977-02-23	1978-06-27	Abbott Laboratories	Dibenzo b,e! 1,4!diazepines
IT7851496A0 (it) *	1977-10-31	1978-10-13	Sandoz Ag	Menti pirazinobenzossazepine loro preparazione e loro impiego quali medica
CH643263A5 (de) *	1979-05-11	1984-05-30	Sandoz Ag	Benzodiazepine, ihre herstellung und verwendung.
CA1154762A (fr) *	1979-08-03	1983-10-04	Georg Rainer	Composes tetraazatricycliques substitues, procede de preparation, applications et medicaments les contenant
US4404137A (en) *	1979-10-16	1983-09-13	Lilly Industries Limited	Pyrazolo [3,4-b][1,5]benzodiazepine compounds

1980
- 1980-10-02 US US06/193,200 patent/US4404137A/en not_active Expired - Lifetime
- 1980-10-11 GR GR63138A patent/GR70720B/el unknown
- 1980-10-13 FR FR8021823A patent/FR2467851A1/fr active Granted
- 1980-10-13 YU YU02615/80A patent/YU261580A/xx unknown
- 1980-10-13 RO RO108967A patent/RO85822B/ro unknown
- 1980-10-13 MX MX809093U patent/MX6233E/es unknown
- 1980-10-13 CS CS806938A patent/CS244409B2/cs unknown
- 1980-10-13 RO RO102349A patent/RO81351B/ro unknown
- 1980-10-13 PH PH24717A patent/PH16288A/en unknown
- 1980-10-13 NZ NZ195248A patent/NZ195248A/xx unknown
- 1980-10-13 IL IL61264A patent/IL61264A/xx unknown
- 1980-10-14 IT IT49899/80A patent/IT1143047B/it active
- 1980-10-14 PT PT71913A patent/PT71913B/pt unknown
- 1980-10-14 AT AT0510180A patent/AT373889B/de not_active IP Right Cessation
- 1980-10-14 CA CA000362328A patent/CA1159056A/fr not_active Expired
- 1980-10-14 CH CH763980A patent/CH646700A5/fr not_active IP Right Cessation
- 1980-10-14 AU AU63252/80A patent/AU538500B2/en not_active Ceased
- 1980-10-15 BG BG057344A patent/BG35042A3/xx unknown
- 1980-10-15 LU LU82853A patent/LU82853A1/fr unknown
- 1980-10-15 JP JP14423180A patent/JPS5663987A/ja active Pending
- 1980-10-15 IE IE2135/80A patent/IE50358B1/en unknown
- 1980-10-15 PL PL1980227306A patent/PL126824B1/pl unknown
- 1980-10-15 ES ES495948A patent/ES8106905A1/es not_active Expired
- 1980-10-15 EP EP80303649A patent/EP0027390B1/fr not_active Expired
- 1980-10-15 HU HU802502A patent/HU182213B/hu not_active IP Right Cessation
- 1980-10-15 KR KR1019800003960A patent/KR850000471B1/ko not_active Expired
- 1980-10-15 BE BE6/47291A patent/BE885729A/fr not_active IP Right Cessation
- 1980-10-15 DD DD80224618A patent/DD153692A5/de unknown
- 1980-10-15 DK DK437480A patent/DK437480A/da not_active Application Discontinuation
- 1980-10-15 FI FI803253A patent/FI67550C/fi not_active IP Right Cessation
- 1980-10-15 DE DE8080303649T patent/DE3068706D1/de not_active Expired
- 1980-10-15 ZA ZA00806342A patent/ZA806342B/xx unknown
- 1980-10-15 BG BG049366A patent/BG34907A3/xx unknown
- 1980-10-15 PL PL1980231270A patent/PL135044B1/pl unknown
- 1980-10-16 AR AR282893A patent/AR228041A1/es active
1982
- 1982-07-21 AR AR290034A patent/AR228101A1/es active
- 1982-07-28 PH PH27643A patent/PH17759A/en unknown
- 1982-09-29 US US06/426,580 patent/US4486591A/en not_active Expired - Fee Related
1983
- 1983-10-11 GB GB838327127A patent/GB8327127D0/en active Pending
1984
- 1984-07-24 KR KR1019840004388A patent/KR850000472B1/ko not_active Expired
- 1984-08-06 US US06/638,181 patent/US4542131A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
AR228101A1 (es)	1983-01-14
FR2467851A1 (fr)	1981-04-30
RO81351B (ro)	1983-02-28
ES495948A0 (es)	1981-09-16
KR850000471B1 (ko)	1985-04-08
PL227306A1 (fr)	1981-09-18
ZA806342B (en)	1982-05-26
BG34907A3 (en)	1983-12-15
EP0027390B1 (fr)	1984-07-25
AT373889B (de)	1984-02-27
NZ195248A (en)	1983-11-18
RO85822B (ro)	1984-11-30
AU6325280A (en)	1981-04-30
FI67550C (fi)	1985-04-10
FI803253L (fi)	1981-04-17
ES8106905A1 (es)	1981-09-16
JPS5663987A (en)	1981-05-30
US4486591A (en)	1984-12-04
DE3068706D1 (en)	1984-08-30
DD153692A5 (de)	1982-01-27
IT1143047B (it)	1986-10-22
US4404137A (en)	1983-09-13
DK437480A (da)	1981-04-17
PL126824B1 (en)	1983-09-30
GB8327127D0 (en)	1983-11-09
PT71913B (en)	1981-08-31
PH16288A (en)	1983-09-05
BE885729A (fr)	1981-04-15
CH646700A5 (fr)	1984-12-14
AU538500B2 (en)	1984-08-16
MX6233E (es)	1985-01-14
PL135044B1 (en)	1985-09-30
LU82853A1 (fr)	1982-05-10
AR228041A1 (es)	1983-01-14
IL61264A (en)	1985-08-30
IE50358B1 (en)	1986-04-02
RO81351A (fr)	1983-02-15
RO85822A (fr)	1984-11-25
IT8049899A0 (it)	1980-10-14
PT71913A (en)	1980-11-01
KR830004300A (ko)	1983-07-09
KR850001463A (ko)	1985-03-18
HU182213B (en)	1983-12-28
EP0027390A1 (fr)	1981-04-22
IE802135L (en)	1981-04-16
PH17759A (en)	1984-12-05
GR70720B (fr)	1983-01-18
CS244409B2 (en)	1986-07-17
PL231270A1 (fr)	1981-12-23
ATA510180A (de)	1983-07-15
IL61264A0 (en)	1980-12-31
CA1159056A (fr)	1983-12-20
US4542131A (en)	1985-09-17
FR2467851B1 (fr)	1985-04-05
YU261580A (en)	1983-12-31
FI67550B (fi)	1984-12-31
KR850000472B1 (ko)	1985-04-08

Publication	Publication Date	Title
BG30474A3 (bg)	1981-06-15	Метод за получаване на 6-п-пропил-8-метоксиметил-или- метилмеркаптометилерголини и сродни съединения
BG31497A3 (bg)	1982-01-15	Метод за получаване на 4-амино-5-алкил-сулфонил ортонизамиди
BG34336A3 (bg)	1983-08-15	Метод за получаване на производни на фталазин -4- ил-оцетна киселина
BG31499A3 (bg)	1982-01-15	Метод за получаване на 1-винилтриазолови производни
BG30019A3 (bg)	1981-03-16	Метод за получаване на тризаместени 1-фенил-2,3,4,5-тетрахидро-1н- 3-бензазепини
BG35189A3 (en)	1984-02-15	Method for preparing derivatives of 6- beta- hydroxyalkylpenicillanic acid
BG33886A3 (en)	1983-05-16	Method for heterocyclic compounds producing
BG38333A3 (bg)	1985-11-15	Метод за получаване на заместени фенилкарбоксиоксими
BG38487A3 (en)	1985-12-16	Method for preparing peptides
BG32851A3 (bg)	1982-10-15	Метод за получаване на 3,4,5,6-тетрахидро-2н- -1-бензоксецини
BG42004A3 (en)	1987-09-15	Method for preparing pyridyl compounds
BG35328A3 (en)	1984-03-15	Method for preparing imidodisulphamidic derivatives
BG29722A3 (bg)	1981-01-15	Метод за получаване на 2,5-дисубституирани пиримидин-4-они
BG34908A3 (bg)	1983-12-15	Метод за получаване на d- 6- n- пропилерголини
BG34907A3 (en)	1983-12-15	Method for preparing benzodiazepine compounds
BG35039A3 (bg)	1984-01-16	Метод за получаване на заместени хетероциклични феноксиамини
BG38638A3 (bg)	1986-01-15	Метод за получаване на арилциклобутил-аминопроизводни
BG31073A3 (bg)	1981-10-15	Метод за получаване на 1,5-заместени-2-пиролидони
BG36935A3 (en)	1985-02-15	Method for preparing benzodiazepine compounds
BG35897A3 (bg)	1984-07-16	Метод за получаване на 5-(дихидрокси-фенокси)-1н-тетразоли
BG38338A3 (en)	1985-11-15	Method for preparing 6 alpha- methylhydrocortisonic derivatives
BG41129A3 (en)	1987-04-15	Method for preparing acetamide derivatives
BG34612A3 (bg)	1983-10-15	Метод за получаване на пиролидинови производни
BG35896A3 (en)	1984-07-16	Method for preparing 3- halogen- 3- cephem compounds
BG35032A3 (bg)	1984-01-16	Метод за получаване на 1, 1, 2- трифенилпропенови производни