BR0214971A - Processo para a produção de um imunossupressor - Google Patents

Processo para a produção de um imunossupressor

Info

Publication number
BR0214971A
BR0214971A BR0214971-0A BR0214971A BR0214971A BR 0214971 A BR0214971 A BR 0214971A BR 0214971 A BR0214971 A BR 0214971A BR 0214971 A BR0214971 A BR 0214971A
Authority
BR
Brazil
Prior art keywords
immunosuppressant
production
producing
immunosupressor
formula
Prior art date
Application number
BR0214971-0A
Other languages
English (en)
Inventor
Acharya Poornaprajna
Gopeeckrishnan Sreenilayam
Sambasivam Ganesh
Original Assignee
Biocon Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biocon Ltd filed Critical Biocon Ltd
Publication of BR0214971A publication Critical patent/BR0214971A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
  • Furan Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

Abstract

"PROCESSO PARA A PRODUçãO DE UM IMUNOSSUPRESSOR". A presente invenção refere-se a um processo para produção de sal de sódio de imunossupressor de fórmula I.
BR0214971-0A 2002-08-29 2002-08-29 Processo para a produção de um imunossupressor BR0214971A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/IN2002/000178 WO2004020426A1 (en) 2002-08-29 2002-08-29 Process for the production of an immunosuppressant

Publications (1)

Publication Number Publication Date
BR0214971A true BR0214971A (pt) 2004-12-14

Family

ID=31972038

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0214971-0A BR0214971A (pt) 2002-08-29 2002-08-29 Processo para a produção de um imunossupressor

Country Status (12)

Country Link
US (1) US7122687B2 (pt)
EP (1) EP1532130B1 (pt)
JP (1) JP4275069B2 (pt)
KR (1) KR100551617B1 (pt)
AT (1) ATE447563T1 (pt)
AU (1) AU2002334381B2 (pt)
BR (1) BR0214971A (pt)
CA (1) CA2468435C (pt)
DE (1) DE60234279D1 (pt)
ES (1) ES2333207T3 (pt)
MX (1) MXNL04000051A (pt)
WO (1) WO2004020426A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005105768A2 (en) * 2004-04-26 2005-11-10 Teva Gyógyszergyár Zàrtköruen Muködo Rèszvènytàrsasàg Process for preparation of mycophenolic acid and ester derivatives thereof
MXPA06005658A (es) 2004-04-27 2007-04-10 Teva Gyogyszergyar Zartkoruen Proceso para preparacion de micofenolato mofetil, y otros esteres de acido micofenolico.
TWI322147B (en) 2004-07-20 2010-03-21 Teva Gyogyszergyar Zartkoruen Mukodo Reszvenytarsasag Crystalline mycophenolate sodium
PL2032712T3 (pl) * 2006-06-29 2010-07-30 Ivax Pharmaceuticals Sro Regulacja wytwarzania kwaśnego metabolitu
WO2008003637A2 (en) * 2006-07-05 2008-01-10 Dsm Ip Assets B.V. Isolation and use of amine salts of mycophenolic acid
MX2008015797A (es) * 2007-04-11 2009-03-06 Teva Gyogyszergyar Zartkoeruen Metodo para reducir el nivel de impurezas en la fermentacion del acido micofenolico.
CN106866594A (zh) * 2017-02-17 2017-06-20 上海华源医药科技发展有限公司 适用于麦考酚钠工业化生产的优化工艺

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA684959B (en) * 1967-11-22 1969-05-22 Lilly Co Eli Agents and methods for inhibiting the growth of malignant tumor cells in warm-blooded mammals
US4727069A (en) * 1987-01-30 1988-02-23 Syntex (U.S.A.) Inc. Heterocyclic aminoalkyl esters of mycophenolic acid, derivatives thereof and pharmaceutical compositions
US5177072A (en) * 1987-01-30 1993-01-05 Syntex (U.S.A.) Inc. Treatment of autoimmune inflammatory, and psoriatic diseases with heterocyclic aminoalkyl esters of mycophenolic acid and derivatives

Also Published As

Publication number Publication date
WO2004020426A1 (en) 2004-03-11
JP4275069B2 (ja) 2009-06-10
CA2468435C (en) 2008-02-19
KR20040079902A (ko) 2004-09-16
JP2005539047A (ja) 2005-12-22
ATE447563T1 (de) 2009-11-15
CA2468435A1 (en) 2004-03-11
ES2333207T3 (es) 2010-02-18
KR100551617B1 (ko) 2006-02-13
US7122687B2 (en) 2006-10-17
EP1532130A1 (en) 2005-05-25
EP1532130B1 (en) 2009-11-04
EP1532130A4 (en) 2008-03-19
AU2002334381A1 (en) 2004-03-19
AU2002334381B2 (en) 2007-01-04
DE60234279D1 (de) 2009-12-17
US20050165243A1 (en) 2005-07-28
MXNL04000051A (es) 2005-02-24

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 12A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2269 DE 01/07/2014.