BRPI0317781B8 - derivado de acilbenzilamina e processos para produção de derivado de benzilamina e de derivado de carbamato - Google Patents
derivado de acilbenzilamina e processos para produção de derivado de benzilamina e de derivado de carbamato Download PDFInfo
- Publication number
- BRPI0317781B8 BRPI0317781B8 BRPI0317781A BRPI0317781A BRPI0317781B8 BR PI0317781 B8 BRPI0317781 B8 BR PI0317781B8 BR PI0317781 A BRPI0317781 A BR PI0317781A BR PI0317781 A BRPI0317781 A BR PI0317781A BR PI0317781 B8 BRPI0317781 B8 BR PI0317781B8
- Authority
- BR
- Brazil
- Prior art keywords
- derivative
- carbamate
- processes
- acylbenzylamine
- general formula
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 4
- 150000003939 benzylamines Chemical class 0.000 title abstract 3
- AKZWRTCWNXHHFR-PDIZUQLASA-N [(3S)-oxolan-3-yl] N-[(2S,3S)-4-[(5S)-5-benzyl-3-[(2R)-2-carbamoyloxy-2,3-dihydro-1H-inden-1-yl]-4-oxo-3H-pyrrol-5-yl]-3-hydroxy-1-phenylbutan-2-yl]carbamate Chemical compound NC(=O)O[C@@H]1Cc2ccccc2C1C1C=N[C@](C[C@H](O)[C@H](Cc2ccccc2)NC(=O)O[C@H]2CCOC2)(Cc2ccccc2)C1=O AKZWRTCWNXHHFR-PDIZUQLASA-N 0.000 title 1
- 125000002252 acyl group Chemical group 0.000 abstract 2
- WGQKYBSKWIADBV-UHFFFAOYSA-N benzylamine Chemical class NCC1=CC=CC=C1 WGQKYBSKWIADBV-UHFFFAOYSA-N 0.000 abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- KXDHJXZQYSOELW-UHFFFAOYSA-M Carbamate Chemical compound NC([O-])=O KXDHJXZQYSOELW-UHFFFAOYSA-M 0.000 abstract 1
- 239000002841 Lewis acid Substances 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 239000003899 bactericide agent Substances 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- -1 haloacyl compound Chemical class 0.000 abstract 1
- 238000003898 horticulture Methods 0.000 abstract 1
- 150000007517 lewis acids Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
- C07C209/62—Preparation of compounds containing amino groups bound to a carbon skeleton by cleaving carbon-to-nitrogen, sulfur-to-nitrogen, or phosphorus-to-nitrogen bonds, e.g. hydrolysis of amides, N-dealkylation of amines or quaternary ammonium compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
- C07C211/26—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
- C07C211/29—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/30—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by doubly-bound oxygen atoms
- C07C233/31—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by doubly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/04—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from amines with formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/18—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by doubly-bound oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
"processo para produção de derivado de benzilamina". a presente invenção refere-se a um processo para produção de um derivado de benzilamina representado pela fórmula geral (3): na qual x^ 1^, r^ 1^ e r^ 2^ são conforme definidos abaixo, que compreende a reação de um derivado de benzila representado pela seguinte fórmula geral (1): na qual x^ 1^ representa um átomo de halogênio e r^ 1^ representa um grupo acila, com um composto de haloacila representado pela fórmula geral (2): r^ 2^-x^ 2^ na qual x^ 2^ representa um átomo de halogênio e r^ 2^ representa um grupo acila, na presença de um ácido de lewis. de acordo com este método, pode ser de preferência preparado um derivado de benzilamina como um intermediário, que é útil para a preparação de um bactericida à base de carbamato para agricultura ou horticultura.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2002376272 | 2002-12-26 | ||
| PCT/JP2003/016995 WO2004058681A1 (ja) | 2002-12-26 | 2003-12-26 | ベンジルアミン誘導体の製造方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0317781B8 true BRPI0317781B8 (pt) | 2019-10-15 |
Family
ID=32677360
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0317781-5B1A BR0317781B1 (pt) | 2002-12-26 | 2003-12-26 | derivado de acilbenzilamina e processos para produção de derivado de benzilamina e de derivado de carbamato |
| BRPI0317781A BRPI0317781B8 (pt) | 2002-12-26 | 2003-12-26 | derivado de acilbenzilamina e processos para produção de derivado de benzilamina e de derivado de carbamato |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0317781-5B1A BR0317781B1 (pt) | 2002-12-26 | 2003-12-26 | derivado de acilbenzilamina e processos para produção de derivado de benzilamina e de derivado de carbamato |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7326813B2 (pt) |
| EP (1) | EP1586552B1 (pt) |
| JP (1) | JP4522263B2 (pt) |
| KR (1) | KR101066433B1 (pt) |
| CN (1) | CN100503551C (pt) |
| AT (1) | ATE478837T1 (pt) |
| AU (1) | AU2003292706B2 (pt) |
| BR (2) | BR0317781B1 (pt) |
| CA (1) | CA2511590C (pt) |
| DE (1) | DE60333950D1 (pt) |
| ES (1) | ES2347329T3 (pt) |
| IL (1) | IL169393A (pt) |
| MX (1) | MXPA05006938A (pt) |
| NZ (1) | NZ541392A (pt) |
| PL (1) | PL207186B1 (pt) |
| RU (1) | RU2362766C2 (pt) |
| TW (1) | TWI325415B (pt) |
| WO (1) | WO2004058681A1 (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008124092A2 (en) | 2007-04-03 | 2008-10-16 | E. I. Du Pont De Nemours And Company | Substituted benzene fungicides |
| TW201116212A (en) | 2009-10-29 | 2011-05-16 | Du Pont | Heterobicycle-substituted azolyl benzene fungicides |
| JP2013018767A (ja) * | 2011-06-03 | 2013-01-31 | Sumitomo Chemical Co Ltd | ベンジルアミン化合物を製造する方法 |
| WO2015157005A1 (en) | 2014-04-10 | 2015-10-15 | E I Du Pont De Nemours And Company | Substituted tolyl fungicide mixtures |
| TWI832917B (zh) | 2018-11-06 | 2024-02-21 | 美商富曼西公司 | 經取代之甲苯基殺真菌劑 |
| PY2133975A (es) | 2020-05-06 | 2022-01-19 | Fmc Corp | Fungicidas de tolilo sustituido y sus mezclas |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4566901A (en) | 1982-05-06 | 1986-01-28 | Ciba-Geigy Corporation | Novel oxime ethers, the preparation thereof, compositions containing them and the use thereof |
| FR2559766B1 (fr) | 1984-02-16 | 1986-05-16 | Poudres & Explosifs Ste Nale | Procede de preparation de derives de l'acide carbamique |
| IL74272A (en) | 1984-02-16 | 1991-06-10 | Poudres & Explosifs Ste Nale | Preparation of carbamic acid derivatives |
| US4968829A (en) | 1984-07-18 | 1990-11-06 | Sandoz Ltd. | Novel substituted aromatic compounds |
| US5663199A (en) | 1994-11-30 | 1997-09-02 | Uniroyal Chemical Ltd./Ltee | Anti-viral aromatic O-alkylated oximes, ethers and thioethers |
| US5817814A (en) | 1997-05-01 | 1998-10-06 | Fmc Corporation | Method for the preparation of benzyluracils |
| UA73307C2 (uk) * | 1999-08-05 | 2005-07-15 | Куміаі Кемікал Індастрі Ко., Лтд. | Похідна карбамату і фунгіцид сільськогосподарського/садівницького призначення |
| US6531291B1 (en) | 1999-11-10 | 2003-03-11 | The Trustees Of Columbia University In The City Of New York | Antimicrobial activity of gemfibrozil and related compounds and derivatives and metabolites thereof |
| JP4246996B2 (ja) | 2001-02-02 | 2009-04-02 | クミアイ化学工業株式会社 | イミノオキシメチルピリジン化合物及び農園芸用殺菌剤 |
-
2003
- 2003-12-26 KR KR1020057012006A patent/KR101066433B1/ko not_active Expired - Fee Related
- 2003-12-26 CN CNB2003801089811A patent/CN100503551C/zh not_active Expired - Lifetime
- 2003-12-26 NZ NZ541392A patent/NZ541392A/en not_active IP Right Cessation
- 2003-12-26 DE DE60333950T patent/DE60333950D1/de not_active Expired - Lifetime
- 2003-12-26 AU AU2003292706A patent/AU2003292706B2/en not_active Ceased
- 2003-12-26 ES ES03768351T patent/ES2347329T3/es not_active Expired - Lifetime
- 2003-12-26 TW TW092137078A patent/TWI325415B/zh not_active IP Right Cessation
- 2003-12-26 BR BRPI0317781-5B1A patent/BR0317781B1/pt active IP Right Grant
- 2003-12-26 US US10/540,749 patent/US7326813B2/en not_active Expired - Fee Related
- 2003-12-26 MX MXPA05006938A patent/MXPA05006938A/es active IP Right Grant
- 2003-12-26 AT AT03768351T patent/ATE478837T1/de active
- 2003-12-26 EP EP03768351A patent/EP1586552B1/en not_active Expired - Lifetime
- 2003-12-26 JP JP2004562958A patent/JP4522263B2/ja not_active Expired - Lifetime
- 2003-12-26 RU RU2005123690/04A patent/RU2362766C2/ru not_active IP Right Cessation
- 2003-12-26 CA CA2511590A patent/CA2511590C/en not_active Expired - Fee Related
- 2003-12-26 BR BRPI0317781A patent/BRPI0317781B8/pt not_active IP Right Cessation
- 2003-12-26 PL PL377143A patent/PL207186B1/pl unknown
- 2003-12-26 WO PCT/JP2003/016995 patent/WO2004058681A1/ja not_active Ceased
-
2005
- 2005-06-26 IL IL169393A patent/IL169393A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| EP1586552A1 (en) | 2005-10-19 |
| JP4522263B2 (ja) | 2010-08-11 |
| IL169393A (en) | 2010-06-30 |
| KR101066433B1 (ko) | 2011-09-23 |
| PL377143A1 (pl) | 2006-01-23 |
| MXPA05006938A (es) | 2005-10-26 |
| US7326813B2 (en) | 2008-02-05 |
| WO2004058681A1 (ja) | 2004-07-15 |
| ES2347329T3 (es) | 2010-10-28 |
| TWI325415B (en) | 2010-06-01 |
| RU2005123690A (ru) | 2006-01-20 |
| CN100503551C (zh) | 2009-06-24 |
| CN1802343A (zh) | 2006-07-12 |
| PL207186B1 (pl) | 2010-11-30 |
| DE60333950D1 (de) | 2010-10-07 |
| JPWO2004058681A1 (ja) | 2006-04-27 |
| AU2003292706A1 (en) | 2004-07-22 |
| NZ541392A (en) | 2008-06-30 |
| BR0317781A (pt) | 2005-11-22 |
| TW200418764A (en) | 2004-10-01 |
| CA2511590A1 (en) | 2004-07-15 |
| AU2003292706B2 (en) | 2010-01-21 |
| CA2511590C (en) | 2011-12-20 |
| RU2362766C2 (ru) | 2009-07-27 |
| US20060155141A1 (en) | 2006-07-13 |
| EP1586552A4 (en) | 2007-03-14 |
| EP1586552B1 (en) | 2010-08-25 |
| KR20050088227A (ko) | 2005-09-02 |
| BR0317781B1 (pt) | 2013-10-01 |
| ATE478837T1 (de) | 2010-09-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B21A | Patent or certificate of addition expired [chapter 21.1 patent gazette] |
Free format text: PATENTE EXTINTA EM 26/12/2023 |