BRPI0411484A - composto, formulação farmacêutica, métodos de tratamento ou prevenção de distúrbios de lipìdeo (dislipidemia), e de diabetes do tipo 2, uso de um composto, e, composição farmacêutica - Google Patents

composto, formulação farmacêutica, métodos de tratamento ou prevenção de distúrbios de lipìdeo (dislipidemia), e de diabetes do tipo 2, uso de um composto, e, composição farmacêutica

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Publication number
BRPI0411484A
BRPI0411484A BRPI0411484-1A BRPI0411484A BRPI0411484A BR PI0411484 A BRPI0411484 A BR PI0411484A BR PI0411484 A BRPI0411484 A BR PI0411484A BR PI0411484 A BRPI0411484 A BR PI0411484A
Authority
BR
Brazil
Prior art keywords
compound
methods
diabetes
lipid disorders
type
Prior art date
Application number
BRPI0411484-1A
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English (en)
Inventor
Lanna Li
Christina Olsson
Eva-Lotte Lindstedt Alstermark
Original Assignee
Astrazeneca Ab
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27636750&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0411484(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI0411484A publication Critical patent/BRPI0411484A/pt

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    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/02—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C233/11—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to carbon atoms of an unsaturated carbon skeleton containing six-membered aromatic rings
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
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    • C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
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    • C07C233/51—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
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Abstract

"COMPOSTO, FORMULAçãO FARMACêUTICA, MéTODOS DE TRATAMENTO OU PREVENçãO DE DISTúRBIOS DE LIPìDEO (DISLIPIDEMIA), E DE DIABETES DO TIPO 2, USO DE UM COMPOSTO E, COMPOSIçãO FARMACêUTICA" A presente invenção refere-se a um composto da fórmula (I), a processos para preparar tais compostos, a sua utilidade no tratamento de condições clinicas que incluem distúrbios de lipideo (dislipideminas), estejam ou não associadas com a resistência à insulina, métodos para o seu uso terapêutico e a composições farmacêuticas contendo o mesmo.
BRPI0411484-1A 2003-06-18 2004-06-17 composto, formulação farmacêutica, métodos de tratamento ou prevenção de distúrbios de lipìdeo (dislipidemia), e de diabetes do tipo 2, uso de um composto, e, composição farmacêutica BRPI0411484A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0314079.5A GB0314079D0 (en) 2003-06-18 2003-06-18 Therapeutic agents
PCT/EP2004/006597 WO2004113270A2 (en) 2003-06-18 2004-06-17 Propionic acid derivatives useful in the treatment of lipid disorders

Publications (1)

Publication Number Publication Date
BRPI0411484A true BRPI0411484A (pt) 2006-07-25

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BRPI0411484-1A BRPI0411484A (pt) 2003-06-18 2004-06-17 composto, formulação farmacêutica, métodos de tratamento ou prevenção de distúrbios de lipìdeo (dislipidemia), e de diabetes do tipo 2, uso de um composto, e, composição farmacêutica

Country Status (22)

Country Link
US (4) US20050148656A1 (pt)
EP (2) EP1676833A1 (pt)
JP (2) JP2006527730A (pt)
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