BRPI0414500A - formulação farmacêutica composição para tratar uma infecção vaginal, e, métodos para tratar uma infecção vaginal, para estabilizar uma formulação de clindamicina, para tratar ou prevenir uma recorrência de uma infecção vaginal em uma paciente e para tratar condições vaginais - Google Patents

formulação farmacêutica composição para tratar uma infecção vaginal, e, métodos para tratar uma infecção vaginal, para estabilizar uma formulação de clindamicina, para tratar ou prevenir uma recorrência de uma infecção vaginal em uma paciente e para tratar condições vaginais

Info

Publication number
BRPI0414500A
BRPI0414500A BRPI0414500-3A BRPI0414500A BRPI0414500A BR PI0414500 A BRPI0414500 A BR PI0414500A BR PI0414500 A BRPI0414500 A BR PI0414500A BR PI0414500 A BRPI0414500 A BR PI0414500A
Authority
BR
Brazil
Prior art keywords
treat
vaginal
vaginal infection
infection
formulation
Prior art date
Application number
BRPI0414500-3A
Other languages
English (en)
Inventor
Thomas Riley
R Saul Levinson
Robert C Cuca
Elio Mariani
Original Assignee
Drugtech Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Drugtech Corp filed Critical Drugtech Corp
Publication of BRPI0414500A publication Critical patent/BRPI0414500A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0034Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
    • A61K9/0036Devices retained in the vagina or cervix for a prolonged period, e.g. intravaginal rings, medicated tampons, medicated diaphragms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0034Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/02Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

"FORMULAçãO FARMACêUTICA COMPOSIçãO PARA TRATAR UMA INFECçãO VAGINAL, E, MéTODOS PARA TRATAR UMA INFECçãO VAGINAL, PARA ESTABILIZAR UMA FORMULAçãO DE CLINDAMICINA, PARA TRATAR OU PREVENIR UMA RECORRêNCIA DE UMA INFECçãO VAGINAL EM UMA PACIENTE E PARA TRATAR CONDIçõES VAGINAIS". Uma formulação farmacêutica para tratar condições vaginais em uma paciente humana compreende: pelo menos um agente ativo; uma forma de dosagem de liberação modificada que proporciona liberação prolongada de agente anti-infeccioso sob administração vaginal ao paciente; e na qual a formulação, quando contiver uma dose total de agente anti-infeccioso de cerca de 25 <109>g a cerca de 500 mg baseada no agente ativo produzirá uma curva de concentração plásmica versus tempo (ng/mL versus horas) possuindo uma área sob a curva (AUC) menor do que cerca de 600 ng/mL.h.
BRPI0414500-3A 2003-09-19 2004-09-20 formulação farmacêutica composição para tratar uma infecção vaginal, e, métodos para tratar uma infecção vaginal, para estabilizar uma formulação de clindamicina, para tratar ou prevenir uma recorrência de uma infecção vaginal em uma paciente e para tratar condições vaginais BRPI0414500A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US50401703P 2003-09-19 2003-09-19
US50713803P 2003-10-01 2003-10-01
PCT/US2004/030672 WO2005027807A1 (en) 2003-09-19 2004-09-20 Pharmaceutical delivery system

Publications (1)

Publication Number Publication Date
BRPI0414500A true BRPI0414500A (pt) 2006-11-07

Family

ID=34381092

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0414500-3A BRPI0414500A (pt) 2003-09-19 2004-09-20 formulação farmacêutica composição para tratar uma infecção vaginal, e, métodos para tratar uma infecção vaginal, para estabilizar uma formulação de clindamicina, para tratar ou prevenir uma recorrência de uma infecção vaginal em uma paciente e para tratar condições vaginais

Country Status (11)

Country Link
US (2) US20050095245A1 (pt)
EP (1) EP1667619A4 (pt)
JP (1) JP2007505927A (pt)
CN (1) CN1852690B (pt)
AR (1) AR047108A1 (pt)
AU (1) AU2004274000B2 (pt)
BR (1) BRPI0414500A (pt)
CA (1) CA2540129A1 (pt)
MY (1) MY144021A (pt)
SG (1) SG146638A1 (pt)
WO (1) WO2005027807A1 (pt)

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Also Published As

Publication number Publication date
EP1667619A1 (en) 2006-06-14
US20130102548A1 (en) 2013-04-25
US20050095245A1 (en) 2005-05-05
CN1852690B (zh) 2010-04-14
AU2004274000A1 (en) 2005-03-31
US9789057B2 (en) 2017-10-17
EP1667619A4 (en) 2007-10-10
CN1852690A (zh) 2006-10-25
AU2004274000B2 (en) 2009-07-30
CA2540129A1 (en) 2005-03-31
AR047108A1 (es) 2006-01-11
MY144021A (en) 2011-07-29
WO2005027807A1 (en) 2005-03-31
SG146638A1 (en) 2008-10-30
JP2007505927A (ja) 2007-03-15

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