BRPI0513310A - análogos de tetrapeptìdeo - Google Patents

análogos de tetrapeptìdeo

Info

Publication number
BRPI0513310A
BRPI0513310A BRPI0513310-6A BRPI0513310A BRPI0513310A BR PI0513310 A BRPI0513310 A BR PI0513310A BR PI0513310 A BRPI0513310 A BR PI0513310A BR PI0513310 A BRPI0513310 A BR PI0513310A
Authority
BR
Brazil
Prior art keywords
tetrapeptide analogs
tetrapeptide
analogs
tetrapeptid
cancer
Prior art date
Application number
BRPI0513310-6A
Other languages
English (en)
Inventor
Bin Chao
Thomas L Deckwerth
Paul S Furth
Steven D Linton
Alfred P Spada
Brett R Ullman
Michael I Weinhouse
Original Assignee
Idun Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idun Pharmaceuticals Inc filed Critical Idun Pharmaceuticals Inc
Publication of BRPI0513310A publication Critical patent/BRPI0513310A/pt

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    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
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    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/06—Tripeptides
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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
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Abstract

ANáLOGOS DE TETRAPEPTìDEO Compostos, composições e métodos para tratamento de doenças hiperproliferativas, como câncer, são fornecidos.
BRPI0513310-6A 2004-07-12 2005-07-12 análogos de tetrapeptìdeo BRPI0513310A (pt)

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BRPI0511350A (pt) * 2004-07-02 2007-12-04 Genentech Inc composto, métodos de indução da apoptose em uma célula, de sensibilização de uma célula à um sinal apoptótico, de inibição da ligação de uma proteìna iap e de tratamento de uma doença e cáncer e usos de um composto

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CR8919A (es) 2007-08-31
EP1773348A4 (en) 2009-05-20
WO2006017295A3 (en) 2007-07-12
JP2011102312A (ja) 2011-05-26
AU2005271831A1 (en) 2006-02-16
EA200700225A1 (ru) 2008-02-28
JP2008505976A (ja) 2008-02-28
EP1773348A2 (en) 2007-04-18
IL180677A0 (en) 2008-04-13
NO20070782L (no) 2007-04-02
TNSN07005A1 (fr) 2008-06-02
ZA200700357B (en) 2008-11-26
GB0700629D0 (en) 2007-02-21
WO2006017295A2 (en) 2006-02-16
EP2457896A1 (en) 2012-05-30
KR20070043831A (ko) 2007-04-25
US20100190688A1 (en) 2010-07-29
EP2457895A1 (en) 2012-05-30
MX2007000490A (es) 2007-06-11
CA2573644A1 (en) 2006-02-16
GB2430935A (en) 2007-04-11
MA28841B1 (fr) 2007-09-03

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