BRPI0513848A - formulação de pélete de liberação prolongada contendo pramipexol ou um sal farmaceuticamente aceitável deste, método para fabricação da mesma e uso desta - Google Patents

formulação de pélete de liberação prolongada contendo pramipexol ou um sal farmaceuticamente aceitável deste, método para fabricação da mesma e uso desta

Info

Publication number
BRPI0513848A
BRPI0513848A BRPI0513848-5A BRPI0513848A BRPI0513848A BR PI0513848 A BRPI0513848 A BR PI0513848A BR PI0513848 A BRPI0513848 A BR PI0513848A BR PI0513848 A BRPI0513848 A BR PI0513848A
Authority
BR
Brazil
Prior art keywords
pharmaceutically acceptable
pramipexole
acceptable salt
prolonged
release pellet
Prior art date
Application number
BRPI0513848-5A
Other languages
English (en)
Inventor
Thomas Friedl
Rolf-Stefan Brickl
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34926162&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0513848(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of BRPI0513848A publication Critical patent/BRPI0513848A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Psychology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

FORMULAçãO DE PéLETE DE LIBERAçãO PROLONGADA CONTENDO PRAMIPEXOL OU UM SAL FARMACEUTICAMENTE ACEITáVEL DESTE, MéTODO PARA FABRICAçãO DA MESMA E USO DESTA. A presente invenção refere-se a um pélete de liberação prolongada compreendendo um ingrediente ativo selecionado de pramipexol e os sais farmaceuticamente aceitáveis deste, e pelo menos um excipiente modificador de liberação.
BRPI0513848-5A 2004-08-13 2005-07-25 formulação de pélete de liberação prolongada contendo pramipexol ou um sal farmaceuticamente aceitável deste, método para fabricação da mesma e uso desta BRPI0513848A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04019249 2004-08-13
PCT/EP2005/053609 WO2006015943A2 (en) 2004-08-13 2005-07-25 Extended release pellet formulation containing pramipexole or a pharmaceutically acceptable salt thereof, method for manufacturing the same and use thereof

Publications (1)

Publication Number Publication Date
BRPI0513848A true BRPI0513848A (pt) 2008-05-20

Family

ID=34926162

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0513848-5A BRPI0513848A (pt) 2004-08-13 2005-07-25 formulação de pélete de liberação prolongada contendo pramipexol ou um sal farmaceuticamente aceitável deste, método para fabricação da mesma e uso desta

Country Status (19)

Country Link
US (3) US20060051419A1 (pt)
EP (3) EP2431027A1 (pt)
JP (1) JP4971159B2 (pt)
KR (2) KR20070050081A (pt)
CN (3) CN101022788B (pt)
AU (1) AU2005271193B2 (pt)
BR (1) BRPI0513848A (pt)
CA (1) CA2576386A1 (pt)
EA (2) EA201001086A1 (pt)
EC (1) ECSP077243A (pt)
EG (1) EG26209A (pt)
IL (1) IL181281A0 (pt)
MX (1) MX2007001850A (pt)
NO (1) NO20070944L (pt)
NZ (1) NZ553645A (pt)
SG (1) SG164375A1 (pt)
UA (3) UA97084C2 (pt)
WO (1) WO2006015943A2 (pt)
ZA (1) ZA200700313B (pt)

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