BRPI0509394A - derivados de diazina, sua manufatura e uso como agentes farmacêuticos - Google Patents

derivados de diazina, sua manufatura e uso como agentes farmacêuticos

Info

Publication number
BRPI0509394A
BRPI0509394A BRPI0509394-5A BRPI0509394A BRPI0509394A BR PI0509394 A BRPI0509394 A BR PI0509394A BR PI0509394 A BRPI0509394 A BR PI0509394A BR PI0509394 A BRPI0509394 A BR PI0509394A
Authority
BR
Brazil
Prior art keywords
manufacture
pharmaceutical agents
compounds
diazine derivatives
diazine
Prior art date
Application number
BRPI0509394-5A
Other languages
English (en)
Inventor
Birgit Bossenmaier
Walter-Gunar Friebe
Wolfgang Jenni
Matthias Rueth
Edgar Voss
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34924554&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0509394(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BRPI0509394A publication Critical patent/BRPI0509394A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Catalysts (AREA)

Abstract

"DERIVADOS DE DIAZINA, SUA MANUFATURA E USO COMO AGENTES FARMACêUTICOS". Os objetivos da presente invenção são os compostos de fórmula (I), os seus sais farmaceuticamente aceitáveis, formas enantioméricas, diastereoisómeros e racematos, a preparação dos compostos acima mencionados, os medicamentos que os contêm e a sua manufatura, bem como o usa dos compostos acima mencionados no controle ou na prevenção de doenças, tais como o câncer.
BRPI0509394-5A 2004-04-02 2005-03-31 derivados de diazina, sua manufatura e uso como agentes farmacêuticos BRPI0509394A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04008130 2004-04-02
PCT/EP2005/003347 WO2005097785A1 (en) 2004-04-02 2005-03-31 Novel diazine derivatives, their manufacture and use as pharmaceutical agents

Publications (1)

Publication Number Publication Date
BRPI0509394A true BRPI0509394A (pt) 2007-09-18

Family

ID=34924554

Family Applications (2)

Application Number Title Priority Date Filing Date
BRPI0509394-5A BRPI0509394A (pt) 2004-04-02 2005-03-31 derivados de diazina, sua manufatura e uso como agentes farmacêuticos
BRPI0509360-0A BRPI0509360A (pt) 2004-04-02 2005-03-31 processo para preparação de derivados de diazina

Family Applications After (1)

Application Number Title Priority Date Filing Date
BRPI0509360-0A BRPI0509360A (pt) 2004-04-02 2005-03-31 processo para preparação de derivados de diazina

Country Status (12)

Country Link
US (2) US20080132699A1 (pt)
EP (2) EP1758897A1 (pt)
JP (2) JP2007530627A (pt)
KR (2) KR20060131958A (pt)
CN (2) CN1934102A (pt)
AR (1) AR048455A1 (pt)
AU (2) AU2005231937A1 (pt)
BR (2) BRPI0509394A (pt)
CA (2) CA2561203A1 (pt)
RU (2) RU2006138425A (pt)
TW (1) TW200602329A (pt)
WO (2) WO2005097777A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0413605D0 (en) * 2004-06-17 2004-07-21 Addex Pharmaceuticals Sa Novel compounds
WO2010064134A2 (en) * 2008-12-05 2010-06-10 Cadila Pharmaceuticals Ltd. Process of synthesis of paliperidone
US20200077658A1 (en) 2016-12-16 2020-03-12 Basf Se Pesticidal Compounds
CN115353479A (zh) * 2022-07-27 2022-11-18 常州琦诺生物科技有限公司 一种5-溴-2-碘嘧啶的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2952141B2 (ja) * 1993-01-08 1999-09-20 キヤノン株式会社 液晶性化合物、それを含む液晶組成物、及びこれを用いた液晶素子
DE19517186A1 (de) * 1995-05-11 1996-11-14 Bayer Ag Verfahren zur Herstellung substituierter 2-Fluor-pyrimidine
CA2260999C (en) 1996-07-19 2006-07-11 Takeda Chemical Industries, Ltd. Heterocyclic compounds, their production and use in tyrosine kinase inhibition
PE20011178A1 (es) * 2000-04-07 2001-11-19 Takeda Chemical Industries Ltd Compuestos heterociclicos y su produccion
KR20030013360A (ko) * 2000-07-19 2003-02-14 다케다 야쿠힌 고교 가부시키가이샤 1-치환-1,2,3-트리아졸 유도체의 제조 방법
EP1439178A4 (en) 2001-10-05 2005-11-16 Takeda Pharmaceutical Heterocyclic compounds, oxazole derivatives, process for their preparation and their use
JP2003277379A (ja) * 2002-01-17 2003-10-02 Takeda Chem Ind Ltd 含窒素複素環化合物、その製造法および用途
WO2003059907A1 (en) * 2002-01-17 2003-07-24 Takeda Chemical Industries, Ltd. Nitrogenous heterocyclic compounds, process for preparation of the same and use thereof
BR0309671A (pt) 2002-04-25 2005-05-03 Pharmacia Corp ácidos de piperidinil- e piperazinil-sulfonilmetil hidroxâmicos e seu uso como inibidores de protease

Also Published As

Publication number Publication date
AR048455A1 (es) 2006-04-26
US7179812B2 (en) 2007-02-20
JP2007530626A (ja) 2007-11-01
EP1737846A1 (en) 2007-01-03
KR20060131958A (ko) 2006-12-20
KR100843533B1 (ko) 2008-07-03
CA2561206A1 (en) 2005-10-20
WO2005097777A1 (en) 2005-10-20
TW200602329A (en) 2006-01-16
WO2005097785A1 (en) 2005-10-20
AU2005231936A1 (en) 2005-10-20
EP1758897A1 (en) 2007-03-07
US20050222228A1 (en) 2005-10-06
US20080132699A1 (en) 2008-06-05
KR20070006822A (ko) 2007-01-11
CN1934106A (zh) 2007-03-21
RU2006138425A (ru) 2008-06-20
JP2007530627A (ja) 2007-11-01
CA2561203A1 (en) 2005-10-20
RU2006138424A (ru) 2008-05-10
AU2005231937A1 (en) 2005-10-20
CN1934102A (zh) 2007-03-21
BRPI0509360A (pt) 2007-09-11

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A, 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012.