BRPI0618451A2 - derivados de piridopirazina, seu uso, composição farmacêutica e estojo - Google Patents

derivados de piridopirazina, seu uso, composição farmacêutica e estojo Download PDF

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Publication number
BRPI0618451A2
BRPI0618451A2 BRPI0618451-0A BRPI0618451A BRPI0618451A2 BR PI0618451 A2 BRPI0618451 A2 BR PI0618451A2 BR PI0618451 A BRPI0618451 A BR PI0618451A BR PI0618451 A2 BRPI0618451 A2 BR PI0618451A2
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Brazil
Prior art keywords
pharmaceutical composition
kit
derivatives
pyridopyrazine derivatives
pyridopyrazine
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BRPI0618451-0A
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English (en)
Inventor
Irene Seipelt
Eckhard Claus
Eckhard Guenther
Tilmann Schuster
Michael Czech
Emmanuel Polymeropoulos
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Aterna Zentaris Gmbh
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Publication of BRPI0618451A2 publication Critical patent/BRPI0618451A2/pt

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Cardiology (AREA)
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Abstract

DERIVADOS DE PIRIDOPIRAZINA, SEU USO, COMPOSIçãO FARMACêUTICA E ESTOJO. A presente invenção refere-se a novos compostos de piridopirazina, que são adequados para o tratamento ou profilaxia de condições fisiológicas e/ou patofisiológicas induzidas e/ou moduladas por processos de transdução de sinais em mamíferos, especialmente no ser humano.
BRPI0618451-0A 2005-11-11 2006-11-10 derivados de piridopirazina, seu uso, composição farmacêutica e estojo BRPI0618451A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US73570705P 2005-11-11 2005-11-11
EP05024692A EP1790342A1 (de) 2005-11-11 2005-11-11 Pyridopyrazin-Derivate und deren Verwendung als Modulatoren der Signaltransduktionswege
PCT/EP2006/068323 WO2007079999A2 (de) 2005-11-11 2006-11-10 Pyridopyrazin-derivate und deren verwendung als modulatoren der signaltransduktionswege

Publications (1)

Publication Number Publication Date
BRPI0618451A2 true BRPI0618451A2 (pt) 2011-08-30

Family

ID=36424666

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0618451-0A BRPI0618451A2 (pt) 2005-11-11 2006-11-10 derivados de piridopirazina, seu uso, composição farmacêutica e estojo

Country Status (20)

Country Link
US (1) US8937068B2 (pt)
EP (2) EP1790342A1 (pt)
JP (1) JP5448450B2 (pt)
KR (1) KR101473662B1 (pt)
CN (1) CN101330918B (pt)
AR (1) AR056216A1 (pt)
AU (1) AU2006334721B2 (pt)
BR (1) BRPI0618451A2 (pt)
CA (1) CA2628186A1 (pt)
ES (1) ES2543962T3 (pt)
IL (1) IL191160A (pt)
NO (1) NO20082509L (pt)
NZ (1) NZ595879A (pt)
PL (1) PL1962854T3 (pt)
RU (1) RU2487713C2 (pt)
SG (1) SG10201401061XA (pt)
TW (1) TWI423973B (pt)
UA (1) UA95464C2 (pt)
WO (1) WO2007079999A2 (pt)
ZA (1) ZA200803867B (pt)

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UA95464C2 (en) 2011-08-10
EP1962854B1 (de) 2015-05-06
WO2007079999A2 (de) 2007-07-19
IL191160A (en) 2016-03-31
US8937068B2 (en) 2015-01-20
RU2008123219A (ru) 2009-12-20
TW200736253A (en) 2007-10-01
CN101330918A (zh) 2008-12-24
EP1790342A1 (de) 2007-05-30
CN101330918B (zh) 2015-09-02
WO2007079999A3 (de) 2007-10-04
PL1962854T3 (pl) 2015-10-30
SG10201401061XA (en) 2014-07-30
JP2009515854A (ja) 2009-04-16
KR20080068116A (ko) 2008-07-22
RU2487713C2 (ru) 2013-07-20
KR101473662B1 (ko) 2014-12-17
TWI423973B (zh) 2014-01-21
AU2006334721B2 (en) 2011-08-11
JP5448450B2 (ja) 2014-03-19
ES2543962T3 (es) 2015-08-26
NZ595879A (en) 2013-07-26
NO20082509L (no) 2008-07-23
EP1962854A2 (de) 2008-09-03
AR056216A1 (es) 2007-09-26
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US20070123494A1 (en) 2007-05-31
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ZA200803867B (en) 2009-05-27

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