BRPI0819328A2 - Inibidores de replicação de vírus da imunodeficiência humana - Google Patents

Inibidores de replicação de vírus da imunodeficiência humana

Info

Publication number: BRPI0819328A2
Authority: BR; Brazil
Prior art keywords: immunodeficiency virus; human immunodeficiency; virus replication; replication inhibitors; inhibitors
Prior art date: 2007-11-15

Application number

Other languages

English (en)

Inventor

Rebekah J Carson

Lee Fader

Stephen Kawai

Serge Landry

Youla S Tsantrizos

Christian Brochu

Sebastien Morin

Mathieu Parisien

Bruno Simoneau

Original Assignee

Boehringer Ingelheim Int

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-11-15

Filing date

2008-11-03

Publication date

2015-05-12

2008-11-03 Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int

2015-05-12 Publication of BRPI0819328A2 publication Critical patent/BRPI0819328A2/pt

2016-02-10 Publication of BRPI0819328A8 publication Critical patent/BRPI0819328A8/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Virology (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Molecular Biology (AREA)
Chemical Kinetics & Catalysis (AREA)
Tropical Medicine & Parasitology (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
AIDS & HIV (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

BRPI0819328A 2007-11-15 2008-11-03 Compostos inibidores de replicação de vírus da imunodeficiência humana, composição farmacêutica e uso dos ditos compostos BRPI0819328A8 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US98834207P	2007-11-15	2007-11-15
PCT/CA2008/001935 WO2009062288A1 (en)	2007-11-15	2008-11-03	Inhibitors of human immunodeficiency virus replication

Publications (2)

Publication Number	Publication Date
BRPI0819328A2 true BRPI0819328A2 (pt)	2015-05-12
BRPI0819328A8 BRPI0819328A8 (pt)	2016-02-10

Family

ID=40638277

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0819328A BRPI0819328A8 (pt)	2007-11-15	2008-11-03	Compostos inibidores de replicação de vírus da imunodeficiência humana, composição farmacêutica e uso dos ditos compostos

Country Status (18)

Country	Link
US (1)	US7956068B2 (pt)
EP (2)	EP2220095B1 (pt)
JP (1)	JP5269085B2 (pt)
KR (1)	KR20100108337A (pt)
CN (1)	CN102124011A (pt)
AR (1)	AR069334A1 (pt)
AU (1)	AU2008323561B2 (pt)
BR (1)	BRPI0819328A8 (pt)
CA (1)	CA2705312C (pt)
CL (1)	CL2008003405A1 (pt)
ES (1)	ES2402322T3 (pt)
IL (1)	IL205746A0 (pt)
MX (1)	MX2010005292A (pt)
NZ (1)	NZ585297A (pt)
RU (1)	RU2503679C2 (pt)
TW (1)	TW200920363A (pt)
WO (1)	WO2009062288A1 (pt)
ZA (1)	ZA201003305B (pt)

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US8629276B2 (en)	2012-02-15	2014-01-14	Bristol-Myers Squibb Company	Inhibitors of human immunodeficiency virus replication
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UY34750A (es) *	2012-04-20	2013-11-29	Gilead Sciences Inc	?compuestos para el tratamiento del hiv, composiciones,métodos de preparación, intermediarios y métodos terapéuticos?.
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US8906929B2 (en) *	2012-08-16	2014-12-09	Bristol-Myers Squibb Company	Inhibitors of human immunodeficiency virus replication
EP2716639A1 (en)	2012-10-05	2014-04-09	Laboratoire Biodim	Inhibitors of viral replication, their process of preparation and their therapeutical uses
EP2716632A1 (en)	2012-10-05	2014-04-09	Laboratoire Biodim	Inhibitors of viral replication, their process of preparation and their therapeutical uses
EP2719685A1 (en)	2012-10-11	2014-04-16	Laboratoire Biodim	Inhibitors of viral replication, their process of preparation and their therapeutical uses
TW201441197A (zh)	2013-01-31	2014-11-01	Shionogi & Co	Ｈｉｖ複製抑制劑
WO2014164467A1 (en)	2013-03-13	2014-10-09	Bristol-Myers Squibb Company	Inhibitors of human immunodeficiency virus replication
ES2619708T3 (es)	2013-03-13	2017-06-26	VIIV Healthcare UK (No.5) Limited	Inhibidores de la replicación del virus de inmunodeficiencia humana
WO2014164409A1 (en)	2013-03-13	2014-10-09	Bristol-Myers Squibb Company	Inhibitors of human immunodeficiency virus replication
JP2016512558A (ja)	2013-03-14	2016-04-28	ブリストル−マイヤーズスクイブカンパニーＢｒｉｓｔｏｌ−ＭｙｅｒｓＳｑｕｉｂｂＣｏｍｐａｎｙ	ヒト免疫不全ウイルス複製の阻害剤
CN105008369B (zh)	2013-03-14	2017-07-11	百时美施贵宝公司	人类免疫缺陷病毒复制抑制剂
US9908893B2 (en)	2013-06-11	2018-03-06	Latvian Institute Of Organic Synthesis	Thieno [2,3-b] pyridines as multidrug resistance modulators
EP2821104A1 (en)	2013-07-05	2015-01-07	Laboratoire Biodim	Inhibitors of viral replication, their process of preparation and their therapeutical uses
EP2821082A1 (en)	2013-07-05	2015-01-07	Laboratoire Biodim	Method of producing an inactivated lentivirus, especially HIV, vaccine, kit and method of use
EP3105236B1 (en)	2014-02-12	2017-10-18	ViiV Healthcare UK (No.5) Limited	Benzothiazole macrocycles as inhibitors of human immunodeficiency virus replication
WO2015126758A1 (en)	2014-02-18	2015-08-27	Bristol-Myers Squibb Company	Imidazopyrimidine macrocycles as inhibitors of human immunodeficiency virus replication
US9409922B2 (en)	2014-02-18	2016-08-09	Bristol-Myers Squibb Company	Imidazopyridine macrocycles as inhibitors of human immunodeficiency virus replication
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TWI700284B (zh)	2015-05-29	2020-08-01	日商塩野義製藥股份有限公司	具有ｈｉｖ複製抑制作用之含氮３環性衍生物
US20180170903A1 (en)	2015-07-06	2018-06-21	VIIV Healthcare UK (No.5) Limited	Pyridin-3-yl acetic acid derivatives as inhibitors of human immunodeficiency virus replication
RU2018102554A (ru)	2015-07-08	2019-08-08	ВАЙВ ХЕЛТКЕР ЮКей (N5) ЛИМИТЕД	Производные пиридин-3-ил уксусной кислоты в качестве ингибиторов репликации вируса иммунодефицита человека
US20180170904A1 (en)	2015-07-09	2018-06-21	VIIV Healthcare UK (No.5) Limited	Pyridin-3-yl acetic acid derivatives as inhibitors of human immunodeficiency virus replication
RU2018103031A (ru)	2015-07-09	2019-08-09	ВАЙВ ХЕЛТКЕР ЮКей (N5) ЛИМИТЕД	Производные пиридин-3-ил уксусной кислоты в качестве ингибиторов репликации вируса иммунодефицита человека
KR20180035910A (ko)	2015-08-07	2018-04-06	비브 헬스케어 유케이 (넘버5) 리미티드	인간 면역결핍 바이러스 복제의 억제제로서 피리딘-3-일 아세트산 유도체
WO2017025913A1 (en)	2015-08-10	2017-02-16	VIIV Healthcare UK (No.5) Limited	Imidazopyridine macrocycles as inhibitors of human immunodeficiency virus replication
TWI657086B (zh)	2015-08-11	2019-04-21	英商Viiv醫療保健英國(No.5)有限公司	做為人類免疫缺陷病毒複製抑制劑之５－（ｎ－苯甲基四氫異喹啉－６－基）吡啶－３－基乙酸衍生物
CN108137553A (zh)	2015-08-12	2018-06-08	Viiv保健英国第五有限公司	作为人免疫缺陷病毒复制的抑制剂的5-(n-[6,5]-稠合双环芳基四氢异喹啉-6-基)吡啶-3-基乙酸衍生物
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JP2019515000A (ja)	2016-05-11	2019-06-06	ヴィーブヘルスケアユーケー（ナンバー５）リミテッド	ヒト免疫不全ウイルス複製の阻害剤としてのピリジン−３−イル酢酸誘導体
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CN109641822B (zh) *	2016-08-12	2022-03-11	拜耳作物科学股份公司	制备取代苯乙烯衍生物的方法
EP3565810A1 (en)	2017-01-03	2019-11-13	ViiV Healthcare UK (No.5) Limited	Pyridin-3-yl acetic acid derivatives as inhibitors of human immunodeficiency virus replication
TW201835068A (zh)	2017-01-03	2018-10-01	英商Viiv醫療保健英國(No.5)有限公司	作為人類免疫缺乏病毒複製之抑制劑之吡啶-3-基乙酸衍生物
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WO2020003093A1 (en)	2018-06-25	2020-01-02	VIIV Healthcare UK (No.5) Limited	Pyridin-3-yl acetic acid derivatives as inhibitors of human immunodeficiency virus replication
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2008
- 2008-11-03 ES ES08850892T patent/ES2402322T3/es active Active
- 2008-11-03 KR KR1020107013084A patent/KR20100108337A/ko not_active Ceased
- 2008-11-03 NZ NZ585297A patent/NZ585297A/en not_active IP Right Cessation
- 2008-11-03 WO PCT/CA2008/001935 patent/WO2009062288A1/en not_active Ceased
- 2008-11-03 EP EP08850892A patent/EP2220095B1/en active Active
- 2008-11-03 BR BRPI0819328A patent/BRPI0819328A8/pt not_active IP Right Cessation
- 2008-11-03 CN CN2008801247470A patent/CN102124011A/zh active Pending
- 2008-11-03 MX MX2010005292A patent/MX2010005292A/es active IP Right Grant
- 2008-11-03 US US12/743,143 patent/US7956068B2/en active Active
- 2008-11-03 AU AU2008323561A patent/AU2008323561B2/en not_active Ceased
- 2008-11-03 CA CA2705312A patent/CA2705312C/en not_active Expired - Fee Related
- 2008-11-03 JP JP2010533394A patent/JP5269085B2/ja active Active
- 2008-11-03 RU RU2010123989/04A patent/RU2503679C2/ru not_active IP Right Cessation
- 2008-11-03 EP EP12199561A patent/EP2574610A1/en not_active Withdrawn
- 2008-11-14 TW TW097144270A patent/TW200920363A/zh unknown
- 2008-11-14 AR ARP080104989A patent/AR069334A1/es not_active Application Discontinuation
- 2008-11-14 CL CL2008003405A patent/CL2008003405A1/es unknown
2010
- 2010-05-11 ZA ZA2010/03305A patent/ZA201003305B/en unknown
- 2010-05-13 IL IL205746A patent/IL205746A0/en unknown

Also Published As

Publication number	Publication date
RU2503679C2 (ru)	2014-01-10
TW200920363A (en)	2009-05-16
MX2010005292A (es)	2010-07-05
EP2220095A1 (en)	2010-08-25
WO2009062288A1 (en)	2009-05-22
US20100305115A1 (en)	2010-12-02
ZA201003305B (en)	2011-03-30
ES2402322T3 (es)	2013-04-30
CN102124011A (zh)	2011-07-13
CA2705312C (en)	2013-06-25
AU2008323561A1 (en)	2009-05-22
EP2220095B1 (en)	2013-01-02
IL205746A0 (en)	2010-11-30
BRPI0819328A8 (pt)	2016-02-10
EP2220095A4 (en)	2011-01-26
EP2574610A1 (en)	2013-04-03
US7956068B2 (en)	2011-06-07
RU2010123989A (ru)	2011-12-20
JP2011503117A (ja)	2011-01-27
JP5269085B2 (ja)	2013-08-21
NZ585297A (en)	2012-06-29
CA2705312A1 (en)	2009-05-22
AU2008323561B2 (en)	2013-07-18
KR20100108337A (ko)	2010-10-06
CL2008003405A1 (es)	2010-02-12
AR069334A1 (es)	2010-01-13

Publication	Publication Date	Title
BRPI0819328A2 (pt)	2015-05-12	Inibidores de replicação de vírus da imunodeficiência humana
BRPI0820307A2 (pt)	2019-09-24	inibidores de replicação do vírus da imunodeficiência humana
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