BRPI0821160A2 - Octahidroquinolizinas, composição farmacêutica contendo as mesmas e uso de ditos compostos - Google Patents
Octahidroquinolizinas, composição farmacêutica contendo as mesmas e uso de ditos compostosInfo
- Publication number
- BRPI0821160A2 BRPI0821160A2 BRPI0821160-4A BRPI0821160A BRPI0821160A2 BR PI0821160 A2 BRPI0821160 A2 BR PI0821160A2 BR PI0821160 A BRPI0821160 A BR PI0821160A BR PI0821160 A2 BRPI0821160 A2 BR PI0821160A2
- Authority
- BR
- Brazil
- Prior art keywords
- octahidroquinolizines
- compounds
- pharmaceutical composition
- composition containing
- containing same
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/02—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Cardiology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Heart & Thoracic Surgery (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07450235A EP2072515B1 (en) | 2007-12-19 | 2007-12-19 | Substituted quinazolidines for antidiabetic treatment |
| AT13152008 | 2008-08-25 | ||
| PCT/AT2008/000458 WO2009076693A1 (en) | 2007-12-19 | 2008-12-17 | Octahydroquinoli zines for antidiabetic treatment |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0821160A2 true BRPI0821160A2 (pt) | 2015-06-16 |
Family
ID=40430049
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0821160-4A BRPI0821160A2 (pt) | 2007-12-19 | 2008-12-17 | Octahidroquinolizinas, composição farmacêutica contendo as mesmas e uso de ditos compostos |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20110003808A1 (pt) |
| EP (1) | EP2222673A1 (pt) |
| JP (1) | JP2011506485A (pt) |
| KR (1) | KR20100107469A (pt) |
| CN (1) | CN101918402A (pt) |
| AP (1) | AP2010005317A0 (pt) |
| AU (1) | AU2008338287B2 (pt) |
| BR (1) | BRPI0821160A2 (pt) |
| CA (1) | CA2710006A1 (pt) |
| EA (1) | EA201070750A1 (pt) |
| IL (1) | IL205752A0 (pt) |
| MA (1) | MA32012B1 (pt) |
| MX (1) | MX2010006173A (pt) |
| NZ (1) | NZ585307A (pt) |
| WO (1) | WO2009076693A1 (pt) |
| ZA (1) | ZA201003316B (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010022412A1 (en) * | 2008-08-25 | 2010-03-04 | 55Pharma Drug Discovery & Development Ag | Octahydroquinolizines for antidiabetic treatment |
| JP6520440B2 (ja) * | 2014-06-16 | 2019-05-29 | 有限会社バイオシステムコンサルティング | 新規化合物 |
| CN110746282A (zh) * | 2019-11-04 | 2020-02-04 | 天津市安凯特科技发展有限公司 | 一种4-氯-2-丁酮的合成方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA795318B (en) * | 1978-10-13 | 1980-09-24 | Hoffmann La Roche | Phenyl quinolizidines |
| US7538110B2 (en) * | 2005-10-27 | 2009-05-26 | Adolor Corporation | Opioid antagonists |
-
2008
- 2008-12-17 BR BRPI0821160-4A patent/BRPI0821160A2/pt not_active IP Right Cessation
- 2008-12-17 US US12/809,513 patent/US20110003808A1/en not_active Abandoned
- 2008-12-17 MX MX2010006173A patent/MX2010006173A/es active IP Right Grant
- 2008-12-17 AU AU2008338287A patent/AU2008338287B2/en not_active Expired - Fee Related
- 2008-12-17 WO PCT/AT2008/000458 patent/WO2009076693A1/en not_active Ceased
- 2008-12-17 KR KR1020107015983A patent/KR20100107469A/ko not_active Withdrawn
- 2008-12-17 EP EP08862420A patent/EP2222673A1/en not_active Withdrawn
- 2008-12-17 EA EA201070750A patent/EA201070750A1/ru unknown
- 2008-12-17 CN CN2008801225325A patent/CN101918402A/zh active Pending
- 2008-12-17 JP JP2010538265A patent/JP2011506485A/ja active Pending
- 2008-12-17 NZ NZ585307A patent/NZ585307A/en not_active IP Right Cessation
- 2008-12-17 AP AP2010005317A patent/AP2010005317A0/en unknown
- 2008-12-17 CA CA2710006A patent/CA2710006A1/en not_active Abandoned
-
2010
- 2010-05-11 ZA ZA2010/03316A patent/ZA201003316B/en unknown
- 2010-05-13 IL IL205752A patent/IL205752A0/en unknown
- 2010-07-14 MA MA33011A patent/MA32012B1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU2008338287B2 (en) | 2012-06-07 |
| WO2009076693A1 (en) | 2009-06-25 |
| EA201070750A1 (ru) | 2010-12-30 |
| KR20100107469A (ko) | 2010-10-05 |
| JP2011506485A (ja) | 2011-03-03 |
| US20110003808A1 (en) | 2011-01-06 |
| AU2008338287A1 (en) | 2009-06-25 |
| MX2010006173A (es) | 2010-09-30 |
| EP2222673A1 (en) | 2010-09-01 |
| CA2710006A1 (en) | 2009-06-25 |
| ZA201003316B (en) | 2011-08-31 |
| MA32012B1 (fr) | 2011-01-03 |
| CN101918402A (zh) | 2010-12-15 |
| IL205752A0 (en) | 2010-11-30 |
| AP2010005317A0 (en) | 2010-08-31 |
| NZ585307A (en) | 2011-11-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 5A, 6A E 7A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2343 DE 01-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |