BRPI0823378A2 - análogos de glucagon - Google Patents

análogos de glucagon

Info

Publication number: BRPI0823378A2
Authority: BR; Brazil
Prior art keywords: glucagon analogs; glucagon; analogs
Prior art date: 2008-12-15

Application number

BRPI0823378A

Other languages

English (en)

Inventor

Due Larsen Bjarne

Riber Ditte

Meier Eddi

Rosengren Daugaard Jens

Skovgaard Marie

Original Assignee

Zealand Pharma As

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-12-15

Filing date

2008-12-15

Publication date

2019-09-24

2008-12-15 Application filed by Zealand Pharma As filed Critical Zealand Pharma As

2019-09-24 Publication of BRPI0823378A2 publication Critical patent/BRPI0823378A2/pt

Links

MASNOZXLGMXCHN-ZLPAWPGGSA-N glucagon Chemical class C([C@@H](C(=O)N[C@H](C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H]([C@@H](C)O)C(O)=O)C(C)C)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CO)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CO)NC(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CC=1C=CC=CC=1)NC(=O)[C@@H](NC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC=1NC=NC=1)[C@@H](C)O)[C@@H](C)O)C1=CC=CC=C1 MASNOZXLGMXCHN-ZLPAWPGGSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12N—MICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
- C12N15/00—Mutation or genetic engineering; DNA or RNA concerning genetic engineering, vectors, e.g. plasmids, or their isolation, preparation or purification; Use of hosts therefor
- C12N15/09—Recombinant DNA-technology
- C12N15/11—DNA or RNA fragments; Modified forms thereof; Non-coding nucleic acids having a biological activity
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Diabetes (AREA)
Genetics & Genomics (AREA)
Endocrinology (AREA)
Zoology (AREA)
Gastroenterology & Hepatology (AREA)
Molecular Biology (AREA)
Hematology (AREA)
Obesity (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biophysics (AREA)
Biochemistry (AREA)
Biomedical Technology (AREA)
Toxicology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Biotechnology (AREA)
General Engineering & Computer Science (AREA)
Wood Science & Technology (AREA)
Emergency Medicine (AREA)
Immunology (AREA)
Epidemiology (AREA)
Vascular Medicine (AREA)
Microbiology (AREA)
Child & Adolescent Psychology (AREA)
Neurosurgery (AREA)

BRPI0823378A 2008-12-15 2008-12-15 análogos de glucagon BRPI0823378A2 (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/GB2008/004121 WO2010070251A1 (en)	2008-12-15	2008-12-15	Glucagon analogues

Publications (1)

Publication Number	Publication Date
BRPI0823378A2 true BRPI0823378A2 (pt)	2019-09-24

Family

ID=40428061

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0823378A BRPI0823378A2 (pt)	2008-12-15	2008-12-15	análogos de glucagon

Country Status (19)

Country	Link
US (2)	US8685919B2 (pt)
EP (2)	EP2370459A1 (pt)
JP (1)	JP5635529B2 (pt)
KR (2)	KR20150116912A (pt)
CN (1)	CN102282167B (pt)
AP (1)	AP2011005774A0 (pt)
AU (1)	AU2008365555B2 (pt)
BR (1)	BRPI0823378A2 (pt)
CA (1)	CA2747109A1 (pt)
EA (1)	EA020537B1 (pt)
HK (1)	HK1203531A1 (pt)
IL (1)	IL213477A0 (pt)
MA (1)	MA32970B1 (pt)
MX (1)	MX2011006313A (pt)
MY (1)	MY160219A (pt)
SG (1)	SG172170A1 (pt)
TN (1)	TN2011000295A1 (pt)
UA (1)	UA104605C2 (pt)
WO (1)	WO2010070251A1 (pt)

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2008
- 2008-12-15 EA EA201190047A patent/EA020537B1/ru not_active IP Right Cessation
- 2008-12-15 KR KR1020157027018A patent/KR20150116912A/ko not_active Ceased
- 2008-12-15 US US13/139,493 patent/US8685919B2/en not_active Expired - Fee Related
- 2008-12-15 AU AU2008365555A patent/AU2008365555B2/en not_active Ceased
- 2008-12-15 MY MYPI2011002751A patent/MY160219A/en unknown
- 2008-12-15 BR BRPI0823378A patent/BRPI0823378A2/pt not_active IP Right Cessation
- 2008-12-15 EP EP08875670A patent/EP2370459A1/en not_active Withdrawn
- 2008-12-15 UA UAA201108817A patent/UA104605C2/uk unknown
- 2008-12-15 CN CN200880132682.4A patent/CN102282167B/zh not_active Expired - Fee Related
- 2008-12-15 SG SG2011043700A patent/SG172170A1/en unknown
- 2008-12-15 WO PCT/GB2008/004121 patent/WO2010070251A1/en not_active Ceased
- 2008-12-15 CA CA2747109A patent/CA2747109A1/en not_active Abandoned
- 2008-12-15 KR KR1020117016184A patent/KR20110126589A/ko not_active Ceased
- 2008-12-15 AP AP2011005774A patent/AP2011005774A0/xx unknown
- 2008-12-15 JP JP2011540187A patent/JP5635529B2/ja not_active Expired - Fee Related
- 2008-12-15 EP EP14175826.8A patent/EP2799447B1/en active Active
- 2008-12-15 MX MX2011006313A patent/MX2011006313A/es active IP Right Grant
- 2008-12-15 MA MA34020A patent/MA32970B1/fr unknown
2011
- 2011-06-10 TN TN2011000295A patent/TN2011000295A1/fr unknown
- 2011-06-12 IL IL213477A patent/IL213477A0/en unknown
2014
- 2014-03-03 US US14/195,533 patent/US20150080295A1/en not_active Abandoned
2015
- 2015-05-05 HK HK15104289.5A patent/HK1203531A1/en unknown

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Publication number	Publication date
CA2747109A1 (en)	2010-06-24
JP2012511899A (ja)	2012-05-31
US20110286982A1 (en)	2011-11-24
CN102282167A (zh)	2011-12-14
TN2011000295A1 (en)	2012-12-17
EA020537B1 (ru)	2014-11-28
EP2370459A1 (en)	2011-10-05
WO2010070251A1 (en)	2010-06-24
JP5635529B2 (ja)	2014-12-03
EP2799447B1 (en)	2016-11-23
AU2008365555A1 (en)	2011-07-21
EP2799447A3 (en)	2014-12-31
KR20150116912A (ko)	2015-10-16
US20150080295A1 (en)	2015-03-19
SG172170A1 (en)	2011-07-28
AU2008365555B2 (en)	2016-01-14
MA32970B1 (fr)	2012-01-02
KR20110126589A (ko)	2011-11-23
EA201190047A1 (ru)	2012-02-28
MX2011006313A (es)	2011-09-27
AP2011005774A0 (en)	2011-06-30
HK1203531A1 (en)	2015-10-30
MY160219A (en)	2017-02-28
CN102282167B (zh)	2014-08-13
EP2799447A2 (en)	2014-11-05
US8685919B2 (en)	2014-04-01
IL213477A0 (en)	2011-07-31
UA104605C2 (uk)	2014-02-25

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2019-10-01	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
2020-01-21	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2543 DE 01-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

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