BRPI0906248A2 - composto, composição farmacêutica para inibir a formação de microtúbulos e método para preparar um composto - Google Patents

composto, composição farmacêutica para inibir a formação de microtúbulos e método para preparar um composto

Info

Publication number
BRPI0906248A2
BRPI0906248A2 BRPI0906248A BRPI0906248A BRPI0906248A2 BR PI0906248 A2 BRPI0906248 A2 BR PI0906248A2 BR PI0906248 A BRPI0906248 A BR PI0906248A BR PI0906248 A BRPI0906248 A BR PI0906248A BR PI0906248 A2 BRPI0906248 A2 BR PI0906248A2
Authority
BR
Brazil
Prior art keywords
compound
preparing
pharmaceutical composition
microtubule formation
inhibiting microtubule
Prior art date
Application number
BRPI0906248A
Other languages
English (en)
Inventor
Byeong-Hoon Han
Dal-Hyun Kim
Gyu-Tae Park
Hee-Ryong Kang
Ho-Jin Choi
Jae-Hoon Choi
Jae-Kwang Lee
Kyung-Joo Lee
Nam-Song-Choi
Seung-Kee Moon
Soo-Jin Kim
Soon-Kil Ahn
Su-Yeal Bae
Sung-Sook Lee
Young-Hoon Kim
Original Assignee
Chong Kun Dang Pharm Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chong Kun Dang Pharm Corp filed Critical Chong Kun Dang Pharm Corp
Publication of BRPI0906248A2 publication Critical patent/BRPI0906248A2/pt
Publication of BRPI0906248B1 publication Critical patent/BRPI0906248B1/pt
Publication of BRPI0906248B8 publication Critical patent/BRPI0906248B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
BRPI0906248A 2008-03-26 2009-03-05 composto, composição farmacêutica para inibir a formação de microtúbulos e método para preparar um composto BRPI0906248B8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR20080027820 2008-03-26
PCT/KR2009/001095 WO2009119980A2 (ko) 2008-03-26 2009-03-05 미세소관 형성 저해제로서 유용한 벤조페논 티아졸 유도체 및 이의 제조 방법

Publications (3)

Publication Number Publication Date
BRPI0906248A2 true BRPI0906248A2 (pt) 2016-10-25
BRPI0906248B1 BRPI0906248B1 (pt) 2020-01-21
BRPI0906248B8 BRPI0906248B8 (pt) 2021-05-25

Family

ID=41114435

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0906248A BRPI0906248B8 (pt) 2008-03-26 2009-03-05 composto, composição farmacêutica para inibir a formação de microtúbulos e método para preparar um composto

Country Status (15)

Country Link
US (1) US8362267B2 (pt)
EP (1) EP2272845B1 (pt)
JP (1) JP5378499B2 (pt)
KR (1) KR101069735B1 (pt)
CN (1) CN101981029B (pt)
AU (1) AU2009229709B2 (pt)
BR (1) BRPI0906248B8 (pt)
CA (1) CA2719243C (pt)
DK (1) DK2272845T3 (pt)
ES (1) ES2536794T3 (pt)
HU (1) HUE025268T2 (pt)
MX (1) MX2010010561A (pt)
PL (1) PL2272845T3 (pt)
PT (1) PT2272845E (pt)
WO (1) WO2009119980A2 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2019517506A (ja) * 2016-07-29 2019-06-24 チョン クン ダン ファーマシューティカル コーポレーション 血管破壊剤を含む肝臓癌治療用の組成物
US9980953B2 (en) * 2016-09-26 2018-05-29 Chong Kun Dang Pharmaceutical Corp. Combined composition for preventing or treating cancer comprising a benzophenone thiazole derivatives as a VDA and topoisomerase inhibitor
CN107163011B (zh) * 2017-05-27 2019-10-01 上海应用技术大学 3-(3,4,5-三甲氧基苯甲酰)-苯并呋喃类微管蛋白抑制剂及其制备方法和用途
JP6956254B2 (ja) * 2017-07-26 2021-11-02 チョン クン ダン ファーマシューティカル コーポレーション 血管遮断剤および免疫チェックポイント阻害剤を含む癌の予防または治療用の組成物
KR102216772B1 (ko) 2018-05-18 2021-02-17 주식회사 종근당 혈관차단제 및 탁산 화합물을 포함하는 암 예방 또는 치료용 조성물

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA05009434A (es) 2003-03-05 2005-11-23 Celgene Corp Compuestos de difeniletileno y usos de los mismos.
RU2396250C2 (ru) * 2003-07-24 2010-08-10 Лео Фарма А/С Новые производные аминобензофенона
EP1828148B1 (en) 2004-12-13 2010-01-20 Leo Pharma A/S Triazole substituted aminobenzophenone compounds
KR100932093B1 (ko) * 2006-09-27 2009-12-16 주식회사종근당 미세소관 형성 저해제로서 유용한 벤조페논 유도체

Also Published As

Publication number Publication date
US8362267B2 (en) 2013-01-29
PL2272845T3 (pl) 2015-08-31
BRPI0906248B8 (pt) 2021-05-25
CA2719243C (en) 2013-06-25
KR101069735B1 (ko) 2011-10-04
EP2272845B1 (en) 2015-03-04
DK2272845T3 (en) 2015-05-04
PT2272845E (pt) 2015-06-01
JP5378499B2 (ja) 2013-12-25
AU2009229709A1 (en) 2009-10-01
CN101981029A (zh) 2011-02-23
HUE025268T2 (en) 2016-02-29
CN101981029B (zh) 2014-04-02
WO2009119980A2 (ko) 2009-10-01
EP2272845A2 (en) 2011-01-12
MX2010010561A (es) 2010-10-25
BRPI0906248B1 (pt) 2020-01-21
WO2009119980A3 (ko) 2009-12-17
US20110021582A1 (en) 2011-01-27
AU2009229709B2 (en) 2011-12-08
CA2719243A1 (en) 2009-10-01
JP2011515461A (ja) 2011-05-19
KR20090102639A (ko) 2009-09-30
ES2536794T3 (es) 2015-05-28
EP2272845A4 (en) 2014-01-01

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Legal Events

Date Code Title Description
B25D Requested change of name of applicant approved

Owner name: CHONG KUN DANG HOLDINGS CORP. (KR)

B25A Requested transfer of rights approved

Owner name: CHONG KUN DANG PHARMACEUTICAL CORP. (KR)

B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 21/01/2020, OBSERVADAS AS CONDICOES LEGAIS.

B16C Correction of notification of the grant [chapter 16.3 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 05/03/2009 OBSERVADAS AS CONDICOES LEGAIS. PATENTE CONCEDIDA CONFORME ADI 5.529/DF