BRPI0907364A2 - Antagonistas aminoalquilbifenil n,n-disubstituídos de receptores d2 de prostaglandina - Google Patents
Antagonistas aminoalquilbifenil n,n-disubstituídos de receptores d2 de prostaglandinaInfo
- Publication number
- BRPI0907364A2 BRPI0907364A2 BRPI0907364-7A BRPI0907364A BRPI0907364A2 BR PI0907364 A2 BRPI0907364 A2 BR PI0907364A2 BR PI0907364 A BRPI0907364 A BR PI0907364A BR PI0907364 A2 BRPI0907364 A2 BR PI0907364A2
- Authority
- BR
- Brazil
- Prior art keywords
- prostaglandin
- receptor antagonists
- aminoalkylbiphenyl
- disubstituted
- disubstituted aminoalkylbiphenyl
- Prior art date
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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- C07C323/62—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
- C07C323/63—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/04—Systems containing only non-condensed rings with a four-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
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| US11049608P | 2008-10-31 | 2008-10-31 | |
| PCT/US2009/032499 WO2009099902A1 (en) | 2008-02-01 | 2009-01-29 | N,n-disubstituted aminoalkylbiphenyl antagonists of prostaglandin d2 receptors |
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| US8426449B2 (en) | 2008-04-02 | 2013-04-23 | Panmira Pharmaceuticals, Llc | Aminoalkylphenyl antagonists of prostaglandin D2 receptors |
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- 2009-01-29 EA EA201001253A patent/EA018901B1/ru not_active IP Right Cessation
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- 2009-01-29 EP EP09709250.6A patent/EP2257524B1/en active Active
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2010
- 2010-07-21 IL IL207130A patent/IL207130A/en active IP Right Grant
- 2010-07-27 CO CO10091359A patent/CO6290752A2/es active IP Right Grant
- 2010-07-30 DO DO2010000234A patent/DOP2010000234A/es unknown
- 2010-08-06 CR CR11621A patent/CR11621A/es not_active Application Discontinuation
- 2010-09-01 EC EC2010010439A patent/ECSP10010439A/es unknown
-
2011
- 2011-10-12 US US13/272,180 patent/US8362044B2/en not_active Expired - Fee Related
- 2011-11-15 US US13/297,160 patent/US8338484B2/en not_active Expired - Fee Related
-
2012
- 2012-11-01 US US13/666,703 patent/US20130158036A1/en not_active Abandoned
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