BRPI0907892A2 - Composto antibiótico azatricíclico, medicamento, composição farmacêutica que o contém e uso do mesmo - Google Patents
Composto antibiótico azatricíclico, medicamento, composição farmacêutica que o contém e uso do mesmoInfo
- Publication number
- BRPI0907892A2 BRPI0907892A2 BRPI0907892-4A BRPI0907892A BRPI0907892A2 BR PI0907892 A2 BRPI0907892 A2 BR PI0907892A2 BR PI0907892 A BRPI0907892 A BR PI0907892A BR PI0907892 A2 BRPI0907892 A2 BR PI0907892A2
- Authority
- BR
- Brazil
- Prior art keywords
- medicine
- pharmaceutical composition
- composition containing
- antibiotic compound
- azatricyclic
- Prior art date
Links
- 230000003115 biocidal effect Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/16—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/03—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/04—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/16—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IB2008050603 | 2008-02-20 | ||
| IB2008054065 | 2008-10-03 | ||
| PCT/IB2009/050675 WO2009104147A2 (en) | 2008-02-20 | 2009-02-19 | Azatricyclic antibiotic compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0907892A2 true BRPI0907892A2 (pt) | 2015-07-28 |
Family
ID=40986002
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0907892-4A BRPI0907892A2 (pt) | 2008-02-20 | 2009-02-19 | Composto antibiótico azatricíclico, medicamento, composição farmacêutica que o contém e uso do mesmo |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US8349828B2 (pt) |
| EP (1) | EP2257551B1 (pt) |
| JP (1) | JP5349500B2 (pt) |
| KR (1) | KR101590202B1 (pt) |
| CN (1) | CN102015710B (pt) |
| AR (1) | AR070455A1 (pt) |
| AU (1) | AU2009215327A1 (pt) |
| BR (1) | BRPI0907892A2 (pt) |
| CA (1) | CA2713182C (pt) |
| ES (1) | ES2411930T3 (pt) |
| MX (1) | MX2010008922A (pt) |
| RU (1) | RU2010138648A (pt) |
| TW (1) | TW200940551A (pt) |
| WO (1) | WO2009104147A2 (pt) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8349828B2 (en) | 2008-02-20 | 2013-01-08 | Actelion Pharmaceuticals Ltd. | Azatricyclic antibiotic compounds |
| PT2344495E (pt) * | 2008-10-07 | 2015-04-01 | Actelion Pharmaceuticals Ltd | Compostos antibióticos de oxazolidinona tricíclica |
| EP2346862B1 (en) * | 2008-10-10 | 2012-09-12 | Actelion Pharmaceuticals Ltd. | 2-benzothiophenyl-and 2-naphthyl-0xaz0lidin0nes and their azaisostere analogues as antibacterial agents |
| JPWO2012108376A1 (ja) | 2011-02-07 | 2014-07-03 | 第一三共株式会社 | アミノ基含有ピロリジノン誘導体 |
| CN105949466A (zh) * | 2011-06-30 | 2016-09-21 | 帝斯曼知识产权资产管理有限公司 | 含硅酮单体 |
| MX2014001680A (es) | 2011-08-11 | 2014-05-27 | Actelion Pharmaceuticals Ltd | Derivados de quinazolina-2, 4-diona. |
| CN103958525A (zh) | 2011-11-30 | 2014-07-30 | 埃科特莱茵药品有限公司 | 3,7-二取代八氢-2H-吡啶并[4,3-e][1,3]噁嗪-2-酮抗生素 |
| WO2014024056A1 (en) | 2012-08-06 | 2014-02-13 | Daiichi Sankyo Company, Limited | Pyrrolidine derivatives with antibacterial properties |
| ES2640482T3 (es) | 2013-04-16 | 2017-11-03 | Idorsia Pharmaceuticals Ltd | Derivados biaromáticos antibacterianos |
| ITMI20131782A1 (it) * | 2013-10-25 | 2015-04-26 | Dipharma Francis Srl | Procedimento per la preparazione di un agonista della trombopoietina |
| JP6112724B2 (ja) * | 2013-10-31 | 2017-04-12 | 日本化薬株式会社 | １，５−ナフチリジン誘導体およびそれを有効成分として含んでなる殺虫剤 |
| AR102256A1 (es) | 2014-10-15 | 2017-02-15 | Actelion Pharmaceuticals Ltd | Derivados biaromáticos básicos antibacterianos con sustitución de aminoalcoxi |
| TW201833120A (zh) | 2017-02-17 | 2018-09-16 | 瑞士商愛杜西亞製藥有限公司 | 芳基噁唑啶酮抗生素化合物 |
| CN111527093B (zh) * | 2017-11-29 | 2023-06-09 | 巴格沃克斯研究有限公司 | 抗菌杂环化合物及其合成 |
Family Cites Families (43)
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|---|---|---|---|---|
| JPS5746987A (en) * | 1980-09-05 | 1982-03-17 | Mitsubishi Chem Ind Ltd | 3,4-dihydrocarbostyril derivative and agricultural and horticultural germicide containing the same as active constituent |
| IT1212552B (it) | 1982-10-20 | 1989-11-30 | Italo Britannica L Manet Ti H | Alcanolaminossi derivati di 3,4-diidro-2h-1.4-benzotiazin-3-one, loro procedimento di produzione e loro utilizzazione farmaceutica |
| US5298518A (en) | 1989-09-29 | 1994-03-29 | Eisai Co., Ltd. | Biphenylmethane derivative and pharmacological use |
| US5254682A (en) | 1989-12-08 | 1993-10-19 | Merck & Co., Inc. | Cyclic renin inhibitors containing 3(S)-amino-4-cyclohexyl-2(R)-hydroxy-butanoic acid or 4-cyclo-hexyl-(2R, 3S)-dihydroxybutanoic acid or related analogs |
| RU2181362C2 (ru) | 1996-10-24 | 2002-04-20 | Новартис Аг | Производные аминофосфоновых и -фосфиновых кислот, способ их получения и фармацевтические составы на их основе |
| AU1026901A (en) | 1999-10-29 | 2001-05-08 | Syngenta Participations Ag | Novel herbicides |
| TW200409637A (en) | 2002-06-26 | 2004-06-16 | Glaxo Group Ltd | Compounds |
| WO2005016883A2 (en) | 2003-08-14 | 2005-02-24 | Icos Corporation | Acrylamide derivatives as vla-1 integrin antagonists and uses thereof |
| WO2006024741A2 (fr) | 2004-07-30 | 2006-03-09 | Palumed S.A. | Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien |
| FR2873695A1 (fr) * | 2004-07-30 | 2006-02-03 | Palumed Sa | Molecules hybrides qa ou q est une aminoquinoleine et a est un antibiotique ou un inhibiteur de resistance), leur synthese et leurs utilisations en tant qu'agent antibacterien |
| DE102004041163A1 (de) | 2004-08-25 | 2006-03-02 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Neue Verbindungen mit antibakterieller Aktivität |
| CA2580621A1 (en) | 2004-09-24 | 2006-03-30 | Actelion Pharmaceuticals Ltd | New bicyclic antibiotics |
| JP5314244B2 (ja) | 2004-10-27 | 2013-10-16 | 富山化学工業株式会社 | 新規な含窒素複素環化合物およびその塩 |
| WO2006125974A1 (en) | 2005-05-24 | 2006-11-30 | Astrazeneca Ab | Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity |
| WO2007016610A2 (en) | 2005-08-02 | 2007-02-08 | Glaxo Group Limited | Antibacterial agents |
| AU2006335042A1 (en) | 2005-10-21 | 2007-07-19 | Glaxo Group Limited | Compounds |
| ES2344523T3 (es) * | 2005-12-22 | 2010-08-30 | Glaxo Group Limited | Compuestos heterociclicos, su preparacion y su uso como agentes antibacterianos. |
| US20090318431A1 (en) * | 2006-02-14 | 2009-12-24 | Pfizer Inc. | Benzoxazinone and benzoxazepinone oxazolidinones as antibacterial agents |
| ATE469649T1 (de) | 2006-03-23 | 2010-06-15 | Actelion Pharmaceuticals Ltd | Antibiotische cyclohexyl- oder piperidinylcarboxamid-derivate |
| ATE481406T1 (de) | 2006-04-06 | 2010-10-15 | Glaxo Group Ltd | Pyrrolochinoxalinonderivate als antibakterielle mittel |
| GB0608263D0 (en) | 2006-04-26 | 2006-06-07 | Glaxo Group Ltd | Compounds |
| PL2032551T3 (pl) | 2006-06-16 | 2012-01-31 | Pharma Mar Sa | Przeciwnowotworowe związki dihydropiran-2-onu |
| GB0613208D0 (en) | 2006-07-03 | 2006-08-09 | Glaxo Group Ltd | Compounds |
| TW200819457A (en) | 2006-08-30 | 2008-05-01 | Actelion Pharmaceuticals Ltd | Spiro antibiotic derivatives |
| JP2010511018A (ja) | 2006-12-01 | 2010-04-08 | ガラパゴス・ナムローゼ・フェンノートシャップ | 変性疾患及び炎症性疾患の治療に有用なトリアゾロピリジン化合物 |
| CL2007003693A1 (es) | 2006-12-22 | 2008-06-27 | Actelion Pharmaceuticals Ltd | Compuestos derivados de pirido [3,2-b] [1,4] tiazina; composicion farmaceutica que contiene dichos compuestos; y su uso en el tratamiento de infecciones bacterianas. |
| GB0705672D0 (en) | 2007-03-23 | 2007-05-02 | Glaxo Group Ltd | Compounds |
| US7998992B2 (en) | 2007-03-30 | 2011-08-16 | Institute Of Medicinal Molecular Design, Inc. | Oxazolidinone derivative having inhibitory activity on 11β-hydroxysteroid dehydrogenase type 1 |
| WO2008120003A1 (en) | 2007-04-03 | 2008-10-09 | Astrazeneca Ab | Substituted piperidines for use in the treatment of bacterial infections |
| CL2008001002A1 (es) | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
| CL2008001003A1 (es) | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
| EP1980251A1 (en) | 2007-04-13 | 2008-10-15 | Glaxo Group Limited | Pyrrolo[3,2,1-ij]quinoline-4-one derivatives for treating tuberculosis |
| GB0707708D0 (en) | 2007-04-20 | 2007-05-30 | Glaxo Group Ltd | Compounds |
| JP5389013B2 (ja) | 2007-04-20 | 2014-01-15 | グラクソ グループ リミテッド | 抗菌剤としての三環式含窒素化合物 |
| GB0707706D0 (en) | 2007-04-20 | 2007-05-30 | Glaxo Group Ltd | Compounds |
| WO2008150827A1 (en) | 2007-05-29 | 2008-12-11 | Smithkline Beecham Corporation | Naphthyridine, derivatives as p13 kinase inhibitors |
| AR066879A1 (es) | 2007-06-08 | 2009-09-16 | Novartis Ag | Derivados de quinoxalina como inhibidores de la actividad de cinasa de tirosina de las cinasas janus |
| JP5274553B2 (ja) | 2007-06-15 | 2013-08-28 | アクテリオン ファーマシューティカルズ リミテッド | ３−アミノ−６−（１−アミノ−エチル）−テトラヒドロピラン誘導体 |
| EP2005995A1 (en) | 2007-06-22 | 2008-12-24 | Glaxo Group Limited | Heterocyclic compounds for the treatment of tuberculosis |
| JP5323088B2 (ja) | 2007-12-18 | 2013-10-23 | アクテリオン ファーマシューティカルズ リミテッド | ５−アミノシクリルメチル−オキサゾリジン−２−オン誘導体 |
| GB0800367D0 (en) | 2008-01-09 | 2008-02-20 | Glaxo Group Ltd | Compounds |
| US8349828B2 (en) | 2008-02-20 | 2013-01-08 | Actelion Pharmaceuticals Ltd. | Azatricyclic antibiotic compounds |
| ES2398939T3 (es) | 2008-02-22 | 2013-03-22 | Actelion Pharmaceuticals Ltd. | Derivados de oxazolidinona |
-
2009
- 2009-02-19 US US12/918,749 patent/US8349828B2/en not_active Expired - Fee Related
- 2009-02-19 BR BRPI0907892-4A patent/BRPI0907892A2/pt not_active IP Right Cessation
- 2009-02-19 CN CN2009801060558A patent/CN102015710B/zh not_active Expired - Fee Related
- 2009-02-19 KR KR1020107019907A patent/KR101590202B1/ko not_active Expired - Fee Related
- 2009-02-19 RU RU2010138648/04A patent/RU2010138648A/ru unknown
- 2009-02-19 ES ES09712156T patent/ES2411930T3/es active Active
- 2009-02-19 WO PCT/IB2009/050675 patent/WO2009104147A2/en not_active Ceased
- 2009-02-19 CA CA2713182A patent/CA2713182C/en not_active Expired - Fee Related
- 2009-02-19 TW TW098105338A patent/TW200940551A/zh unknown
- 2009-02-19 EP EP09712156.0A patent/EP2257551B1/en not_active Not-in-force
- 2009-02-19 MX MX2010008922A patent/MX2010008922A/es not_active Application Discontinuation
- 2009-02-19 AU AU2009215327A patent/AU2009215327A1/en not_active Abandoned
- 2009-02-19 JP JP2010547289A patent/JP5349500B2/ja not_active Expired - Fee Related
- 2009-02-20 AR ARP090100595A patent/AR070455A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2411930T3 (es) | 2013-07-09 |
| CN102015710B (zh) | 2013-04-24 |
| AR070455A1 (es) | 2010-04-07 |
| MX2010008922A (es) | 2010-09-07 |
| JP2011512398A (ja) | 2011-04-21 |
| KR20100124273A (ko) | 2010-11-26 |
| US8349828B2 (en) | 2013-01-08 |
| WO2009104147A2 (en) | 2009-08-27 |
| KR101590202B1 (ko) | 2016-01-29 |
| JP5349500B2 (ja) | 2013-11-20 |
| EP2257551B1 (en) | 2013-04-10 |
| WO2009104147A3 (en) | 2009-11-05 |
| US20100331318A1 (en) | 2010-12-30 |
| CN102015710A (zh) | 2011-04-13 |
| TW200940551A (en) | 2009-10-01 |
| CA2713182A1 (en) | 2009-08-27 |
| RU2010138648A (ru) | 2012-03-27 |
| EP2257551A2 (en) | 2010-12-08 |
| CA2713182C (en) | 2016-09-13 |
| AU2009215327A1 (en) | 2009-08-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 4A, 5A E 6A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2344 DE 08-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |