BRPI0912074A2 - composto e composição farmacêutica - Google Patents

composto e composição farmacêutica

Info

Publication number: BRPI0912074A2
Authority: BR; Brazil
Prior art keywords: compound; pharmaceutical composition; pharmaceutical; composition
Prior art date: 2008-08-12

Application number

Other languages

English (en)

Inventor

Mark L Greenlee

Robert WILKENING

James Apgar

Kenneth James Wildonger

Dongfang Meng

Dann L Parker Jr

Original Assignee

Merck Sharp & Dohme

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-08-12

Filing date

2009-08-07

Publication date

2018-10-02

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41669132&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0912074(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2009-08-07 Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme

2018-10-02 Publication of BRPI0912074A2 publication Critical patent/BRPI0912074A2/pt

2021-08-03 Publication of BRPI0912074B1 publication Critical patent/BRPI0912074B1/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
- A01N43/647—Triazoles; Hydrogenated triazoles
- A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4196—1,2,4-Triazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
- C07J63/008—Expansion of ring D by one atom, e.g. D homo steroids

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Wood Science & Technology (AREA)
General Chemical & Material Sciences (AREA)
Plant Pathology (AREA)
Engineering & Computer Science (AREA)
Dentistry (AREA)
Agronomy & Crop Science (AREA)
Zoology (AREA)
Environmental Sciences (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
Pest Control & Pesticides (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Steroid Compounds (AREA)
Peptides Or Proteins (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Cosmetics (AREA)

BRPI0912074-2A 2008-08-12 2009-08-07 Composto e composição farmacêutica BRPI0912074B1 (pt)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US13610608P	2008-08-12	2008-08-12
US61/136,106		2008-08-12
PCT/US2009/004557 WO2010019203A1 (en)	2008-08-12	2009-08-07	Antifungal agents

Publications (2)

Publication Number	Publication Date
BRPI0912074A2 true BRPI0912074A2 (pt)	2018-10-02
BRPI0912074B1 BRPI0912074B1 (pt)	2021-08-03

Family

ID=41669132

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0912074-2A BRPI0912074B1 (pt)	2008-08-12	2009-08-07	Composto e composição farmacêutica

Country Status (30)

Country	Link
EP (1)	EP2326172B1 (pt)
KR (1)	KR101686075B1 (pt)
AR (1)	AR073037A1 (pt)
BR (1)	BRPI0912074B1 (pt)
CL (1)	CL2011000292A1 (pt)
CO (1)	CO6351686A2 (pt)
CR (1)	CR20110075A (pt)
DK (1)	DK2326172T3 (pt)
DO (1)	DOP2011000053A (pt)
EA (1)	EA018337B1 (pt)
ES (1)	ES2526652T3 (pt)
GT (1)	GT201100039A (pt)
HN (1)	HN2011000404A (pt)
HR (1)	HRP20150009T1 (pt)
IL (2)	IL210975A (pt)
MA (1)	MA32628B1 (pt)
MX (1)	MX2011001656A (pt)
MY (1)	MY156955A (pt)
NI (1)	NI201100035A (pt)
NZ (1)	NZ590914A (pt)
PE (1)	PE20110676A1 (pt)
PL (1)	PL2326172T3 (pt)
PT (1)	PT2326172E (pt)
RS (1)	RS53731B1 (pt)
SI (1)	SI2326172T1 (pt)
SV (1)	SV2011003839A (pt)
TW (1)	TWI439458B (pt)
UA (1)	UA105639C2 (pt)
WO (1)	WO2010019203A1 (pt)
ZA (1)	ZA201100788B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SI3247711T1 (sl)	2015-01-19	2022-07-29	Scynexis, Inc.	Nove soli in polimorfi SCY-078
EA201992413A1 (ru) *	2017-04-10	2020-03-16	Сайнексис, Инк.	Противогрибковые средства, используемые в комбинации
KR102807716B1 (ko) *	2017-08-04	2025-05-13	싸이넥시스, 인크.	산성 pH에서 증진된 활성을 갖는 항진균제
JP7562542B2 (ja) *	2019-01-30	2024-10-07	サイネクシス，インコーポレーテッド	真菌性骨－関節感染症を治療するためのトリテルペノイド系抗真菌薬
IL288165B2 (en) *	2019-05-16	2026-05-01	Scynexis Inc	Antifungal agents for decolonization of Candida auris
US20230218652A1 (en)	2020-05-29	2023-07-13	Centre National De La Recherche Scientifique	Antifungal prodrugs

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5756472A (en)	1996-01-31	1998-05-26	Merck & Co., Inc.	Antifungal agent obtained from hormonema
CA2244142C (en) *	1996-01-31	2005-03-29	Merck & Co., Inc.	Antifungal compound from hormonema sp.
EP1497281A4 (en) *	2002-04-17	2005-11-02	Ranbaxy Lab Ltd	AZOLE DERIVATIVES AS ANTIFUNGAL AGENTS
WO2007127012A1 (en) *	2006-04-03	2007-11-08	Merck & Co., Inc.	Antifungal agents

2009
- 2009-08-07 EA EA201100350A patent/EA018337B1/ru unknown
- 2009-08-07 MY MYPI2011000483A patent/MY156955A/en unknown
- 2009-08-07 BR BRPI0912074-2A patent/BRPI0912074B1/pt active IP Right Grant
- 2009-08-07 KR KR1020117005837A patent/KR101686075B1/ko active Active
- 2009-08-07 HR HRP20150009AT patent/HRP20150009T1/hr unknown
- 2009-08-07 EP EP09806944.6A patent/EP2326172B1/en active Active
- 2009-08-07 UA UAA201102860A patent/UA105639C2/uk unknown
- 2009-08-07 WO PCT/US2009/004557 patent/WO2010019203A1/en not_active Ceased
- 2009-08-07 NZ NZ590914A patent/NZ590914A/en unknown
- 2009-08-07 ES ES09806944.6T patent/ES2526652T3/es active Active
- 2009-08-07 RS RS20150006A patent/RS53731B1/sr unknown
- 2009-08-07 MX MX2011001656A patent/MX2011001656A/es active IP Right Grant
- 2009-08-07 SI SI200931102T patent/SI2326172T1/sl unknown
- 2009-08-07 PE PE2011000156A patent/PE20110676A1/es active IP Right Grant
- 2009-08-07 PT PT98069446T patent/PT2326172E/pt unknown
- 2009-08-07 DK DK09806944.6T patent/DK2326172T3/da active
- 2009-08-07 PL PL09806944T patent/PL2326172T3/pl unknown
- 2009-08-10 TW TW098126822A patent/TWI439458B/zh active
- 2009-08-12 AR ARP090103123A patent/AR073037A1/es active IP Right Grant
2011
- 2011-01-31 ZA ZA2011/00788A patent/ZA201100788B/en unknown
- 2011-01-31 IL IL210975A patent/IL210975A/en active IP Right Grant
- 2011-02-08 CR CR20110075A patent/CR20110075A/es unknown
- 2011-02-10 NI NI201100035A patent/NI201100035A/es unknown
- 2011-02-11 DO DO2011000053A patent/DOP2011000053A/es unknown
- 2011-02-11 CL CL2011000292A patent/CL2011000292A1/es unknown
- 2011-02-11 SV SV2011003839A patent/SV2011003839A/es active IP Right Grant
- 2011-02-11 GT GT201100039A patent/GT201100039A/es unknown
- 2011-02-11 CO CO11016262A patent/CO6351686A2/es active IP Right Grant
- 2011-02-11 HN HN2011000404A patent/HN2011000404A/es unknown
- 2011-03-11 MA MA33691A patent/MA32628B1/fr unknown
2015
- 2015-10-12 IL IL242031A patent/IL242031A0/en unknown

Also Published As

Publication number	Publication date
AR073037A1 (es)	2010-10-06
IL210975A0 (en)	2011-04-28
NZ590914A (en)	2011-11-25
RS53731B1 (sr)	2015-06-30
PT2326172E (pt)	2015-02-04
EP2326172B1 (en)	2014-10-22
KR101686075B1 (ko)	2016-12-13
WO2010019203A8 (en)	2011-03-17
UA105639C2 (uk)	2014-06-10
DK2326172T3 (da)	2015-01-26
EA201100350A1 (ru)	2011-08-30
BRPI0912074B1 (pt)	2021-08-03
CL2011000292A1 (es)	2011-11-04
HN2011000404A (es)	2013-09-23
PE20110676A1 (es)	2011-09-23
PL2326172T3 (pl)	2015-03-31
MY156955A (en)	2016-04-15
MX2011001656A (es)	2011-05-25
WO2010019203A1 (en)	2010-02-18
IL242031A0 (en)	2015-11-30
ES2526652T3 (es)	2015-01-14
CO6351686A2 (es)	2011-12-20
SI2326172T1 (sl)	2015-02-27
EP2326172A4 (en)	2012-06-06
TWI439458B (zh)	2014-06-01
MA32628B1 (fr)	2011-09-01
KR20110045054A (ko)	2011-05-03
TW201011004A (en)	2010-03-16
HK1158017A1 (en)	2012-07-13
HRP20150009T1 (hr)	2015-02-27
EA018337B1 (ru)	2013-07-30
ZA201100788B (en)	2012-05-01
SV2011003839A (es)	2011-07-06
DOP2011000053A (es)	2011-04-30
CR20110075A (es)	2011-06-03
GT201100039A (es)	2013-08-21
IL210975A (en)	2015-10-29
NI201100035A (es)	2011-09-20
EP2326172A1 (en)	2011-06-01

Publication	Publication Date	Title
LTPA2018014I1 (lt)	2018-12-10	Farmacinė kompozicija 514
LTC2140867I2 (lt)	2018-11-12	Farmacinė kompozicija
BRPI0906962A2 (pt)	2015-07-14	Composto, e, composição farmacêutica
BRPI0906556A2 (pt)	2015-07-07	Composto, e, composição farmacêutica
BRPI0721651A2 (pt)	2014-04-01	Composição farmacêutica
BRPI0917681A2 (pt)	2015-08-04	Composto, e, composição farmacêutica
EP2240022A4 (en)	2012-04-25	PHARMACEUTICAL COMPOSITIONS
BRPI0715712A2 (pt)	2014-06-24	Composição farmacêutica
BRPI0719393A2 (pt)	2015-03-31	Composição farmacêutica
DK3492069T3 (da)	2022-03-14	Farmaceutiske sammensætninger omfattende jern-oxy-hydroxid
BRPI0920521A2 (pt)	2018-01-16	combinação farmacêutica
EP2373681A4 (en)	2013-11-06	PHARMACEUTICAL COMPOSITIONS
DK2120884T3 (da)	2011-02-07	Farmaceutisk sammensætning
BRPI0905715A2 (pt)	2015-07-14	Composição farmacêutica e kit de componentes
IT1392101B1 (it)	2012-02-09	Composizione comprendente isoflavoni
DK2285413T3 (da)	2012-08-27	Farmaceutisk sammensætning
DK2285357T3 (da)	2014-06-02	Farmaceutisk sammensætning omfattende brivaracetam
BRPI0819232A2 (pt)	2016-11-01	composto heterocíclico e composição farmacêutica do mesmo
BRPI0908132A2 (pt)	2015-08-04	Composto de benzodiazepina e composição farmacêutica
EP2236149A4 (en)	2012-12-26	MEDICAL COMPOSITION
BRPI0720234A2 (pt)	2013-12-24	Composição farmacêutica
BRPI0716445A2 (pt)	2013-09-17	composiÇço farmacÊutica
BRPI0921313A2 (pt)	2015-12-29	composição farmaucêutica
PT2209464E (pt)	2014-09-05	Composição farmacêutica antimalárica
BRPI0922286A2 (pt)	2015-12-29	composto de quinolona e composição farmacêutica.

Legal Events

Date	Code	Title	Description
2018-10-16	B06F	Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
2020-06-23	B07D	Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]	Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.
2020-09-29	B07E	Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
2020-10-27	B06U	Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
2021-02-17	B06A	Patent application procedure suspended [chapter 6.1 patent gazette]
2021-05-25	B09A	Decision: intention to grant [chapter 9.1 patent gazette]
2021-08-03	B16A	Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]	Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 07/08/2009, OBSERVADAS AS CONDICOES LEGAIS. PATENTE CONCEDIDA CONFORME ADI 5.529/DF, QUE DETERMINA A ALTERACAO DO PRAZO DE CONCESSAO.