BRPI0914238A2 - Processo para a preparação da forma cristalina i de hidrogenossulfato de clopidogrel. - Google Patents

Processo para a preparação da forma cristalina i de hidrogenossulfato de clopidogrel.

Info

Publication number: BRPI0914238A2
Authority: BR; Brazil
Prior art keywords: preparation; crystalline form; clopidogrel hydrogensulfate; hydrogensulfate; clopidogrel
Prior art date: 2008-06-24

Application number

BRPI0914238-0A

Other languages

English (en)

Inventor

Giorgio Soriato

Roberto Brescello

Daniele Urbani

Livius Cotarca

Original Assignee

Zach System Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-06-24

Filing date

2009-06-11

Publication date

2015-08-04

2009-06-11 Application filed by Zach System Spa filed Critical Zach System Spa

2015-08-04 Publication of BRPI0914238A2 publication Critical patent/BRPI0914238A2/pt

Links

229950010477 clopidogrel hydrogen sulphate Drugs 0.000 title 1
FDEODCTUSIWGLK-UHFFFAOYSA-N hydrogen sulfate;hydron;methyl 2-(2-chlorophenyl)-2-(6,7-dihydro-4h-thieno[3,2-c]pyridin-5-yl)acetate Chemical compound OS(O)(=O)=O.C1CC=2SC=CC=2CN1C(C(=O)OC)C1=CC=CC=C1Cl FDEODCTUSIWGLK-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

BRPI0914238-0A 2008-06-24 2009-06-11 Processo para a preparação da forma cristalina i de hidrogenossulfato de clopidogrel. BRPI0914238A2 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP08104529		2008-06-24
PCT/EP2009/057228 WO2009156279A2 (en)	2008-06-24	2009-06-11	Process for the preparation of clopidogrel hydrogen sulfate crystalline form i

Publications (1)

Publication Number	Publication Date
BRPI0914238A2 true BRPI0914238A2 (pt)	2015-08-04

Family

ID=41445014

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0914238-0A BRPI0914238A2 (pt)	2008-06-24	2009-06-11	Processo para a preparação da forma cristalina i de hidrogenossulfato de clopidogrel.

Country Status (8)

Country	Link
US (1)	US20110118467A1 (pt)
EP (1)	EP2300480A2 (pt)
CN (1)	CN102083837B (pt)
AU (1)	AU2009264395B2 (pt)
BR (1)	BRPI0914238A2 (pt)
CA (1)	CA2725997A1 (pt)
IL (1)	IL209589A0 (pt)
WO (1)	WO2009156279A2 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN102432625A (zh) *	2011-11-05	2012-05-02	江南大学	一种制备高纯度i型氯吡格雷硫酸氢盐的结晶方法
CN103360406A (zh) *	2012-03-26	2013-10-23	黑龙江福和华星制药集团股份有限公司	一种制备i型硫酸氢氯吡格雷的方法
KR101710922B1 (ko)	2015-06-03	2017-02-28	경동제약 주식회사	클로피도그렐 황산염 결정형 i형의 제조방법

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CZ297472B6 (cs) *	2002-08-27	2006-12-13	Zentiva, A.S.	Zpusob výroby clopidogrelu hydrogensulfátu krystalické formy I
WO2005012300A1 (en) *	2003-08-04	2005-02-10	Wockhardt Limited	A novel process for the manufacture of (+)-(s)-clopidogrel bisulfate form-i
DE10337773A1 (de) *	2003-08-13	2005-03-24	Krka Tovarna Zdravil, D.D.	Kristallisation von festen Formen von Clopidogrel-Additionssalzen
ATE455778T1 (de) *	2003-11-03	2010-02-15	Cadila Healthcare Ltd	Verfahren zur herstellung form i von (s)-(+)- clopidogrelbisulfat
US7629465B2 (en) *	2004-03-05	2009-12-08	Ipca Laboratories Ltd.	Industrial process for preparation of Clopidogrel hydrogen sulphate
WO2007017886A1 (en) *	2005-08-11	2007-02-15	Arch Pharmalabs Limited	Novel process for preparation of clopidogrel bisulphate polymorphic form i
CN100500670C (zh) *	2006-01-18	2009-06-17	上海应用技术学院	I型硫酸氯吡格雷的合成方法

2009
- 2009-06-11 WO PCT/EP2009/057228 patent/WO2009156279A2/en not_active Ceased
- 2009-06-11 AU AU2009264395A patent/AU2009264395B2/en not_active Ceased
- 2009-06-11 CN CN200980123605.7A patent/CN102083837B/zh not_active Expired - Fee Related
- 2009-06-11 CA CA2725997A patent/CA2725997A1/en not_active Abandoned
- 2009-06-11 EP EP09769128A patent/EP2300480A2/en not_active Withdrawn
- 2009-06-11 US US12/996,990 patent/US20110118467A1/en not_active Abandoned
- 2009-06-11 BR BRPI0914238-0A patent/BRPI0914238A2/pt not_active IP Right Cessation
2010
- 2010-11-25 IL IL209589A patent/IL209589A0/en unknown

Also Published As

Publication number	Publication date
US20110118467A1 (en)	2011-05-19
EP2300480A2 (en)	2011-03-30
AU2009264395B2 (en)	2013-12-05
CN102083837A (zh)	2011-06-01
WO2009156279A3 (en)	2011-01-13
CA2725997A1 (en)	2009-12-30
AU2009264395A1 (en)	2009-12-30
WO2009156279A2 (en)	2009-12-30
IL209589A0 (en)	2011-01-31
CN102083837B (zh)	2013-09-18

Similar Documents

Publication	Publication Date	Title
BRPI0910916A2 (pt)	2015-07-28	Processo para a produção de um dianidroaçúcar
BRPI0911254A2 (pt)	2015-10-06	processo para a preparação de um composto
BRPI0810238A2 (pt)	2014-10-29	Processo para produção de pcc
BR112012014490A2 (pt)	2015-09-15	processo para a preparação substituída de 1-o-acil-2-desóxi-2-fluoro-4-tio-beta-d-arabinofuranoses
BRPI0915572A2 (pt)	2017-06-27	processo para a fabricação de epicloroidrina
BRPI1013561A8 (pt)	2015-09-22	processo para a preparação de alogliptina
BRPI1014911A2 (pt)	2016-07-26	processo para fabricação de resinas carregadas
BRPI1014812A2 (pt)	2015-08-25	Processo para a produção de alacoóis
BRPI0914788A2 (pt)	2015-08-11	Processo para a produção de um produto intermediário de etexilato de dabigatran
BRPI0922490A2 (pt)	2015-08-04	Método para produção de beta-santaleno
BR112012005418A2 (pt)	2016-04-12	processo para a produção de grânulos
BRPI0909393A2 (pt)	2015-12-22	processo para a preparação de polibutadieno
BRPI0813960A2 (pt)	2015-01-06	Processo para produção de biarilas
BRPI1013830A2 (pt)	2010-10-28	Processo para a iodação de compostos aromáticos
BRPI1008987A2 (pt)	2016-03-22	processo para preparar 3,3,3-trifluoropropeno
BRPI0908900A2 (pt)	2019-09-24	processo para a produção de polióis
BRPI1013075A2 (pt)	2016-04-05	processo para produção de grânulos
BR112012001731A2 (pt)	2015-09-01	Processo para a preparação de 1-benzil-3-hidroximetil-1h-indazol
BRPI0914792A2 (pt)	2015-10-20	processo para a preparação de polióis
BRPI0913644A2 (pt)	2015-11-24	processo para a prepração de derivados de pirimidina substituída.
BRPI0920705A2 (pt)	2015-12-29	processo para a produção de compostos aquilaromáticos
BRPI1010571A2 (pt)	2019-09-24	processo para a preparação de um composto útil como um inibidor de tafla.
BRPI0821386A2 (pt)	2015-06-16	Processo para a preparação de r-lansoprazol amorfo estável
BRPI1008557A2 (pt)	2015-09-15	processo para a preparação de 5-/6-nitrofluoresceína
BRPI0912512A2 (pt)	2015-07-28	Processo para a preparação de compostos

Legal Events

Date	Code	Title	Description
2015-12-08	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]	Free format text: REFERENTE A 6A ANUIDADE.
2016-04-05	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2344 DE 08-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.