BRPI0917540A2 - composto, sal farmacologicamente aceitavél, composição farmacêutica, e, uso de um composto ou sal farmacologicamente aceitável - Google Patents

composto, sal farmacologicamente aceitavél, composição farmacêutica, e, uso de um composto ou sal farmacologicamente aceitável

Info

Publication number
BRPI0917540A2
BRPI0917540A2 BRPI0917540A BRPI0917540A BRPI0917540A2 BR PI0917540 A2 BRPI0917540 A2 BR PI0917540A2 BR PI0917540 A BRPI0917540 A BR PI0917540A BR PI0917540 A BRPI0917540 A BR PI0917540A BR PI0917540 A2 BRPI0917540 A2 BR PI0917540A2
Authority
BR
Brazil
Prior art keywords
compound
salt
pharmaceutical composition
pharmaceutically acceptable
pharmacologically acceptable
Prior art date
Application number
BRPI0917540A
Other languages
English (en)
Inventor
Hironao Saito
Hironori Matsunaga
Masami Ohtsuka
Masanori Ichikawa
Noriyasu Haginoya
Tomoyuki Tsunemi
Yoshihiro Shibata
Original Assignee
Daiichi Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Sankyo Co Ltd filed Critical Daiichi Sankyo Co Ltd
Publication of BRPI0917540A2 publication Critical patent/BRPI0917540A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
BRPI0917540A 2008-08-05 2009-08-04 composto, sal farmacologicamente aceitavél, composição farmacêutica, e, uso de um composto ou sal farmacologicamente aceitável BRPI0917540A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2008201670 2008-08-05
JP2009078540 2009-03-27
PCT/JP2009/063807 WO2010016490A1 (ja) 2008-08-05 2009-08-04 イミダゾピリジン-2-オン誘導体

Publications (1)

Publication Number Publication Date
BRPI0917540A2 true BRPI0917540A2 (pt) 2015-11-17

Family

ID=41663708

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0917540A BRPI0917540A2 (pt) 2008-08-05 2009-08-04 composto, sal farmacologicamente aceitavél, composição farmacêutica, e, uso de um composto ou sal farmacologicamente aceitável

Country Status (21)

Country Link
US (2) US8436012B2 (pt)
EP (1) EP2308877B1 (pt)
JP (1) JP5630867B2 (pt)
KR (1) KR20110039307A (pt)
CN (1) CN102171210B (pt)
AU (1) AU2009278442B2 (pt)
BR (1) BRPI0917540A2 (pt)
CA (1) CA2732950C (pt)
CO (1) CO6300866A2 (pt)
DK (1) DK2308877T3 (pt)
ES (1) ES2459047T3 (pt)
IL (1) IL211042A (pt)
MX (1) MX2011001019A (pt)
MY (1) MY153606A (pt)
NZ (1) NZ590688A (pt)
PL (1) PL2308877T3 (pt)
PT (1) PT2308877E (pt)
RU (1) RU2478636C2 (pt)
TW (1) TWI436998B (pt)
WO (1) WO2010016490A1 (pt)
ZA (1) ZA201100799B (pt)

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Also Published As

Publication number Publication date
MY153606A (en) 2015-02-27
US8785438B2 (en) 2014-07-22
CN102171210A (zh) 2011-08-31
IL211042A (en) 2014-12-31
US20110082138A1 (en) 2011-04-07
MX2011001019A (es) 2011-03-25
IL211042A0 (en) 2011-04-28
TW201011021A (en) 2010-03-16
US8436012B2 (en) 2013-05-07
CA2732950A1 (en) 2010-02-11
US20130338156A1 (en) 2013-12-19
JP5630867B2 (ja) 2014-11-26
AU2009278442A1 (en) 2010-02-11
CN102171210B (zh) 2014-04-23
RU2478636C2 (ru) 2013-04-10
AU2009278442B2 (en) 2013-09-26
CA2732950C (en) 2013-10-01
EP2308877B1 (en) 2014-01-22
CO6300866A2 (es) 2011-07-21
NZ590688A (en) 2012-09-28
TWI436998B (zh) 2014-05-11
DK2308877T3 (da) 2014-04-22
PL2308877T3 (pl) 2014-07-31
ZA201100799B (en) 2011-10-26
KR20110039307A (ko) 2011-04-15
RU2011108453A (ru) 2012-09-10
EP2308877A4 (en) 2012-03-14
PT2308877E (pt) 2014-05-02
JPWO2010016490A1 (ja) 2012-01-26
ES2459047T3 (es) 2014-05-07
WO2010016490A1 (ja) 2010-02-11
EP2308877A1 (en) 2011-04-13
HK1155444A1 (en) 2012-05-18

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