CH437327A - Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydropyrido (4,3-d) pyrimidinen - Google Patents

Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydropyrido (4,3-d) pyrimidinen

Info

Publication number
CH437327A
CH437327A CH302963A CH302963A CH437327A CH 437327 A CH437327 A CH 437327A CH 302963 A CH302963 A CH 302963A CH 302963 A CH302963 A CH 302963A CH 437327 A CH437327 A CH 437327A
Authority
CH
Switzerland
Prior art keywords
tetrahydropyrido
pyrimidines
preparation
new
Prior art date
Application number
CH302963A
Other languages
English (en)
Inventor
Ohnacker Gerhard Dr Dipl-Chem
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of CH437327A publication Critical patent/CH437327A/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CH302963A 1962-03-22 1963-03-11 Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydropyrido (4,3-d) pyrimidinen CH437327A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DET21813A DE1197466B (de) 1962-03-22 1962-03-22 Verfahren zur Herstellung von neuen 5, 6, 7, 8-Tetrahydropyrido-[4, 3-d]pyrimidinen

Publications (1)

Publication Number Publication Date
CH437327A true CH437327A (de) 1967-06-15

Family

ID=7550280

Family Applications (2)

Application Number Title Priority Date Filing Date
CH302963A CH437327A (de) 1962-03-22 1963-03-11 Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydropyrido (4,3-d) pyrimidinen
CH1780166A CH462186A (de) 1962-03-22 1963-03-11 Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydro-pyrido(4,3-d)pyrimidinen

Family Applications After (1)

Application Number Title Priority Date Filing Date
CH1780166A CH462186A (de) 1962-03-22 1963-03-11 Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydro-pyrido(4,3-d)pyrimidinen

Country Status (5)

Country Link
US (1) US3248395A (de)
CH (2) CH437327A (de)
DE (1) DE1197466B (de)
FR (1) FR2450M (de)
GB (1) GB1033384A (de)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3725405A (en) * 1970-06-18 1973-04-03 American Home Prod 2,4,7-TRISUBSTITUTED-{8 PYRIDO 2,3-d{9 PYRIMIDINE-6-CARBOXAMIDES
US3939268A (en) * 1971-04-10 1976-02-17 Boehringer Ingelheim Gmbh 2,4-Diamino substituted pyridol(3,2-d)pyrimidine as antithrombotic agents
JPS5130077B2 (de) * 1971-12-28 1976-08-30
US4085102A (en) * 1974-11-25 1978-04-18 E. R. Squibb & Sons, Inc. 2-Amino-8-arylideno-3,4,5,6,7,8-hexahydro-4-arlypyrido[4,3-d]pyrimidines
US5137890A (en) * 1990-02-14 1992-08-11 Ortho Pharmaceutical Corporation 4-phenyl tetrahydropyrido(4,3-d)pyrimidines
US5059602A (en) * 1990-08-27 1991-10-22 Hoechst-Roussel Pharmaceuticals Inc. 4-substituted dihydropyrido(4,3-d)pyrimidines as analgesics and topical antiinflammatory agents for the treatment of skin disorders
US5212310A (en) * 1991-12-19 1993-05-18 Neurogen Corporation Certain aryl fused imidazopyrimidines; a new class of GABA brain receptor ligands
ATE456836T1 (de) * 1996-09-04 2010-02-15 Intertrust Tech Corp Zuverlässige infrastrukturhilfssysteme, verfahren und techniken für sicheren elektronischen handel, elektronische transaktionen, handelsablaufsteuerung und automatisierung, verteilte verarbeitung und rechteverwaltung
US7105667B2 (en) * 2001-05-01 2006-09-12 Bristol-Myers Squibb Co. Fused heterocyclic compounds and use thereof
WO2002088079A2 (en) * 2001-05-01 2002-11-07 Bristol-Myers Squibb Company Dual inhibitors of pde 7 and pde 4
AU2003242252A1 (en) * 2002-06-07 2003-12-22 Kyowa Hakko Kogyo Co., Ltd. Bicyclic pyrimidine derivatives
EP1663994B1 (de) 2003-08-05 2012-03-07 Vertex Pharmaceuticals Incorporated Tetrahydrochinazolin-verbindungen als inhibitoren von spannungsabhängigen ionenkanälen
SG146683A1 (en) * 2003-09-17 2008-10-30 Janssen Pharmaceutica Nv Fused heterocyclic compounds as serotonin receptor modulators
JP5198256B2 (ja) * 2005-05-04 2013-05-15 エボテク エージー 縮合複素環式化合物、並びにそれらの組成物及び使用
US7598255B2 (en) * 2005-08-04 2009-10-06 Janssen Pharmaceutica Nv Pyrimidine compounds as serotonin receptor modulators
WO2009097578A1 (en) 2008-02-01 2009-08-06 Takeda Pharmaceutical Company Limited Oxim derivatives as hsp90 inhibitors
US8163763B2 (en) * 2008-07-31 2012-04-24 Genentech, Inc. Pyrimidine compounds, compositions and methods of use
WO2010120991A1 (en) * 2009-04-17 2010-10-21 Wyeth Llc 5, 6, 7, 8-tetrahydropyrido[4,3-d]pyrimidine compounds, their use as mtor, pi3, and hsmg-1 kinase inhibitors, and their syntheses
EP2445346A4 (de) * 2009-06-24 2012-12-05 Genentech Inc Oxoheterozyklische fusionierte pyrimidinverbindungen und -zusammensetzungen sowie verfahren zu ihrer verwendung
US8691827B2 (en) 2009-08-17 2014-04-08 Merck Sharp & Dohme Corp. Amino tetrahydro-pyridopyrimidine PDE10 inhibitors
ES2567168T3 (es) * 2009-11-12 2016-04-20 F. Hoffmann-La Roche Ag Compuestos purina y pirazolopirimidina N7-sustituidos, composiciones y métodos de utilización
WO2011058027A2 (en) * 2009-11-12 2011-05-19 F. Hoffmann-La Roche Ag N-9-substituted purine compounds, compositions and methods of use
UA112517C2 (uk) 2010-07-06 2016-09-26 Новартіс Аг Тетрагідропіридопіримідинові похідні

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2697710A (en) * 1953-01-02 1954-12-21 Burroughs Wellcome Co Pyrido (2,3-d) pyrimidines and method of preparing same
US2926166A (en) * 1954-01-04 1960-02-23 Burroughs Wellcome Co Pyrido (2, 3-d) pyrimidine compounds and method of making
US2802826A (en) * 1955-07-13 1957-08-13 Hoffmann La Roche Octahydro-pyrido [4, 3-d] pyrimidine compounds
US2890152A (en) * 1956-11-29 1959-06-09 Schering Corp Topical anti-inflammatory compositions
US2994640A (en) * 1957-02-22 1961-08-01 Byk Gulden Lomberg Chem Fab Anti-inflammatory therapy with purine molecular compounds
DE1110649B (de) * 1957-11-22 1961-07-13 Ciba Geigy Verfahren zur Herstellung von 1-Isopropyl-pyrazolo[3, 4-d]pyrimidinen

Also Published As

Publication number Publication date
DE1197466B (de) 1965-07-29
US3248395A (en) 1966-04-26
CH462186A (de) 1968-09-15
GB1033384A (en) 1966-06-22
FR2450M (fr) 1964-04-06

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