CH462186A - Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydro-pyrido(4,3-d)pyrimidinen - Google Patents

Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydro-pyrido(4,3-d)pyrimidinen

Info

Publication number
CH462186A
CH462186A CH1780166A CH1780166A CH462186A CH 462186 A CH462186 A CH 462186A CH 1780166 A CH1780166 A CH 1780166A CH 1780166 A CH1780166 A CH 1780166A CH 462186 A CH462186 A CH 462186A
Authority
CH
Switzerland
Prior art keywords
tetrahydropyrido
pyrimidines
preparation
new
Prior art date
Application number
CH1780166A
Other languages
English (en)
Inventor
Gerhard Dr Ohnacker
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of CH462186A publication Critical patent/CH462186A/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CH1780166A 1962-03-22 1963-03-11 Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydro-pyrido(4,3-d)pyrimidinen CH462186A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DET21813A DE1197466B (de) 1962-03-22 1962-03-22 Verfahren zur Herstellung von neuen 5, 6, 7, 8-Tetrahydropyrido-[4, 3-d]pyrimidinen

Publications (1)

Publication Number Publication Date
CH462186A true CH462186A (de) 1968-09-15

Family

ID=7550280

Family Applications (2)

Application Number Title Priority Date Filing Date
CH302963A CH437327A (de) 1962-03-22 1963-03-11 Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydropyrido (4,3-d) pyrimidinen
CH1780166A CH462186A (de) 1962-03-22 1963-03-11 Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydro-pyrido(4,3-d)pyrimidinen

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CH302963A CH437327A (de) 1962-03-22 1963-03-11 Verfahren zur Herstellung von neuen 5,6,7,8-Tetrahydropyrido (4,3-d) pyrimidinen

Country Status (5)

Country Link
US (1) US3248395A (de)
CH (2) CH437327A (de)
DE (1) DE1197466B (de)
FR (1) FR2450M (de)
GB (1) GB1033384A (de)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3725405A (en) * 1970-06-18 1973-04-03 American Home Prod 2,4,7-TRISUBSTITUTED-{8 PYRIDO 2,3-d{9 PYRIMIDINE-6-CARBOXAMIDES
US3939268A (en) * 1971-04-10 1976-02-17 Boehringer Ingelheim Gmbh 2,4-Diamino substituted pyridol(3,2-d)pyrimidine as antithrombotic agents
JPS5130077B2 (de) * 1971-12-28 1976-08-30
US4085102A (en) * 1974-11-25 1978-04-18 E. R. Squibb & Sons, Inc. 2-Amino-8-arylideno-3,4,5,6,7,8-hexahydro-4-arlypyrido[4,3-d]pyrimidines
US5137890A (en) * 1990-02-14 1992-08-11 Ortho Pharmaceutical Corporation 4-phenyl tetrahydropyrido(4,3-d)pyrimidines
US5059602A (en) * 1990-08-27 1991-10-22 Hoechst-Roussel Pharmaceuticals Inc. 4-substituted dihydropyrido(4,3-d)pyrimidines as analgesics and topical antiinflammatory agents for the treatment of skin disorders
US5212310A (en) * 1991-12-19 1993-05-18 Neurogen Corporation Certain aryl fused imidazopyrimidines; a new class of GABA brain receptor ligands
DE69636466T2 (de) * 1996-09-04 2007-08-09 Intertrust Technologies Corp., Sunnyvale Treuhand infrastruktur unterstützungssysteme, verfahren und techniken zum sicheren elektronischen handel, elektronische transaktionen, steuerung und automatisierung von handelsverfahren, verteilte datenverarbeitung und verwalten von rechten
US7105667B2 (en) * 2001-05-01 2006-09-12 Bristol-Myers Squibb Co. Fused heterocyclic compounds and use thereof
WO2002088079A2 (en) * 2001-05-01 2002-11-07 Bristol-Myers Squibb Company Dual inhibitors of pde 7 and pde 4
AU2003242252A1 (en) * 2002-06-07 2003-12-22 Kyowa Hakko Kogyo Co., Ltd. Bicyclic pyrimidine derivatives
NZ545717A (en) 2003-08-05 2009-12-24 Vertex Pharma Hydrogenated quinazoline derivatives as inhibitors of voltage-gated ion channels
DE602004019118D1 (de) * 2003-09-17 2009-03-05 Janssen Pharmaceutica Nv Kondensierte heterocyclische verbindungen als modulatoren des serotoninrezeptors
WO2006119504A2 (en) * 2005-05-04 2006-11-09 Renovis, Inc. Fused heterocyclic compounds, and compositions and uses thereof
US7598255B2 (en) * 2005-08-04 2009-10-06 Janssen Pharmaceutica Nv Pyrimidine compounds as serotonin receptor modulators
US8071766B2 (en) 2008-02-01 2011-12-06 Takeda Pharmaceutical Company Limited HSP90 inhibitors
EP2318377B1 (de) * 2008-07-31 2013-08-21 Genentech, Inc. Pyrimidinverbindungen und -zusammensetzungen sowie verfahren zu ihrer verwendung
WO2010120991A1 (en) * 2009-04-17 2010-10-21 Wyeth Llc 5, 6, 7, 8-tetrahydropyrido[4,3-d]pyrimidine compounds, their use as mtor, pi3, and hsmg-1 kinase inhibitors, and their syntheses
US20100331305A1 (en) * 2009-06-24 2010-12-30 Genentech, Inc. Oxo-heterocycle fused pyrimidine compounds, compositions and methods of use
WO2011022213A1 (en) * 2009-08-17 2011-02-24 Merck Sharp & Dohme Corp. Amino tetrahydro-pyridopyrimidine pde10 inhibitors
CN102711766B (zh) * 2009-11-12 2014-06-04 霍夫曼-拉罗奇有限公司 N-9-取代的嘌呤化合物、组合物和使用方法
CN102712642B (zh) * 2009-11-12 2015-08-12 霍夫曼-拉罗奇有限公司 N-7取代的嘌呤和吡唑并嘧啶化合物、组合物和使用方法
UA112517C2 (uk) 2010-07-06 2016-09-26 Новартіс Аг Тетрагідропіридопіримідинові похідні

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2697710A (en) * 1953-01-02 1954-12-21 Burroughs Wellcome Co Pyrido (2,3-d) pyrimidines and method of preparing same
US2926166A (en) * 1954-01-04 1960-02-23 Burroughs Wellcome Co Pyrido (2, 3-d) pyrimidine compounds and method of making
US2802826A (en) * 1955-07-13 1957-08-13 Hoffmann La Roche Octahydro-pyrido [4, 3-d] pyrimidine compounds
US2890152A (en) * 1956-11-29 1959-06-09 Schering Corp Topical anti-inflammatory compositions
US2994640A (en) * 1957-02-22 1961-08-01 Byk Gulden Lomberg Chem Fab Anti-inflammatory therapy with purine molecular compounds
DE1110649B (de) * 1957-11-22 1961-07-13 Ciba Geigy Verfahren zur Herstellung von 1-Isopropyl-pyrazolo[3, 4-d]pyrimidinen

Also Published As

Publication number Publication date
DE1197466B (de) 1965-07-29
US3248395A (en) 1966-04-26
FR2450M (fr) 1964-04-06
GB1033384A (en) 1966-06-22
CH437327A (de) 1967-06-15

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