CL2007002643A1 - Compuestos derivados de 5-fenil-nicotinamida, moduladores del receptor de cb1; procedimiento de preparacion; composiciones farmaceuticas; y uso para el tratamiento y/o profilaxis de trastornos de la nutricion, diabetes tipo ii y dependencia de sustan - Google Patents

Compuestos derivados de 5-fenil-nicotinamida, moduladores del receptor de cb1; procedimiento de preparacion; composiciones farmaceuticas; y uso para el tratamiento y/o profilaxis de trastornos de la nutricion, diabetes tipo ii y dependencia de sustan

Info

Publication number: CL2007002643A1
Authority: CL; Chile
Prior art keywords: sustan; profilaxis; nicotinamide; diabetes; dependence
Prior art date: 2006-09-14

Application number

CL200702643A

Other languages

English (en)

Inventor

Hebeisen Stephan Roever Paul

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-09-14

Filing date

2007-09-12

Publication date

2008-04-18

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38924794&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2007002643(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2007-09-12 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2008-04-18 Publication of CL2007002643A1 publication Critical patent/CL2007002643A1/es

Links

NKMMJBMWTNPJCV-UHFFFAOYSA-N 5-phenylpyridine-3-carboxamide Chemical compound NC(=O)C1=CN=CC(C=2C=CC=CC=2)=C1 NKMMJBMWTNPJCV-UHFFFAOYSA-N 0.000 title 1
150000001875 compounds Chemical class 0.000 title 1
238000000034 method Methods 0.000 title 1
208000030212 nutrition disease Diseases 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1
208000001072 type 2 diabetes mellitus Diseases 0.000 title 1

Classifications

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- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/56—Amides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
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- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Diabetes (AREA)
Psychiatry (AREA)
Addiction (AREA)
Hematology (AREA)
Pain & Pain Management (AREA)
Obesity (AREA)
Endocrinology (AREA)
Urology & Nephrology (AREA)
Oncology (AREA)
Epidemiology (AREA)
Hospice & Palliative Care (AREA)
Cardiology (AREA)
Communicable Diseases (AREA)
Heart & Thoracic Surgery (AREA)
Reproductive Health (AREA)
Emergency Medicine (AREA)
Otolaryngology (AREA)
Rheumatology (AREA)
Child & Adolescent Psychology (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Vascular Medicine (AREA)

CL200702643A 2006-09-14 2007-09-12 Compuestos derivados de 5-fenil-nicotinamida, moduladores del receptor de cb1; procedimiento de preparacion; composiciones farmaceuticas; y uso para el tratamiento y/o profilaxis de trastornos de la nutricion, diabetes tipo ii y dependencia de sustan CL2007002643A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP06120672		2006-09-14

Publications (1)

Publication Number	Publication Date
CL2007002643A1 true CL2007002643A1 (es)	2008-04-18

Family

ID=38924794

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CL200702643A CL2007002643A1 (es)	2006-09-14	2007-09-12	Compuestos derivados de 5-fenil-nicotinamida, moduladores del receptor de cb1; procedimiento de preparacion; composiciones farmaceuticas; y uso para el tratamiento y/o profilaxis de trastornos de la nutricion, diabetes tipo ii y dependencia de sustan

Country Status (17)

Country	Link
US (1)	US7781593B2 (es)
EP (1)	EP2066636B1 (es)
JP (1)	JP5133344B2 (es)
KR (1)	KR101116024B1 (es)
CN (1)	CN101516849A (es)
AR (1)	AR062769A1 (es)
AT (1)	ATE530529T1 (es)
AU (1)	AU2007296691B2 (es)
BR (1)	BRPI0716535A2 (es)
CA (1)	CA2662409A1 (es)
CL (1)	CL2007002643A1 (es)
ES (1)	ES2372546T3 (es)
IL (1)	IL197152A0 (es)
MX (1)	MX2009002632A (es)
PE (1)	PE20081373A1 (es)
TW (1)	TW200820971A (es)
WO (1)	WO2008031734A1 (es)

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EP2074096B1 (en) *	2006-10-04	2012-06-27	F. Hoffmann-La Roche AG	3-pyridinecarboxamide and 2-pyrazinecarboxamide derivatives as hdl-cholesterol raising agents
WO2008040649A2 (en) *	2006-10-04	2008-04-10	F. Hoffmann-La Roche Ag	Pyrazine-2-carboxamide derivatives as cb2 receptor modulators
EP2025674A1 (de)	2007-08-15	2009-02-18	sanofi-aventis	Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
US8088920B2 (en) *	2008-03-31	2012-01-03	Hoffmann-La Roche Inc.	3-trifluoromethyl-pyrazine-2-carboxylic acid amide derivatives as HDL-cholesterol raising agents
US7897621B2 (en) *	2008-03-31	2011-03-01	Hoffmann-La Roche Inc.	2-trifluoromethylnicotinamide derivatives as HDL-cholesterol raising agents
US8410107B2 (en)	2010-10-15	2013-04-02	Hoffmann-La Roche Inc.	N-pyridin-3-yl or N-pyrazin-2-yl carboxamides
US8669254B2 (en)	2010-12-15	2014-03-11	Hoffman-La Roche Inc.	Pyridine, pyridazine, pyrimidine or pyrazine carboxamides as HDL-cholesterol raising agents

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2007
- 2007-08-29 US US11/846,667 patent/US7781593B2/en not_active Expired - Fee Related
- 2007-09-03 AT AT07803154T patent/ATE530529T1/de active
- 2007-09-03 CA CA002662409A patent/CA2662409A1/en not_active Abandoned
- 2007-09-03 ES ES07803154T patent/ES2372546T3/es active Active
- 2007-09-03 CN CNA2007800338694A patent/CN101516849A/zh active Pending
- 2007-09-03 BR BRPI0716535-8A2A patent/BRPI0716535A2/pt not_active IP Right Cessation
- 2007-09-03 JP JP2009527775A patent/JP5133344B2/ja not_active Expired - Fee Related
- 2007-09-03 EP EP07803154A patent/EP2066636B1/en not_active Not-in-force
- 2007-09-03 AU AU2007296691A patent/AU2007296691B2/en not_active Expired - Fee Related
- 2007-09-03 WO PCT/EP2007/059167 patent/WO2008031734A1/en not_active Ceased
- 2007-09-03 KR KR1020097005139A patent/KR101116024B1/ko not_active Expired - Fee Related
- 2007-09-03 MX MX2009002632A patent/MX2009002632A/es active IP Right Grant
- 2007-09-11 TW TW096133922A patent/TW200820971A/zh unknown
- 2007-09-12 CL CL200702643A patent/CL2007002643A1/es unknown
- 2007-09-12 AR ARP070104041A patent/AR062769A1/es unknown
- 2007-09-13 PE PE2007001236A patent/PE20081373A1/es not_active Application Discontinuation
2009
- 2009-02-19 IL IL197152A patent/IL197152A0/en unknown

Also Published As

Publication number	Publication date
AR062769A1 (es)	2008-12-03
TW200820971A (en)	2008-05-16
US20080070931A1 (en)	2008-03-20
ATE530529T1 (de)	2011-11-15
ES2372546T3 (es)	2012-01-23
JP2010503633A (ja)	2010-02-04
EP2066636A1 (en)	2009-06-10
BRPI0716535A2 (pt)	2013-09-24
KR20090040381A (ko)	2009-04-23
AU2007296691A1 (en)	2008-03-20
WO2008031734A1 (en)	2008-03-20
CA2662409A1 (en)	2008-03-20
AU2007296691B2 (en)	2012-12-20
KR101116024B1 (ko)	2012-02-13
MX2009002632A (es)	2009-03-24
CN101516849A (zh)	2009-08-26
IL197152A0 (en)	2009-11-18
JP5133344B2 (ja)	2013-01-30
PE20081373A1 (es)	2008-09-18
US7781593B2 (en)	2010-08-24
EP2066636B1 (en)	2011-10-26

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