CL2007002836A1 - Compuestos derivados de 1,3,5-triazina o pirimidina, inhibidores de quinasa; composicion farmaceutica; y uso para tratar una enfermedad mediada por quinasa, tal como cancer. - Google Patents

Compuestos derivados de 1,3,5-triazina o pirimidina, inhibidores de quinasa; composicion farmaceutica; y uso para tratar una enfermedad mediada por quinasa, tal como cancer.

Info

Publication number: CL2007002836A1
Authority: CL; Chile
Prior art keywords: triazine; pyrimidine; kinase; cancer; treat
Prior art date: 2006-10-02

Application number

CL200702836A

Other languages

English (en)

Inventor

Pamela A Xie Yongping Albaugh

Original Assignee

Irm Llc Y Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-10-02

Filing date

2007-10-02

Publication date

2008-05-23

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38955203&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2007002836(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2007-10-02 Application filed by Irm Llc Y Novartis Ag filed Critical Irm Llc Y Novartis Ag

2008-05-23 Publication of CL2007002836A1 publication Critical patent/CL2007002836A1/es

Links

JIHQDMXYYFUGFV-UHFFFAOYSA-N 1,3,5-triazine Chemical compound C1=NC=NC=N1 JIHQDMXYYFUGFV-UHFFFAOYSA-N 0.000 title 1
206010028980 Neoplasm Diseases 0.000 title 1
108091000080 Phosphotransferase Proteins 0.000 title 1
CZPWVGJYEJSRLH-UHFFFAOYSA-N Pyrimidine Chemical compound C1=CN=CN=C1 CZPWVGJYEJSRLH-UHFFFAOYSA-N 0.000 title 1
201000011510 cancer Diseases 0.000 title 1
150000001875 compounds Chemical class 0.000 title 1
201000010099 disease Diseases 0.000 title 1
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 1
239000003112 inhibitor Substances 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1
102000020233 phosphotransferase Human genes 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Physical Education & Sports Medicine (AREA)
Immunology (AREA)
Biomedical Technology (AREA)
Orthopedic Medicine & Surgery (AREA)
Diabetes (AREA)
Neurosurgery (AREA)
Rheumatology (AREA)
Hematology (AREA)
Pulmonology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Oncology (AREA)
Pain & Pain Management (AREA)
Dermatology (AREA)
Endocrinology (AREA)
Vascular Medicine (AREA)
Tropical Medicine & Parasitology (AREA)
Psychiatry (AREA)
Transplantation (AREA)
Hospice & Palliative Care (AREA)
Urology & Nephrology (AREA)
Psychology (AREA)
Toxicology (AREA)
Obesity (AREA)

CL200702836A 2006-10-02 2007-10-02 Compuestos derivados de 1,3,5-triazina o pirimidina, inhibidores de quinasa; composicion farmaceutica; y uso para tratar una enfermedad mediada por quinasa, tal como cancer. CL2007002836A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US82787306P	2006-10-02	2006-10-02

Publications (1)

Publication Number	Publication Date
CL2007002836A1 true CL2007002836A1 (es)	2008-05-23

Family

ID=38955203

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CL200702836A CL2007002836A1 (es)	2006-10-02	2007-10-02	Compuestos derivados de 1,3,5-triazina o pirimidina, inhibidores de quinasa; composicion farmaceutica; y uso para tratar una enfermedad mediada por quinasa, tal como cancer.

Country Status (22)

Country	Link
US (1)	US8202876B2 (es)
EP (1)	EP2057146A1 (es)
JP (1)	JP5153777B2 (es)
KR (1)	KR101101675B1 (es)
CN (2)	CN103739595A (es)
AR (1)	AR063099A1 (es)
AU (1)	AU2007305016B2 (es)
BR (1)	BRPI0719797A8 (es)
CA (1)	CA2663366C (es)
CL (1)	CL2007002836A1 (es)
CO (1)	CO6180440A2 (es)
CR (1)	CR10670A (es)
EA (1)	EA015751B1 (es)
IL (1)	IL197724A0 (es)
MA (1)	MA30772B1 (es)
MX (1)	MX2009003456A (es)
NO (1)	NO20091759L (es)
PE (1)	PE20080828A1 (es)
SM (1)	SMAP200900020A (es)
TN (1)	TN2009000105A1 (es)
TW (1)	TW200823200A (es)
WO (1)	WO2008042639A1 (es)

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2007
- 2007-09-24 MX MX2009003456A patent/MX2009003456A/es active IP Right Grant
- 2007-09-24 KR KR1020097006724A patent/KR101101675B1/ko not_active Expired - Fee Related
- 2007-09-24 CN CN201310581142.7A patent/CN103739595A/zh active Pending
- 2007-09-24 AU AU2007305016A patent/AU2007305016B2/en not_active Ceased
- 2007-09-24 CA CA2663366A patent/CA2663366C/en not_active Expired - Fee Related
- 2007-09-24 WO PCT/US2007/079340 patent/WO2008042639A1/en not_active Ceased
- 2007-09-24 EP EP07814982A patent/EP2057146A1/en not_active Withdrawn
- 2007-09-24 EA EA200970347A patent/EA015751B1/ru not_active IP Right Cessation
- 2007-09-24 BR BRPI0719797A patent/BRPI0719797A8/pt not_active Application Discontinuation
- 2007-09-24 JP JP2009531524A patent/JP5153777B2/ja not_active Expired - Fee Related
- 2007-09-24 CN CNA2007800368577A patent/CN101522661A/zh active Pending
- 2007-09-24 US US12/444,129 patent/US8202876B2/en not_active Expired - Fee Related
- 2007-10-02 AR ARP070104361A patent/AR063099A1/es unknown
- 2007-10-02 CL CL200702836A patent/CL2007002836A1/es unknown
- 2007-10-02 TW TW096136908A patent/TW200823200A/zh unknown
- 2007-10-02 PE PE2007001326A patent/PE20080828A1/es not_active Application Discontinuation
2009
- 2009-03-19 CR CR10670A patent/CR10670A/es not_active Application Discontinuation
- 2009-03-19 IL IL197724A patent/IL197724A0/en unknown
- 2009-03-27 SM SM200900020T patent/SMAP200900020A/it unknown
- 2009-03-27 TN TN2009000105A patent/TN2009000105A1/fr unknown
- 2009-04-02 CO CO09034040A patent/CO6180440A2/es not_active Application Discontinuation
- 2009-04-02 MA MA31753A patent/MA30772B1/fr unknown
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Also Published As

Publication number	Publication date
SMAP200900020A (it)	2009-05-11
MA30772B1 (fr)	2009-10-01
TW200823200A (en)	2008-06-01
CR10670A (es)	2009-05-13
US20100029605A1 (en)	2010-02-04
BRPI0719797A8 (pt)	2017-12-26
NO20091759L (no)	2009-07-01
BRPI0719797A2 (pt)	2017-10-24
CA2663366A1 (en)	2008-04-10
CN103739595A (zh)	2014-04-23
CA2663366C (en)	2012-02-07
AU2007305016B2 (en)	2011-11-03
TN2009000105A1 (en)	2010-08-19
EA015751B1 (ru)	2011-12-30
WO2008042639A1 (en)	2008-04-10
EP2057146A1 (en)	2009-05-13
JP2010505862A (ja)	2010-02-25
PE20080828A1 (es)	2008-08-12
CN101522661A (zh)	2009-09-02
IL197724A0 (en)	2009-12-24
JP5153777B2 (ja)	2013-02-27
EA200970347A1 (ru)	2009-10-30
MX2009003456A (es)	2009-04-14
CO6180440A2 (es)	2010-07-19
AU2007305016A1 (en)	2008-04-10
KR20090060322A (ko)	2009-06-11
AR063099A1 (es)	2008-12-30
US8202876B2 (en)	2012-06-19
KR101101675B1 (ko)	2011-12-30

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