CL2011000571A1 - Uso de una combinacion de: a) un compuesto de formula (1) o una sal farmaceuticamente aceptable del mismo, b) interferon alfa y c) ribavirina para preparar un medicamento util para el tratamiento de una infeccion viral de la hepatitis c (hcv) o para aliviar uno o mas sintomas de la misma. - Google Patents
Uso de una combinacion de: a) un compuesto de formula (1) o una sal farmaceuticamente aceptable del mismo, b) interferon alfa y c) ribavirina para preparar un medicamento util para el tratamiento de una infeccion viral de la hepatitis c (hcv) o para aliviar uno o mas sintomas de la misma.Info
- Publication number
- CL2011000571A1 CL2011000571A1 CL2011000571A CL2011000571A CL2011000571A1 CL 2011000571 A1 CL2011000571 A1 CL 2011000571A1 CL 2011000571 A CL2011000571 A CL 2011000571A CL 2011000571 A CL2011000571 A CL 2011000571A CL 2011000571 A1 CL2011000571 A1 CL 2011000571A1
- Authority
- CL
- Chile
- Prior art keywords
- ribavirin
- hepatitis
- compound
- formula
- hcv
- Prior art date
Links
- 102000006992 Interferon-alpha Human genes 0.000 title abstract 2
- 108010047761 Interferon-alpha Proteins 0.000 title abstract 2
- IWUCXVSUMQZMFG-AFCXAGJDSA-N Ribavirin Chemical compound N1=C(C(=O)N)N=CN1[C@H]1[C@H](O)[C@H](O)[C@@H](CO)O1 IWUCXVSUMQZMFG-AFCXAGJDSA-N 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 229950000038 interferon alfa Drugs 0.000 title abstract 2
- 229960000329 ribavirin Drugs 0.000 title abstract 2
- HZCAHMRRMINHDJ-DBRKOABJSA-N ribavirin Natural products O[C@@H]1[C@H](O)[C@@H](CO)O[C@H]1N1N=CN=C1 HZCAHMRRMINHDJ-DBRKOABJSA-N 0.000 title abstract 2
- 208000036142 Viral infection Diseases 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 208000006454 hepatitis Diseases 0.000 title 1
- 231100000283 hepatitis Toxicity 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
- 208000024891 symptom Diseases 0.000 title 1
- 230000009385 viral infection Effects 0.000 title 1
- 208000005176 Hepatitis C Diseases 0.000 abstract 1
- 208000010710 hepatitis C virus infection Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/7056—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing five-membered rings with nitrogen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/06—Tripeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/19—Cytokines; Lymphokines; Interferons
- A61K38/21—Interferons [IFN]
- A61K38/212—IFN-alpha
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Molecular Biology (AREA)
- Virology (AREA)
- Oncology (AREA)
- Zoology (AREA)
- Communicable Diseases (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Uso de una combinación farmacéutica de un compuesto de fórmula (1), interferón alfa y ribavirina, para tratar una infección por hepatitis C del genotipo 1; kit farmacéutico.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9775308P | 2008-09-17 | 2008-09-17 | |
| US10903308P | 2008-10-28 | 2008-10-28 | |
| US17193509P | 2009-04-23 | 2009-04-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2011000571A1 true CL2011000571A1 (es) | 2011-07-29 |
Family
ID=41571875
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2011000571A CL2011000571A1 (es) | 2008-09-17 | 2011-03-17 | Uso de una combinacion de: a) un compuesto de formula (1) o una sal farmaceuticamente aceptable del mismo, b) interferon alfa y c) ribavirina para preparar un medicamento util para el tratamiento de una infeccion viral de la hepatitis c (hcv) o para aliviar uno o mas sintomas de la misma. |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US8399484B2 (es) |
| EP (1) | EP2337583A1 (es) |
| JP (1) | JP5539363B2 (es) |
| KR (1) | KR20110054003A (es) |
| CN (1) | CN102159245B (es) |
| AR (1) | AR073516A1 (es) |
| AU (1) | AU2009293493B2 (es) |
| BR (1) | BRPI0918653A2 (es) |
| CA (1) | CA2737376A1 (es) |
| CL (1) | CL2011000571A1 (es) |
| CO (1) | CO6351753A2 (es) |
| EA (1) | EA019965B1 (es) |
| EC (1) | ECSP11010877A (es) |
| IL (1) | IL210152A0 (es) |
| MA (1) | MA32634B1 (es) |
| MX (1) | MX2011002602A (es) |
| MY (1) | MY152824A (es) |
| NZ (1) | NZ591030A (es) |
| PE (1) | PE20110343A1 (es) |
| TW (1) | TWI454263B (es) |
| UA (1) | UA103496C2 (es) |
| UY (1) | UY32124A (es) |
| WO (1) | WO2010033443A1 (es) |
| ZA (1) | ZA201009151B (es) |
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| UY32099A (es) | 2008-09-11 | 2010-04-30 | Enanta Pharm Inc | Inhibidores macrocíclicos de serina proteasas de hepatitis c |
| PE20110343A1 (es) | 2008-09-17 | 2011-06-25 | Boehringer Ingelheim Int | Combinacion de inhibidor de la proteasa ns3 de hcv con interferon y ribavirina |
| AR075584A1 (es) * | 2009-02-27 | 2011-04-20 | Intermune Inc | COMPOSICIONES TERAPEUTICAS QUE COMPRENDEN beta-D-2'-DESOXI-2'-FLUORO-2'-C-METILCITIDINA Y UN DERIVADO DE ACIDO ISOINDOL CARBOXILICO Y SUS USOS. COMPUESTO. |
| CN102741270B (zh) * | 2009-09-28 | 2015-07-22 | 英特穆恩公司 | C型肝炎病毒复制的环肽抑制剂 |
| EA201200650A1 (ru) * | 2009-10-30 | 2012-12-28 | Бёрингер Ингельхайм Интернациональ Гмбх | Курсы комбинированного лечения вируса гепатита с, включающие bi201335, интерферон-альфа и рибавирин |
| MA34547B1 (fr) * | 2010-09-30 | 2013-09-02 | Boehringer Ingelheim Int | Traitement d'association pour traiter une infection par le vhc |
| EP2658859A4 (en) | 2010-12-30 | 2014-07-30 | Enanta Pharm Inc | MACROCYCLIC HEPATITIS C SERIN PROTEASE INHIBITORS |
| KR20140003521A (ko) | 2010-12-30 | 2014-01-09 | 이난타 파마슈티칼스, 인코포레이티드 | 페난트리딘 매크로사이클릭 c형 간염 세린 프로테아제 억제제 |
| JP2014511516A (ja) * | 2011-01-10 | 2014-05-15 | プロテウス デジタル ヘルス, インコーポレイテッド | 挙動変化を助長するためのシステム、方法および物品 |
| US10201584B1 (en) | 2011-05-17 | 2019-02-12 | Abbvie Inc. | Compositions and methods for treating HCV |
| US8492386B2 (en) | 2011-10-21 | 2013-07-23 | Abbvie Inc. | Methods for treating HCV |
| US8466159B2 (en) | 2011-10-21 | 2013-06-18 | Abbvie Inc. | Methods for treating HCV |
| SE1450131A1 (sv) | 2011-10-21 | 2014-05-07 | Abbvie Inc | DAA-kombinationsbehandling (t.ex. med ABT-072 eller ABT-333)för användning vid behandling av HCV |
| DE112012002748T5 (de) | 2011-10-21 | 2014-07-31 | Abbvie Inc. | Verfahren zur Behandlung von HCV umfassend mindestens zwei direkt wirkende antivirale Wirkstoffe, Ribavirin aber nicht Interferon |
| WO2013137869A1 (en) * | 2012-03-14 | 2013-09-19 | Boehringer Ingelheim International Gmbh | Combination therapy for treating hcv infection in an hcv-hiv coinfected patient population |
| US20140242029A1 (en) * | 2013-02-27 | 2014-08-28 | Boehringer Ingelheim International Gmbh | Combination therapy for treating hcv infection in an hcv-hiv coinfected patient population |
| WO2013147750A1 (en) | 2012-03-27 | 2013-10-03 | Boehringer Ingelheim International Gmbh | Oral combination therapy for treating hcv infection in specific patient sub-population |
| WO2013147749A1 (en) | 2012-03-27 | 2013-10-03 | Boehringer Ingelheim International Gmbh | Oral combination therapy for treating hcv infection in specific patient subgenotype populations |
| WO2013143581A1 (en) | 2012-03-28 | 2013-10-03 | Boehringer Ingelheim International Gmbh | Combination therapy for treating hcv infection in specific patient subgenotype sub-population |
| WO2014138374A1 (en) | 2013-03-08 | 2014-09-12 | Boehringer Ingelheim International Gmbh | Oral combination therapy for treating hcv infection in specific patient sub-population |
| EP3089757A1 (en) | 2014-01-03 | 2016-11-09 | AbbVie Inc. | Solid antiviral dosage forms |
| EA201892448A1 (ru) | 2016-04-28 | 2019-06-28 | Эмори Юниверсити | Алкинсодержащие нуклеотидные и нуклеозидные терапевтические композиции и связанные с ними способы применения |
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| PE20110343A1 (es) | 2008-09-17 | 2011-06-25 | Boehringer Ingelheim Int | Combinacion de inhibidor de la proteasa ns3 de hcv con interferon y ribavirina |
| AR073603A1 (es) | 2008-09-18 | 2010-11-17 | Ortho Mcneil Janssen Pharm | Combinaciones sinergicas de un inhibidor macrociclico del vhc y un nucleosido |
| JP5607736B2 (ja) * | 2009-07-07 | 2014-10-15 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | C型肝炎ウイルスプロテアーゼ阻害剤のための医薬組成物 |
| EA201200650A1 (ru) | 2009-10-30 | 2012-12-28 | Бёрингер Ингельхайм Интернациональ Гмбх | Курсы комбинированного лечения вируса гепатита с, включающие bi201335, интерферон-альфа и рибавирин |
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| MA34547B1 (fr) * | 2010-09-30 | 2013-09-02 | Boehringer Ingelheim Int | Traitement d'association pour traiter une infection par le vhc |
-
2009
- 2009-09-14 PE PE2011000635A patent/PE20110343A1/es not_active Application Discontinuation
- 2009-09-14 UA UAA201104531A patent/UA103496C2/uk unknown
- 2009-09-14 KR KR1020117005679A patent/KR20110054003A/ko not_active Ceased
- 2009-09-14 MY MYPI20111139 patent/MY152824A/en unknown
- 2009-09-14 EA EA201100506A patent/EA019965B1/ru not_active IP Right Cessation
- 2009-09-14 NZ NZ591030A patent/NZ591030A/xx not_active IP Right Cessation
- 2009-09-14 MX MX2011002602A patent/MX2011002602A/es active IP Right Grant
- 2009-09-14 WO PCT/US2009/056771 patent/WO2010033443A1/en not_active Ceased
- 2009-09-14 CA CA2737376A patent/CA2737376A1/en not_active Abandoned
- 2009-09-14 EP EP09792492A patent/EP2337583A1/en not_active Withdrawn
- 2009-09-14 JP JP2011527889A patent/JP5539363B2/ja not_active Expired - Fee Related
- 2009-09-14 BR BRPI0918653A patent/BRPI0918653A2/pt not_active IP Right Cessation
- 2009-09-14 AU AU2009293493A patent/AU2009293493B2/en not_active Ceased
- 2009-09-14 CN CN2009801362929A patent/CN102159245B/zh not_active Expired - Fee Related
- 2009-09-16 US US12/560,752 patent/US8399484B2/en active Active
- 2009-09-16 AR ARP090103556A patent/AR073516A1/es unknown
- 2009-09-16 UY UY0001032124A patent/UY32124A/es not_active Application Discontinuation
- 2009-09-16 TW TW098131293A patent/TWI454263B/zh not_active IP Right Cessation
-
2010
- 2010-12-20 ZA ZA2010/09151A patent/ZA201009151B/en unknown
- 2010-12-21 IL IL210152A patent/IL210152A0/en unknown
-
2011
- 2011-03-09 EC EC2011010877A patent/ECSP11010877A/es unknown
- 2011-03-14 MA MA33700A patent/MA32634B1/fr unknown
- 2011-03-16 CO CO11032826A patent/CO6351753A2/es not_active Application Discontinuation
- 2011-03-17 CL CL2011000571A patent/CL2011000571A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2737376A1 (en) | 2010-03-25 |
| UY32124A (es) | 2010-04-30 |
| WO2010033443A1 (en) | 2010-03-25 |
| TWI454263B (zh) | 2014-10-01 |
| JP5539363B2 (ja) | 2014-07-02 |
| AU2009293493B2 (en) | 2014-09-18 |
| UA103496C2 (uk) | 2013-10-25 |
| EP2337583A1 (en) | 2011-06-29 |
| MA32634B1 (fr) | 2011-09-01 |
| IL210152A0 (en) | 2011-03-31 |
| ZA201009151B (en) | 2011-09-28 |
| PE20110343A1 (es) | 2011-06-25 |
| AR073516A1 (es) | 2010-11-10 |
| TW201016218A (en) | 2010-05-01 |
| ECSP11010877A (es) | 2011-04-29 |
| CN102159245A (zh) | 2011-08-17 |
| JP2012502999A (ja) | 2012-02-02 |
| NZ591030A (en) | 2012-10-26 |
| EA019965B1 (ru) | 2014-07-30 |
| CO6351753A2 (es) | 2011-12-20 |
| MX2011002602A (es) | 2011-04-07 |
| HK1156865A1 (en) | 2012-06-22 |
| AU2009293493A1 (en) | 2010-03-25 |
| CN102159245B (zh) | 2013-07-24 |
| KR20110054003A (ko) | 2011-05-24 |
| US20100068182A1 (en) | 2010-03-18 |
| BRPI0918653A2 (pt) | 2015-12-01 |
| MY152824A (en) | 2014-11-28 |
| EA201100506A1 (ru) | 2011-10-31 |
| US8399484B2 (en) | 2013-03-19 |
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