CL2014003228A1 - Sintesis e intermediarios de compuestos heterocíclicos biologicamente activas. - Google Patents

Sintesis e intermediarios de compuestos heterocíclicos biologicamente activas.

Info

Publication number
CL2014003228A1
CL2014003228A1 CL2014003228A CL2014003228A CL2014003228A1 CL 2014003228 A1 CL2014003228 A1 CL 2014003228A1 CL 2014003228 A CL2014003228 A CL 2014003228A CL 2014003228 A CL2014003228 A CL 2014003228A CL 2014003228 A1 CL2014003228 A1 CL 2014003228A1
Authority
CL
Chile
Prior art keywords
intermediates
synthesis
biologically active
heterocyclic compounds
active heterocyclic
Prior art date
Application number
CL2014003228A
Other languages
English (en)
Inventor
Prabha N Ibrahim
Original Assignee
Plexxikon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48577959&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2014003228(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Plexxikon Inc filed Critical Plexxikon Inc
Publication of CL2014003228A1 publication Critical patent/CL2014003228A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CL2014003228A 2012-05-31 2014-11-27 Sintesis e intermediarios de compuestos heterocíclicos biologicamente activas. CL2014003228A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261653994P 2012-05-31 2012-05-31
US13/793,917 US9150570B2 (en) 2012-05-31 2013-03-11 Synthesis of heterocyclic compounds

Publications (1)

Publication Number Publication Date
CL2014003228A1 true CL2014003228A1 (es) 2015-02-27

Family

ID=48577959

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2014003228A CL2014003228A1 (es) 2012-05-31 2014-11-27 Sintesis e intermediarios de compuestos heterocíclicos biologicamente activas.

Country Status (24)

Country Link
US (2) US9150570B2 (es)
EP (1) EP2861591B1 (es)
JP (1) JP6258301B2 (es)
KR (1) KR102078429B1 (es)
CN (2) CN109608450A (es)
AR (1) AR091159A1 (es)
AU (1) AU2013267325B2 (es)
BR (1) BR112014029454B1 (es)
CA (1) CA2874555C (es)
CL (1) CL2014003228A1 (es)
CR (1) CR20140576A (es)
EA (1) EA027928B1 (es)
EC (1) ECSP14033037A (es)
ES (1) ES2687300T3 (es)
IL (1) IL235819B (es)
MX (1) MX2014014465A (es)
MY (1) MY168935A (es)
NZ (1) NZ630453A (es)
PE (1) PE20142335A1 (es)
PH (1) PH12014502613B1 (es)
SG (1) SG11201407851RA (es)
TW (1) TWI603970B (es)
UY (1) UY34825A (es)
WO (1) WO2013181415A1 (es)

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JP2020511467A (ja) 2017-03-20 2020-04-16 プレキシコン インコーポレーテッドＰｌｅｘｘｉｋｏｎ Ｉｎｃ． ブロモドメインを阻害する４−（１−（１，１−ジ（ピリジン−２−イル）エチル）−６−（３，５−ジメチルイソオキサゾール−４−イル）−１Ｈ−ピロロ［３，２−ｂ］ピリジン−３−イル）安息香酸の結晶形
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EA027928B1 (ru) 2017-09-29
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JP6258301B2 (ja) 2018-01-10
US9695169B2 (en) 2017-07-04
MX2014014465A (es) 2015-02-12
NZ630453A (en) 2017-02-24
JP2015518051A (ja) 2015-06-25
BR112014029454B1 (pt) 2022-03-22
IL235819B (en) 2019-10-31
AR091159A1 (es) 2015-01-14
CN104507937A (zh) 2015-04-08
MY168935A (en) 2019-01-10
TW201406754A (zh) 2014-02-16
KR102078429B1 (ko) 2020-02-17
US9150570B2 (en) 2015-10-06
US20150368243A1 (en) 2015-12-24
KR20150021070A (ko) 2015-02-27
UY34825A (es) 2013-12-31
HK1206010A1 (en) 2015-12-31
CN109608450A (zh) 2019-04-12
PH12014502613A1 (en) 2015-01-21
CA2874555A1 (en) 2013-12-05
PE20142335A1 (es) 2015-01-10
AU2013267325B2 (en) 2017-11-02
CR20140576A (es) 2015-01-30
BR112014029454A2 (pt) 2017-06-27
EA201492165A1 (ru) 2015-05-29
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AU2013267325A1 (en) 2015-01-15
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