CR20120584A - Derivados de n3-sustituido-n1-sulfonil-5-flúorpirimidinona - Google Patents

Derivados de n3-sustituido-n1-sulfonil-5-flúorpirimidinona

Info

Publication number
CR20120584A
CR20120584A CR20120584A CR20120584A CR20120584A CR 20120584 A CR20120584 A CR 20120584A CR 20120584 A CR20120584 A CR 20120584A CR 20120584 A CR20120584 A CR 20120584A CR 20120584 A CR20120584 A CR 20120584A
Authority
CR
Costa Rica
Prior art keywords
derivatives
fluorpirimidinone
sulfonil
substitute
fluoropyrimidinone
Prior art date
Application number
CR20120584A
Other languages
English (en)
Inventor
Timothy Boebel
Beth Lorsbach
Timothy Martin
W John Owen
Michael Sullenberger
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of CR20120584A publication Critical patent/CR20120584A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Dentistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente revelación está relacionada con el campo de N3-sustituido-N1-sulfonil-5-flúorpirimi dinona y sus derivados y el uso de estos compuestos como fungicidas.
CR20120584A 2010-04-26 2012-11-15 Derivados de n3-sustituido-n1-sulfonil-5-flúorpirimidinona CR20120584A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32785510P 2010-04-26 2010-04-26

Publications (1)

Publication Number Publication Date
CR20120584A true CR20120584A (es) 2013-01-03

Family

ID=44816310

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20120584A CR20120584A (es) 2010-04-26 2012-11-15 Derivados de n3-sustituido-n1-sulfonil-5-flúorpirimidinona

Country Status (33)

Country Link
US (1) US8263603B2 (es)
EP (1) EP2563129B1 (es)
JP (1) JP5784705B2 (es)
KR (1) KR101793766B1 (es)
CN (1) CN102946730B (es)
AU (1) AU2011245544B2 (es)
BR (1) BR112012027439B1 (es)
CA (1) CA2797226C (es)
CL (1) CL2012002979A1 (es)
CO (1) CO6592042A2 (es)
CR (1) CR20120584A (es)
CY (1) CY1117956T1 (es)
DK (1) DK2563129T3 (es)
EC (1) ECSP12012302A (es)
ES (1) ES2588742T3 (es)
GT (1) GT201200289A (es)
HN (1) HN2012002272A (es)
HR (1) HRP20161107T1 (es)
HU (1) HUE029489T2 (es)
IL (1) IL222646A (es)
LT (1) LT2563129T (es)
ME (1) ME02530B (es)
MX (1) MX2012012530A (es)
NZ (1) NZ603151A (es)
PH (1) PH12012502138B1 (es)
PL (1) PL2563129T3 (es)
PT (1) PT2563129T (es)
RS (1) RS55239B1 (es)
RU (1) RU2562840C2 (es)
SI (1) SI2563129T1 (es)
SM (1) SMT201600298B (es)
UA (1) UA108101C2 (es)
WO (1) WO2011137002A1 (es)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2471371T3 (es) * 2009-08-07 2014-06-26 Dow Agrosciences Llc Derivados de N1-sulfonil-5-fluoropirimidinona
CA2894510A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2h)-carboxamide derivatives
MX2015008443A (es) * 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de 1-(benzoilo-sustituido) -5-fluoro-4-imino-3-metil-3, 4-dihidropirimidin-2 (1h)-ona.
RU2638556C2 (ru) * 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
AU2013370494B2 (en) 2012-12-31 2017-08-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
NZ722419A (en) * 2013-12-31 2018-01-26 Adama Makhteshim Ltd Synergistic fungicidal mixtures and compositions for fungal control
CA2935594C (en) 2013-12-31 2022-05-03 Nakyen Choy 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
JP6862939B2 (ja) * 2016-03-11 2021-04-21 住友化学株式会社 植物病害防除組成物及び植物病害防除方法
EP3575286B1 (en) * 2017-01-26 2022-05-11 Mitsui Chemicals Agro, Inc. Pyridone compound and bactericide for agricultural and horticultural use, which uses said compound as active ingredient
EP3611166B1 (en) 2017-04-10 2022-09-21 Mitsui Chemicals Agro, Inc. Pyridone compound, and agricultural and horticultural fungicide having this as active component
WO2018190350A1 (ja) 2017-04-10 2018-10-18 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
AU2018251415B2 (en) 2017-04-11 2021-08-05 Mitsui Chemicals Crop & Life Solutions, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
EP3636636B1 (en) 2017-06-08 2022-07-06 Mitsui Chemicals Agro, Inc. Pyridone compound and agricultural and horticultural fungicide
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
EP3828177B1 (en) 2018-07-25 2023-11-29 Mitsui Chemicals Crop & Life Solutions, Inc. Pyridone compound and agricultural and horticultural fungicide having this as active component
EP3876717A1 (en) * 2018-11-05 2021-09-15 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
IL321760A (en) * 2019-07-22 2025-08-01 Adama Makhteshim Ltd Fungicidal combinations, mixtures and compositions and uses thereof
PY2057637A (es) 2019-09-23 2021-10-05 Adama Makhteshim Ltd Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto
CN115776980A (zh) * 2020-03-09 2023-03-10 阿达玛马克西姆有限公司 用于制备5-氟-4-亚氨基-3-甲基-1-(甲苯-4-磺酰基)-3,4-二氢-1h-嘧啶-2-酮的方法
EP4146632A1 (en) 2020-05-04 2023-03-15 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
CA3185119A1 (en) 2020-07-08 2022-01-13 Matteo CERNUSCHI Fungicidal mixtures
BR112023014997A2 (pt) 2021-01-27 2023-10-03 Adama Makhteshim Ltd 5-fluoro-4-imino-3-metil-1-tosil-3,4-di-hidropirimidin-2(1h)-ona para controle de doenças de plantas
US20240237649A1 (en) 2021-05-04 2024-07-18 Adama Makhteshim Ltd. Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof
CN118139845A (zh) * 2021-09-15 2024-06-04 安道麦马克西姆有限公司 用于制备5-氟-4-亚氨基-3-甲基-1-(甲苯-4-磺酰基)-3,4-二氢-1h-嘧啶-2-酮的方法
KR20240132077A (ko) * 2022-01-12 2024-09-02 아다마 마켓심 리미티드 프탈이미드 살진균제를 함유하는 조합물을 포함하는 살진균제 혼합물
UY40172A (es) 2022-03-03 2023-10-13 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
EP4609713A3 (en) 2022-05-26 2025-10-29 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AU2024233301A1 (en) 2023-03-09 2025-09-18 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AU2024236967A1 (en) 2023-03-14 2025-09-25 Adama Makhteshim Ltd. Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber
IL308593A (en) 2023-11-15 2025-06-01 Adama Makhteshim Ltd Reducing environmental impact of fungicidal enhancement
PY24105707A (es) 2023-11-28 2025-06-25 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP970239B1 (en) * 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
CN101312649B (zh) * 2005-11-22 2012-03-28 石原产业株式会社 农业园艺用杀菌剂组合物以及植物病害的防除方法
PT2562166E (pt) * 2008-01-22 2015-10-28 Dow Agrosciences Llc Derivados de 5-fluoro-pirimidina como fungicidas
CN102215691B (zh) * 2008-08-01 2015-02-04 陶氏益农公司 5-氟胞嘧啶作为杀真菌剂的用途
ES2471371T3 (es) * 2009-08-07 2014-06-26 Dow Agrosciences Llc Derivados de N1-sulfonil-5-fluoropirimidinona
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону

Also Published As

Publication number Publication date
ES2588742T3 (es) 2016-11-04
DK2563129T3 (en) 2016-09-12
BR112012027439A2 (pt) 2015-09-15
US8263603B2 (en) 2012-09-11
HRP20161107T1 (hr) 2016-12-30
MX2012012530A (es) 2012-12-17
CA2797226C (en) 2019-02-26
CO6592042A2 (es) 2013-01-02
HN2012002272A (es) 2015-04-27
JP5784705B2 (ja) 2015-09-24
EP2563129A4 (en) 2013-08-07
PH12012502138A1 (en) 2013-02-04
EP2563129A1 (en) 2013-03-06
BR112012027439B1 (pt) 2018-01-16
HK1182594A1 (en) 2013-12-06
CY1117956T1 (el) 2017-05-17
PH12012502138B1 (en) 2019-09-25
HUE029489T2 (en) 2017-02-28
RS55239B1 (sr) 2017-02-28
CA2797226A1 (en) 2011-11-03
US20110263627A1 (en) 2011-10-27
GT201200289A (es) 2014-04-08
UA108101C2 (xx) 2015-03-25
CL2012002979A1 (es) 2013-01-25
BR112012027439A8 (pt) 2017-07-11
AU2011245544B2 (en) 2015-04-16
SMT201600298B (it) 2016-11-10
LT2563129T (lt) 2016-10-25
AU2011245544A1 (en) 2012-11-15
WO2011137002A1 (en) 2011-11-03
IL222646A0 (en) 2012-12-31
EP2563129B1 (en) 2016-06-01
IL222646A (en) 2017-01-31
PL2563129T3 (pl) 2017-08-31
ECSP12012302A (es) 2012-12-28
SI2563129T1 (sl) 2016-12-30
KR101793766B1 (ko) 2017-11-03
RU2562840C2 (ru) 2015-09-10
RU2012150293A (ru) 2014-06-10
NZ603151A (en) 2013-10-25
CN102946730B (zh) 2015-02-04
ME02530B (me) 2017-02-20
JP2013525434A (ja) 2013-06-20
KR20130093000A (ko) 2013-08-21
CN102946730A (zh) 2013-02-27
PT2563129T (pt) 2016-09-05

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