ECSP12012302A - Derivados de n3-sustituido-n1-sulfonil-5-flúorpirimidinona - Google Patents

Derivados de n3-sustituido-n1-sulfonil-5-flúorpirimidinona

Info

Publication number
ECSP12012302A
ECSP12012302A ECSP12012302A ECSP12012302A EC SP12012302 A ECSP12012302 A EC SP12012302A EC SP12012302 A ECSP12012302 A EC SP12012302A EC SP12012302 A ECSP12012302 A EC SP12012302A
Authority
EC
Ecuador
Prior art keywords
derivatives
fluorpirimidinone
sulfonil
substitute
fluoropyrimi
Prior art date
Application number
Other languages
English (en)
Inventor
Timothy Boebel
Beth Lorsbach
Timohy Martin
W John Owen
Michael Sullenberger
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of ECSP12012302A publication Critical patent/ECSP12012302A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente revelación está relacionada con el campo de N3-sustituido-N1-sulfonil-5-flúorpirimi dinona y sus derivados y el uso de estos compuestos como fungicidas.
ECSP12012302 2010-04-26 2012-11-23 Derivados de n3-sustituido-n1-sulfonil-5-flúorpirimidinona ECSP12012302A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32785510P 2010-04-26 2010-04-26

Publications (1)

Publication Number Publication Date
ECSP12012302A true ECSP12012302A (es) 2012-12-28

Family

ID=44816310

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP12012302 ECSP12012302A (es) 2010-04-26 2012-11-23 Derivados de n3-sustituido-n1-sulfonil-5-flúorpirimidinona

Country Status (33)

Country Link
US (1) US8263603B2 (es)
EP (1) EP2563129B1 (es)
JP (1) JP5784705B2 (es)
KR (1) KR101793766B1 (es)
CN (1) CN102946730B (es)
AU (1) AU2011245544B2 (es)
BR (1) BR112012027439B1 (es)
CA (1) CA2797226C (es)
CL (1) CL2012002979A1 (es)
CO (1) CO6592042A2 (es)
CR (1) CR20120584A (es)
CY (1) CY1117956T1 (es)
DK (1) DK2563129T3 (es)
EC (1) ECSP12012302A (es)
ES (1) ES2588742T3 (es)
GT (1) GT201200289A (es)
HN (1) HN2012002272A (es)
HR (1) HRP20161107T1 (es)
HU (1) HUE029489T2 (es)
IL (1) IL222646A (es)
LT (1) LT2563129T (es)
ME (1) ME02530B (es)
MX (1) MX2012012530A (es)
NZ (1) NZ603151A (es)
PH (1) PH12012502138B1 (es)
PL (1) PL2563129T3 (es)
PT (1) PT2563129T (es)
RS (1) RS55239B1 (es)
RU (1) RU2562840C2 (es)
SI (1) SI2563129T1 (es)
SM (1) SMT201600298B (es)
UA (1) UA108101C2 (es)
WO (1) WO2011137002A1 (es)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
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AU2010279411B2 (en) * 2009-08-07 2014-10-23 Adama Makhteshim Ltd. N1-sulfonyl-5-fluoropyrimidinone derivatives
UA117123C2 (uk) * 2012-12-28 2018-06-25 Адама Махтешім Лтд. Похідні 1-(заміщений бензоїл)-5-фтор-4-іміно-3-метил-3,4-дигідропіримідин-2(1h)-ону
RU2015131149A (ru) * 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные
HUE047711T2 (hu) 2012-12-28 2020-05-28 Adama Makhteshim Ltd N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok
CA2894553C (en) 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
EA030030B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
EP3097096A4 (en) * 2013-12-31 2017-10-11 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
JP6862939B2 (ja) * 2016-03-11 2021-04-21 住友化学株式会社 植物病害防除組成物及び植物病害防除方法
JP7037507B2 (ja) * 2017-01-26 2022-03-16 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
CA3059675A1 (en) 2017-04-10 2018-10-18 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides comprising the same as active ingredients
TWI793113B (zh) 2017-04-10 2023-02-21 日商三井化學Agro股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
KR102498819B1 (ko) 2017-04-11 2023-02-10 미쓰이가가쿠 아그로 가부시키가이샤 피리돈 화합물 및 그것을 유효성분으로 하는 농원예용 살균제
US11117863B2 (en) 2017-06-08 2021-09-14 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
EP3828177B1 (en) 2018-07-25 2023-11-29 Mitsui Chemicals Crop & Life Solutions, Inc. Pyridone compound and agricultural and horticultural fungicide having this as active component
CR20210270A (es) * 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
PY2037902A (es) * 2019-07-22 2021-09-29 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
TWI808347B (zh) 2019-09-23 2023-07-11 以色列商亞當馬赫特希姆有限公司 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法
MX2022011088A (es) * 2020-03-09 2022-09-29 Adama Makhteshim Ltd Procedimiento para preparar 5-fluoro-4-imino-3-metil-1-(tolueno-4- sulfonil)-3,4-dihidro-1h-pirimidin-2-ona.
BR112022022281A2 (pt) * 2020-05-04 2023-01-03 Adama Makhteshim Ltd Misturas e composições compreendendo 5-fluoro-4-imino-3-metil- 1-tosil-3,4-dihidropirimidin-2-ona e métodos de uso das mesmas
PE20230375A1 (es) 2020-07-08 2023-03-06 Adama Makhteshim Ltd Mezclas fungicidas
EP4284173A1 (en) 2021-01-27 2023-12-06 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1 h)-one for controlling plant diseases
IL308155A (en) 2021-05-04 2024-01-01 Adama Makhteshim Ltd Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one and mixtures, compositions and methods of using them
CN118139845A (zh) * 2021-09-15 2024-06-04 安道麦马克西姆有限公司 用于制备5-氟-4-亚氨基-3-甲基-1-(甲苯-4-磺酰基)-3,4-二氢-1h-嘧啶-2-酮的方法
WO2023135535A1 (en) * 2022-01-12 2023-07-20 Adama Makhteshim Ltd. Fungicidal mixtures comprising combination containing phthalimide fungicides
UY40172A (es) 2022-03-03 2023-10-13 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
EP4609713A3 (en) 2022-05-26 2025-10-29 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
WO2024184859A1 (en) 2023-03-09 2024-09-12 Conese Salvatore Fungicidal combinations, mixtures and compositions and uses thereof
WO2024189563A1 (en) 2023-03-14 2024-09-19 Adama Makhteshim Ltd. Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber
IL308593A (en) 2023-11-15 2025-06-01 Adama Makhteshim Ltd Reducing environmental impact of fungicidal enhancement
WO2025114931A1 (en) 2023-11-28 2025-06-05 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
CN122422314A (zh) 2023-12-08 2026-07-17 三井化学植保株式会社 双环式杂环化合物以及以双环式杂环化合物作为有效成分的农业园艺用杀菌剂

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP970239B1 (en) * 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
EP1952689A4 (en) * 2005-11-22 2012-12-12 Ishihara Sangyo Kaisha GERMICIDAL COMPOSITION FOR AGRICULTURAL AND GARDENING APPLICATIONS AND METHOD FOR CONTROLLING PLANT DISEASES
AR070228A1 (es) * 2008-01-22 2010-03-25 Dow Agrosciences Llc Derivados de 5-fluoro pirimidina
WO2010047866A2 (en) * 2008-08-01 2010-04-29 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide
AU2010279411B2 (en) * 2009-08-07 2014-10-23 Adama Makhteshim Ltd. N1-sulfonyl-5-fluoropyrimidinone derivatives
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону

Also Published As

Publication number Publication date
ES2588742T3 (es) 2016-11-04
EP2563129A4 (en) 2013-08-07
WO2011137002A1 (en) 2011-11-03
IL222646A0 (en) 2012-12-31
SI2563129T1 (sl) 2016-12-30
EP2563129A1 (en) 2013-03-06
RS55239B1 (sr) 2017-02-28
PH12012502138B1 (en) 2019-09-25
HUE029489T2 (en) 2017-02-28
PL2563129T3 (pl) 2017-08-31
BR112012027439A2 (pt) 2015-09-15
MX2012012530A (es) 2012-12-17
BR112012027439A8 (pt) 2017-07-11
KR20130093000A (ko) 2013-08-21
RU2012150293A (ru) 2014-06-10
KR101793766B1 (ko) 2017-11-03
DK2563129T3 (en) 2016-09-12
NZ603151A (en) 2013-10-25
JP2013525434A (ja) 2013-06-20
CY1117956T1 (el) 2017-05-17
UA108101C2 (xx) 2015-03-25
LT2563129T (lt) 2016-10-25
SMT201600298B (it) 2016-11-10
HN2012002272A (es) 2015-04-27
CN102946730A (zh) 2013-02-27
CA2797226C (en) 2019-02-26
JP5784705B2 (ja) 2015-09-24
CL2012002979A1 (es) 2013-01-25
ME02530B (me) 2017-02-20
US20110263627A1 (en) 2011-10-27
CR20120584A (es) 2013-01-03
AU2011245544A1 (en) 2012-11-15
PT2563129T (pt) 2016-09-05
CO6592042A2 (es) 2013-01-02
CA2797226A1 (en) 2011-11-03
AU2011245544B2 (en) 2015-04-16
CN102946730B (zh) 2015-02-04
EP2563129B1 (en) 2016-06-01
PH12012502138A1 (en) 2013-02-04
BR112012027439B1 (pt) 2018-01-16
IL222646A (en) 2017-01-31
GT201200289A (es) 2014-04-08
US8263603B2 (en) 2012-09-11
RU2562840C2 (ru) 2015-09-10
HRP20161107T1 (hr) 2016-12-30
HK1182594A1 (en) 2013-12-06

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