CR9048A - Analogos de anilino-pirimidina - Google Patents
Analogos de anilino-pirimidinaInfo
- Publication number
- CR9048A CR9048A CR9048A CR9048A CR9048A CR 9048 A CR9048 A CR 9048A CR 9048 A CR9048 A CR 9048A CR 9048 A CR9048 A CR 9048A CR 9048 A CR9048 A CR 9048A
- Authority
- CR
- Costa Rica
- Prior art keywords
- anilino
- pyrimidine analogs
- pyrimidine
- analogs
- compounds
- Prior art date
Links
- 150000008059 anilinopyrimidines Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
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- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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Abstract
La presente invencion se relaciona con compuestos de formula I: en donde R1, R2, R3, R4, R5 y R6 son como se definio aqui.
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| GB9924862D0 (en) | 1999-10-20 | 1999-12-22 | Celltech Therapeutics Ltd | Chemical compounds |
| GB0004888D0 (en) | 2000-03-01 | 2000-04-19 | Astrazeneca Uk Ltd | Chemical compounds |
| AU2001278609B2 (en) * | 2000-08-21 | 2005-04-14 | Astrazeneca Ab | Quinazoline derivatives |
| GB0021726D0 (en) * | 2000-09-05 | 2000-10-18 | Astrazeneca Ab | Chemical compounds |
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| MXPA03005696A (es) * | 2000-12-21 | 2003-10-06 | Glaxo Group Ltd | Pirimidinaminas como moduladores de angiogenesis. |
| US20020132823A1 (en) * | 2001-01-17 | 2002-09-19 | Jiahuai Han | Assay method |
| GB0103926D0 (en) * | 2001-02-17 | 2001-04-04 | Astrazeneca Ab | Chemical compounds |
| BR0207096A (pt) * | 2001-02-20 | 2004-01-20 | Astrazeneca Ab | Uso de um composto, compostos, formulação farmacêutica, e, método de tratamento e/ou profilaxia de condições associadas com a inibição de glicogênio sintase quinase-3 |
| MXPA03008888A (es) * | 2001-03-29 | 2005-03-07 | Vertex Pharma | Inhibidores de n-terminal c-jun cinasas (jnk) y otras proteinas cinasas. |
| CA2443234A1 (en) * | 2001-04-10 | 2002-10-24 | Vertex Pharmaceuticals Incorporated | Isoxaxole derivatives as inhibitors of src and other protein kinases |
| DE60214701T2 (de) * | 2001-04-13 | 2007-09-13 | Vertex Pharmaceuticals Inc., Cambridge | Inhibitoren von c-jun-n-terminalen-kinasen (jnk) und anderen proteinkinasen |
| JP4316893B2 (ja) * | 2001-05-16 | 2009-08-19 | バーテックス ファーマシューティカルズ インコーポレイテッド | Srcおよび他のプロテインキナーゼのインヒビター |
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| WO2002096905A1 (en) | 2001-06-01 | 2002-12-05 | Vertex Pharmaceuticals Incorporated | Thiazole compounds useful as inhibitors of protein kinases |
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| US6703414B2 (en) | 2001-09-14 | 2004-03-09 | Arizona Board Of Regents On Behalf Of The University Of Arizona | Device and method for treating restenosis |
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| CA2477505A1 (en) * | 2002-03-01 | 2003-09-12 | Smithkline Beecham Corporation | Diamino-pyrimidines and their use as angiogenesis inhibitors |
| WO2003076434A1 (en) * | 2002-03-09 | 2003-09-18 | Astrazeneca Ab | 4- imidazolyl substuited pyrimidine derivatives with cdk inhibitiory activity |
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| EP1562911B1 (en) * | 2002-11-01 | 2010-01-06 | Vertex Pharmaceuticals Incorporated | Compositions useful as inhibitors of jak and other protein kinases |
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| GB0226582D0 (en) | 2002-11-14 | 2002-12-18 | Cyclacel Ltd | Anti-viral compounds |
-
2005
- 2005-10-13 US US11/248,495 patent/US7799915B2/en not_active Expired - Fee Related
- 2005-10-13 PE PE2005001207A patent/PE20060582A1/es not_active Application Discontinuation
- 2005-10-13 PA PA20058649401A patent/PA8649401A1/es unknown
- 2005-10-13 MX MX2007004488A patent/MX2007004488A/es unknown
- 2005-10-13 EP EP05812654A patent/EP1799652A1/en not_active Withdrawn
- 2005-10-13 RU RU2007114080/04A patent/RU2007114080A/ru not_active Application Discontinuation
- 2005-10-13 TW TW094135620A patent/TW200626559A/zh unknown
- 2005-10-13 JP JP2007536838A patent/JP2008515986A/ja active Pending
- 2005-10-13 WO PCT/US2005/036674 patent/WO2006044457A1/en not_active Ceased
- 2005-10-13 AR ARP050104293A patent/AR051387A1/es not_active Application Discontinuation
- 2005-10-13 CN CNA2005800349350A patent/CN101039919A/zh not_active Withdrawn
- 2005-10-13 BR BRPI0516597-0A patent/BRPI0516597A/pt not_active IP Right Cessation
- 2005-10-13 AU AU2005295788A patent/AU2005295788A1/en not_active Abandoned
- 2005-10-13 GT GT200500286A patent/GT200500286A/es unknown
- 2005-10-13 KR KR1020077010445A patent/KR20070084067A/ko not_active Withdrawn
- 2005-10-13 CA CA002580913A patent/CA2580913A1/en not_active Abandoned
-
2007
- 2007-03-28 NO NO20071642A patent/NO20071642L/no not_active Application Discontinuation
- 2007-03-29 IL IL182316A patent/IL182316A0/en unknown
- 2007-04-11 CR CR9048A patent/CR9048A/es unknown
- 2007-04-12 ZA ZA200703022A patent/ZA200703022B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2580913A1 (en) | 2006-04-27 |
| RU2007114080A (ru) | 2008-11-27 |
| BRPI0516597A (pt) | 2008-09-16 |
| US7799915B2 (en) | 2010-09-21 |
| CN101039919A (zh) | 2007-09-19 |
| NO20071642L (no) | 2007-06-01 |
| TW200626559A (en) | 2006-08-01 |
| IL182316A0 (en) | 2007-07-24 |
| GT200500286A (es) | 2006-06-13 |
| PA8649401A1 (es) | 2006-09-22 |
| AU2005295788A1 (en) | 2006-04-27 |
| KR20070084067A (ko) | 2007-08-24 |
| AR051387A1 (es) | 2007-01-10 |
| EP1799652A1 (en) | 2007-06-27 |
| PE20060582A1 (es) | 2006-08-17 |
| JP2008515986A (ja) | 2008-05-15 |
| MX2007004488A (es) | 2007-09-11 |
| US20060079543A1 (en) | 2006-04-13 |
| WO2006044457A1 (en) | 2006-04-27 |
| ZA200703022B (en) | 2009-04-29 |
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