CU20200099A7 - Compuestos derivados sustituidos de ácidos 6-carboxílicos de bencimidazoles y 4-aza-, 5-aza y 7-aza- benzimidazoles como agonistas glpr-1 útiles para el tratamiento o prevención de enfermedades cardiometabólicas y asociadas - Google Patents

Compuestos derivados sustituidos de ácidos 6-carboxílicos de bencimidazoles y 4-aza-, 5-aza y 7-aza- benzimidazoles como agonistas glpr-1 útiles para el tratamiento o prevención de enfermedades cardiometabólicas y asociadas

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CU20200099A7
CU20200099A7 CU2020000099A CU20200099A CU20200099A7 CU 20200099 A7 CU20200099 A7 CU 20200099A7 CU 2020000099 A CU2020000099 A CU 2020000099A CU 20200099 A CU20200099 A CU 20200099A CU 20200099 A7 CU20200099 A7 CU 20200099A7
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aza
benzimidazoles
cardiometabolic
prevention
treatment
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CU2020000099A
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English (en)
Inventor
Gary Erik Aspnes
Scott W Bagley
John M Curto
David James Edmons
Mark E Flanagan
Kentaro Futatsugi
David A Griffith
Kim Huard
Yajing Lian
Chris Limberakis
Allyn T Londregan
Alan M Mathiowetz
David W Piotrowski
Roger B Ruggeri
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Pfizer
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Publication of CU20200099A7 publication Critical patent/CU20200099A7/es

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Abstract

<p>Se proporcionan en la presente ácidos 6-carboxílicos de bencimidazoles y 4-aza-, 5-aza- y 7-aza-bencimidazoles como agonistas de GLP-1R de fórmula I</p> <p>ESPACIO PARA LA FÓRMULA</p> <p>útiles para el tratamiento o prevención de enfermedades cardiometabólicas y asociadas.</p>
CU2020000099A 2018-06-13 2019-06-11 Compuestos derivados sustituidos de ácidos 6-carboxílicos de bencimidazoles y 4-aza-, 5-aza y 7-aza- benzimidazoles como agonistas glpr-1 útiles para el tratamiento o prevención de enfermedades cardiometabólicas y asociadas CU20200099A7 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201862684696P 2018-06-13 2018-06-13
US201962846944P 2019-05-13 2019-05-13
US201962851206P 2019-05-22 2019-05-22
PCT/IB2019/054867 WO2019239319A1 (en) 2018-06-13 2019-06-11 Glp-1 receptor agonists and uses thereof

Publications (1)

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CU20200099A7 true CU20200099A7 (es) 2021-08-06

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TWI751585B (zh) 2019-06-28 2022-01-01 美商美國禮來大藥廠 類升糖素肽1受體促效劑
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