CZ20031083A3 - 5-Spiropyrimidin-2, 4, 6-trionové inhibitory metaloproteinasy - Google Patents

5-Spiropyrimidin-2, 4, 6-trionové inhibitory metaloproteinasy Download PDF

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Publication number: CZ20031083A3
Authority: CZ; Czechia
Prior art keywords: group; alkyl; pyridin; triazaspiro; ring
Prior art date: 2000-10-26

Application number

CZ20031083A

Other languages

Czech (cs)

English (en)

Inventor

Brian Scott Bronk

Mark Carl Noe

Martin James Wythes

Original Assignee

Pfizer Products Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-10-26

Filing date

2001-10-23

Publication date

2004-03-17

2001-10-23 Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.

2004-03-17 Publication of CZ20031083A3 publication Critical patent/CZ20031083A3/cs

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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
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- C07D487/10—Spiro-condensed systems

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Immunology (AREA)
Physical Education & Sports Medicine (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Oncology (AREA)
Rheumatology (AREA)
Communicable Diseases (AREA)
Orthopedic Medicine & Surgery (AREA)
Dermatology (AREA)
Pain & Pain Management (AREA)
Pulmonology (AREA)
Gynecology & Obstetrics (AREA)
Diabetes (AREA)
Heart & Thoracic Surgery (AREA)
Ophthalmology & Optometry (AREA)
Tropical Medicine & Parasitology (AREA)
Cardiology (AREA)
Pregnancy & Childbirth (AREA)
Hematology (AREA)
Virology (AREA)
Obesity (AREA)
Psychology (AREA)

CZ20031083A 2000-10-26 2001-10-23 5-Spiropyrimidin-2, 4, 6-trionové inhibitory metaloproteinasy CZ20031083A3 (cs)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US24338900P	2000-10-26	2000-10-26

Publications (1)

Publication Number	Publication Date
CZ20031083A3 true CZ20031083A3 (cs)	2004-03-17

Family

ID=22918584

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CZ20031083A CZ20031083A3 (cs)	2000-10-26	2001-10-23	5-Spiropyrimidin-2, 4, 6-trionové inhibitory metaloproteinasy

Country Status (32)

Country	Link
EP (1)	EP1332146A2 (is)
JP (1)	JP2004518635A (is)
KR (1)	KR20040004412A (is)
CN (1)	CN1501937A (is)
AP (1)	AP2001002318A0 (is)
AR (1)	AR035069A1 (is)
AU (1)	AU2002210813A1 (is)
BG (1)	BG107653A (is)
BR (1)	BR0114913A (is)
CA (1)	CA2425283A1 (is)
CZ (1)	CZ20031083A3 (is)
EA (1)	EA005762B1 (is)
EC (1)	ECSP034567A (is)
EE (1)	EE200300196A (is)
GT (1)	GT200100213A (is)
HN (1)	HN2001000244A (is)
HR (1)	HRP20030332A2 (is)
HU (1)	HUP0301577A3 (is)
IL (1)	IL154948A0 (is)
IS (1)	IS6762A (is)
MA (1)	MA26957A1 (is)
MX (1)	MXPA03003735A (is)
NO (1)	NO20031853L (is)
OA (1)	OA12529A (is)
PA (1)	PA8531401A1 (is)
PE (1)	PE20020589A1 (is)
PL (1)	PL366201A1 (is)
SK (1)	SK4972003A3 (is)
SV (1)	SV2003000705A (is)
TN (1)	TNSN01149A1 (is)
WO (1)	WO2002034753A2 (is)
ZA (1)	ZA200302190B (is)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2002064578A1 (en)	2001-02-14	2002-08-22	Warner-Lambert Company Llc	Benzo thiadiazine matrix metalloproteinase inhibitors
PA8539501A1 (es)	2001-02-14	2002-09-30	Warner Lambert Co	Compuestos triazolo como inhibidores de mmp
DOP2002000333A (es)	2001-02-14	2002-09-30	Warner Lambert Co	Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
JP2004518723A (ja)	2001-02-14	2004-06-24	ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー	ピリミジンマトリックスメタロプロテイナーゼ阻害剤
DOP2002000332A (es)	2001-02-14	2002-08-30	Warner Lambert Co	Inhibidores de piridina de metaloproteinasas de la matriz
US6924276B2 (en)	2001-09-10	2005-08-02	Warner-Lambert Company	Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
WO2003032999A1 (en)	2001-10-12	2003-04-24	Warner-Lambert Company Llc	Alkyne matrix metalloproteinase inhibitors
US6962922B2 (en)	2001-10-12	2005-11-08	Warner-Lambert Company Llc	Alkynylated quinazoline compounds
US6894057B2 (en)	2002-03-08	2005-05-17	Warner-Lambert Company	Oxo-azabicyclic compounds
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2001
- 2001-10-23 CA CA002425283A patent/CA2425283A1/en not_active Abandoned
- 2001-10-23 BR BR0114913-0A patent/BR0114913A/pt not_active IP Right Cessation
- 2001-10-23 EP EP01978721A patent/EP1332146A2/en not_active Withdrawn
- 2001-10-23 PL PL01366201A patent/PL366201A1/xx not_active Application Discontinuation
- 2001-10-23 SK SK497-2003A patent/SK4972003A3/sk unknown
- 2001-10-23 EE EEP200300196A patent/EE200300196A/xx unknown
- 2001-10-23 IL IL15494801A patent/IL154948A0/xx unknown
- 2001-10-23 WO PCT/IB2001/001986 patent/WO2002034753A2/en not_active Ceased
- 2001-10-23 MX MXPA03003735A patent/MXPA03003735A/es unknown
- 2001-10-23 HR HR20030332A patent/HRP20030332A2/hr not_active Application Discontinuation
- 2001-10-23 HU HU0301577A patent/HUP0301577A3/hu unknown
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- 2001-10-23 CN CNA018179231A patent/CN1501937A/zh active Pending
- 2001-10-23 EA EA200300306A patent/EA005762B1/ru not_active IP Right Cessation
- 2001-10-23 JP JP2002537743A patent/JP2004518635A/ja not_active Withdrawn
- 2001-10-23 AU AU2002210813A patent/AU2002210813A1/en not_active Abandoned
- 2001-10-23 KR KR10-2003-7005753A patent/KR20040004412A/ko not_active Ceased
- 2001-10-23 CZ CZ20031083A patent/CZ20031083A3/cs unknown
- 2001-10-23 AP APAP/P/2001/002318A patent/AP2001002318A0/en unknown
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- 2001-10-25 TN TNTNSN01149A patent/TNSN01149A1/fr unknown
- 2001-10-26 PA PA20018531401A patent/PA8531401A1/es unknown
2003
- 2003-03-19 ZA ZA200302190A patent/ZA200302190B/en unknown
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- 2003-03-27 IS IS6762A patent/IS6762A/is unknown
- 2003-04-22 MA MA27117A patent/MA26957A1/fr unknown
- 2003-04-24 NO NO20031853A patent/NO20031853L/no not_active Application Discontinuation
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Also Published As

Publication number	Publication date
AU2002210813A1 (en)	2002-05-06
ECSP034567A (es)	2003-06-25
NO20031853L (no)	2003-06-23
PL366201A1 (en)	2005-01-24
HN2001000244A (es)	2003-11-07
JP2004518635A (ja)	2004-06-24
MXPA03003735A (es)	2003-07-28
EP1332146A2 (en)	2003-08-06
WO2002034753A2 (en)	2002-05-02
SV2003000705A (es)	2003-01-13
EA005762B1 (ru)	2005-06-30
BR0114913A (pt)	2003-07-01
HUP0301577A2 (hu)	2003-11-28
CN1501937A (zh)	2004-06-02
MA26957A1 (fr)	2004-12-20
SK4972003A3 (en)	2004-05-04
BG107653A (bg)	2003-12-31
GT200100213A (es)	2002-07-03
HRP20030332A2 (en)	2003-06-30
KR20040004412A (ko)	2004-01-13
AR035069A1 (es)	2004-04-14
IL154948A0 (en)	2003-10-31
WO2002034753A3 (en)	2002-08-15
EA200300306A1 (ru)	2003-08-28
CA2425283A1 (en)	2002-05-02
AP2001002318A0 (en)	2001-12-31
EE200300196A (et)	2003-10-15
OA12529A (en)	2006-06-02
TNSN01149A1 (fr)	2005-11-10
IS6762A (is)	2003-03-27
PE20020589A1 (es)	2002-07-06
ZA200302190B (en)	2004-04-28
NO20031853D0 (no)	2003-04-24
PA8531401A1 (es)	2003-06-30
HUP0301577A3 (en)	2006-02-28

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