ECSP034567A - Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas - Google Patents

Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas

Info

Publication number: ECSP034567A
Authority: EC; Ecuador
Prior art keywords: spiropirimidin; triona; inhibitors; metaloproteinase inhibitors; metaloproteinase
Prior art date: 2000-10-26

Application number

EC2003004567A

Other languages

English (en)

Spanish (es)

Inventor

Mark Carl Noe

Martin James Wythes

Brian S Bronk

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-10-26

Filing date

2003-04-25

Publication date

2003-06-25

2003-04-25 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2003-06-25 Publication of ECSP034567A publication Critical patent/ECSP034567A/es

Links

239000003112 inhibitor Substances 0.000 title abstract 2
125000003341 7 membered heterocyclic group Chemical group 0.000 abstract 1
206010061218 Inflammation Diseases 0.000 abstract 1
102000005741 Metalloproteases Human genes 0.000 abstract 1
108010006035 Metalloproteases Proteins 0.000 abstract 1
206010028980 Neoplasm Diseases 0.000 abstract 1
201000011510 cancer Diseases 0.000 abstract 1
230000004054 inflammatory process Effects 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
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Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Physical Education & Sports Medicine (AREA)
Immunology (AREA)
Reproductive Health (AREA)
Endocrinology (AREA)
Rheumatology (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Dermatology (AREA)
Orthopedic Medicine & Surgery (AREA)
Pain & Pain Management (AREA)
Pulmonology (AREA)
Gynecology & Obstetrics (AREA)
Diabetes (AREA)
Virology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Pregnancy & Childbirth (AREA)
Tropical Medicine & Parasitology (AREA)
Ophthalmology & Optometry (AREA)
Hematology (AREA)
Vascular Medicine (AREA)
Psychiatry (AREA)

EC2003004567A 2000-10-26 2003-04-25 Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas ECSP034567A (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US24338900P	2000-10-26	2000-10-26

Publications (1)

Publication Number	Publication Date
ECSP034567A true ECSP034567A (es)	2003-06-25

Family

ID=22918584

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EC2003004567A ECSP034567A (es)	2000-10-26	2003-04-25	Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas

Country Status (32)

Country	Link
EP (1)	EP1332146A2 (is)
JP (1)	JP2004518635A (is)
KR (1)	KR20040004412A (is)
CN (1)	CN1501937A (is)
AP (1)	AP2001002318A0 (is)
AR (1)	AR035069A1 (is)
AU (1)	AU2002210813A1 (is)
BG (1)	BG107653A (is)
BR (1)	BR0114913A (is)
CA (1)	CA2425283A1 (is)
CZ (1)	CZ20031083A3 (is)
EA (1)	EA005762B1 (is)
EC (1)	ECSP034567A (is)
EE (1)	EE200300196A (is)
GT (1)	GT200100213A (is)
HN (1)	HN2001000244A (is)
HR (1)	HRP20030332A2 (is)
HU (1)	HUP0301577A3 (is)
IL (1)	IL154948A0 (is)
IS (1)	IS6762A (is)
MA (1)	MA26957A1 (is)
MX (1)	MXPA03003735A (is)
NO (1)	NO20031853L (is)
OA (1)	OA12529A (is)
PA (1)	PA8531401A1 (is)
PE (1)	PE20020589A1 (is)
PL (1)	PL366201A1 (is)
SK (1)	SK4972003A3 (is)
SV (1)	SV2003000705A (is)
TN (1)	TNSN01149A1 (is)
WO (1)	WO2002034753A2 (is)
ZA (1)	ZA200302190B (is)

Families Citing this family (40)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
MXPA03005870A (es)	2001-02-14	2005-02-14	Warner Lambert Co	Inhibirores de benzotiadiazina de metaloproteinasas de la matriz.
DOP2002000332A (es)	2001-02-14	2002-08-30	Warner Lambert Co	Inhibidores de piridina de metaloproteinasas de la matriz
JP2004518723A (ja)	2001-02-14	2004-06-24	ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー	ピリミジンマトリックスメタロプロテイナーゼ阻害剤
DOP2002000333A (es)	2001-02-14	2002-09-30	Warner Lambert Co	Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
PA8539501A1 (es)	2001-02-14	2002-09-30	Warner Lambert Co	Compuestos triazolo como inhibidores de mmp
US6924276B2 (en)	2001-09-10	2005-08-02	Warner-Lambert Company	Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
US6962922B2 (en)	2001-10-12	2005-11-08	Warner-Lambert Company Llc	Alkynylated quinazoline compounds
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2001
- 2001-10-23 CZ CZ20031083A patent/CZ20031083A3/cs unknown
- 2001-10-23 PL PL01366201A patent/PL366201A1/xx not_active Application Discontinuation
- 2001-10-23 BR BR0114913-0A patent/BR0114913A/pt not_active IP Right Cessation
- 2001-10-23 HU HU0301577A patent/HUP0301577A3/hu unknown
- 2001-10-23 IL IL15494801A patent/IL154948A0/xx unknown
- 2001-10-23 AP APAP/P/2001/002318A patent/AP2001002318A0/en unknown
- 2001-10-23 KR KR10-2003-7005753A patent/KR20040004412A/ko not_active Ceased
- 2001-10-23 AU AU2002210813A patent/AU2002210813A1/en not_active Abandoned
- 2001-10-23 EE EEP200300196A patent/EE200300196A/xx unknown
- 2001-10-23 HR HR20030332A patent/HRP20030332A2/hr not_active Application Discontinuation
- 2001-10-23 SK SK497-2003A patent/SK4972003A3/sk unknown
- 2001-10-23 CA CA002425283A patent/CA2425283A1/en not_active Abandoned
- 2001-10-23 EP EP01978721A patent/EP1332146A2/en not_active Withdrawn
- 2001-10-23 CN CNA018179231A patent/CN1501937A/zh active Pending
- 2001-10-23 EA EA200300306A patent/EA005762B1/ru not_active IP Right Cessation
- 2001-10-23 JP JP2002537743A patent/JP2004518635A/ja not_active Withdrawn
- 2001-10-23 MX MXPA03003735A patent/MXPA03003735A/es unknown
- 2001-10-23 WO PCT/IB2001/001986 patent/WO2002034753A2/en not_active Ceased
- 2001-10-23 OA OA1200300123A patent/OA12529A/en unknown
- 2001-10-24 HN HN2001000244A patent/HN2001000244A/es unknown
- 2001-10-24 AR ARP010104977A patent/AR035069A1/es unknown
- 2001-10-25 SV SV2001000705A patent/SV2003000705A/es unknown
- 2001-10-25 PE PE2001001060A patent/PE20020589A1/es not_active Application Discontinuation
- 2001-10-25 GT GT200100213A patent/GT200100213A/es unknown
- 2001-10-25 TN TNTNSN01149A patent/TNSN01149A1/fr unknown
- 2001-10-26 PA PA20018531401A patent/PA8531401A1/es unknown
2003
- 2003-03-19 ZA ZA200302190A patent/ZA200302190B/en unknown
- 2003-03-20 BG BG107653A patent/BG107653A/bg unknown
- 2003-03-27 IS IS6762A patent/IS6762A/is unknown
- 2003-04-22 MA MA27117A patent/MA26957A1/fr unknown
- 2003-04-24 NO NO20031853A patent/NO20031853L/no not_active Application Discontinuation
- 2003-04-25 EC EC2003004567A patent/ECSP034567A/es unknown

Also Published As

Publication number	Publication date
CN1501937A (zh)	2004-06-02
NO20031853L (no)	2003-06-23
PL366201A1 (en)	2005-01-24
MXPA03003735A (es)	2003-07-28
AP2001002318A0 (en)	2001-12-31
SV2003000705A (es)	2003-01-13
TNSN01149A1 (fr)	2005-11-10
ZA200302190B (en)	2004-04-28
GT200100213A (es)	2002-07-03
KR20040004412A (ko)	2004-01-13
IS6762A (is)	2003-03-27
BG107653A (bg)	2003-12-31
HN2001000244A (es)	2003-11-07
JP2004518635A (ja)	2004-06-24
SK4972003A3 (en)	2004-05-04
EP1332146A2 (en)	2003-08-06
WO2002034753A2 (en)	2002-05-02
IL154948A0 (en)	2003-10-31
HUP0301577A3 (en)	2006-02-28
CA2425283A1 (en)	2002-05-02
HRP20030332A2 (en)	2003-06-30
WO2002034753A3 (en)	2002-08-15
EE200300196A (et)	2003-10-15
AU2002210813A1 (en)	2002-05-06
MA26957A1 (fr)	2004-12-20
PE20020589A1 (es)	2002-07-06
NO20031853D0 (no)	2003-04-24
HUP0301577A2 (hu)	2003-11-28
OA12529A (en)	2006-06-02
EA005762B1 (ru)	2005-06-30
AR035069A1 (es)	2004-04-14
PA8531401A1 (es)	2003-06-30
EA200300306A1 (ru)	2003-08-28
BR0114913A (pt)	2003-07-01
CZ20031083A3 (cs)	2004-03-17

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PA8531401A1 (es)	2003-06-30	Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas
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HN2000000137A (es)	2001-02-02	Pirimidina-2,4,6-trionas inhibidores de metaloproteinasas
SE0001899D0 (sv)	2000-05-22	New compounds
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