CZ2003553A3 - Farmaceutický prostředek - Google Patents

Farmaceutický prostředek Download PDF

Info

Publication number: CZ2003553A3
Authority: CZ; Czechia
Prior art keywords: agent; pharmaceutical composition; aminolevulinic acid; composition according; photochemotherapeutic
Prior art date: 2000-07-27

Application number

CZ2003553A

Other languages

Czech (cs)

English (en)

Inventor

Jo Klaveness

Vidar Hansson

Aslak Godal

Original Assignee

Photocure Asa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-07-27

Filing date

2001-07-25

Publication date

2003-06-18

2001-07-25 Application filed by Photocure Asa filed Critical Photocure Asa

2003-06-18 Publication of CZ2003553A3 publication Critical patent/CZ2003553A3/cs

Links

239000008194 pharmaceutical composition Substances 0.000 title claims abstract description 25
239000003795 chemical substances by application Substances 0.000 claims abstract description 134
230000003232 mucoadhesive effect Effects 0.000 claims abstract description 57
230000002215 photochemotherapeutic effect Effects 0.000 claims abstract description 54
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims abstract description 33
208000035475 disorder Diseases 0.000 claims abstract description 30
230000005856 abnormality Effects 0.000 claims abstract description 29
239000002738 chelating agent Substances 0.000 claims abstract description 20
238000003745 diagnosis Methods 0.000 claims abstract description 16
239000003814 drug Substances 0.000 claims abstract description 14
239000000203 mixture Substances 0.000 claims description 70
150000002148 esters Chemical class 0.000 claims description 38
ZGXJTSGNIOSYLO-UHFFFAOYSA-N 88755TAZ87 Chemical compound NCC(=O)CCC(O)=O ZGXJTSGNIOSYLO-UHFFFAOYSA-N 0.000 claims description 37
-1 5-aminolevulinic acid ester Chemical class 0.000 claims description 35
229960002749 aminolevulinic acid Drugs 0.000 claims description 30
150000001875 compounds Chemical class 0.000 claims description 26
238000000034 method Methods 0.000 claims description 26
150000003839 salts Chemical class 0.000 claims description 26
125000000217 alkyl group Chemical group 0.000 claims description 21
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FEBUJFMRSBAMES-UHFFFAOYSA-N 2-[(2-{[3,5-dihydroxy-2-(hydroxymethyl)-6-phosphanyloxan-4-yl]oxy}-3,5-dihydroxy-6-({[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}methyl)oxan-4-yl)oxy]-3,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl phosphinite Chemical class OC1C(O)C(O)C(CO)OC1OCC1C(O)C(OC2C(C(OP)C(O)C(CO)O2)O)C(O)C(OC2C(C(CO)OC(P)C2O)O)O1 FEBUJFMRSBAMES-UHFFFAOYSA-N 0.000 claims description 5
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IXPNQXFRVYWDDI-UHFFFAOYSA-N 1-methyl-2,4-dioxo-1,3-diazinane-5-carboximidamide Chemical compound CN1CC(C(N)=N)C(=O)NC1=O IXPNQXFRVYWDDI-UHFFFAOYSA-N 0.000 claims description 4
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NBIIXXVUZAFLBC-UHFFFAOYSA-K phosphate Chemical group [O-]P([O-])([O-])=O NBIIXXVUZAFLBC-UHFFFAOYSA-K 0.000 claims description 3
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QAOWNCQODCNURD-UHFFFAOYSA-L sulfate group Chemical group S(=O)(=O)([O-])[O-] QAOWNCQODCNURD-UHFFFAOYSA-L 0.000 claims description 3
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BECPQYXYKAMYBN-UHFFFAOYSA-N casein, tech. Chemical compound NCCCCC(C(O)=O)N=C(O)C(CC(O)=O)N=C(O)C(CCC(O)=N)N=C(O)C(CC(C)C)N=C(O)C(CCC(O)=O)N=C(O)C(CC(O)=O)N=C(O)C(CCC(O)=O)N=C(O)C(C(C)O)N=C(O)C(CCC(O)=N)N=C(O)C(CCC(O)=N)N=C(O)C(CCC(O)=N)N=C(O)C(CCC(O)=O)N=C(O)C(CCC(O)=O)N=C(O)C(COP(O)(O)=O)N=C(O)C(CCC(O)=N)N=C(O)C(N)CC1=CC=CC=C1 BECPQYXYKAMYBN-UHFFFAOYSA-N 0.000 claims description 2
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Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Epidemiology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Virology (AREA)
Molecular Biology (AREA)
Physiology (AREA)
Dermatology (AREA)
Biochemistry (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Pulmonology (AREA)
Nutrition Science (AREA)
Otolaryngology (AREA)
Ophthalmology & Optometry (AREA)
Biotechnology (AREA)
Gynecology & Obstetrics (AREA)
Medicinal Preparation (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Confectionery (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

CZ2003553A 2000-07-27 2001-07-25 Farmaceutický prostředek CZ2003553A3 (cs)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GBGB0018527.2A GB0018527D0 (en)	2000-07-27	2000-07-27	Composition

Publications (1)

Publication Number	Publication Date
CZ2003553A3 true CZ2003553A3 (cs)	2003-06-18

Family

ID=9896499

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CZ2003553A CZ2003553A3 (cs)	2000-07-27	2001-07-25	Farmaceutický prostředek

Country Status (15)

Country	Link
US (1)	US20040029855A1 (de)
EP (1)	EP1311259B1 (de)
JP (1)	JP2004505040A (de)
KR (1)	KR20030046394A (de)
CN (1)	CN1633285A (de)
AT (1)	ATE297723T1 (de)
AU (2)	AU2002224594B2 (de)
CA (1)	CA2417533A1 (de)
CZ (1)	CZ2003553A3 (de)
DE (1)	DE60111539T2 (de)
ES (1)	ES2243572T3 (de)
GB (1)	GB0018527D0 (de)
HU (1)	HUP0301452A3 (de)
RU (1)	RU2003105461A (de)
WO (1)	WO2002009690A2 (de)

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2000
- 2000-07-27 GB GBGB0018527.2A patent/GB0018527D0/en not_active Ceased
2001
- 2001-07-25 CN CNA018146961A patent/CN1633285A/zh active Pending
- 2001-07-25 JP JP2002515243A patent/JP2004505040A/ja active Pending
- 2001-07-25 RU RU2003105461/15A patent/RU2003105461A/ru not_active Application Discontinuation
- 2001-07-25 CZ CZ2003553A patent/CZ2003553A3/cs unknown
- 2001-07-25 HU HU0301452A patent/HUP0301452A3/hu unknown
- 2001-07-25 KR KR10-2003-7001217A patent/KR20030046394A/ko not_active Withdrawn
- 2001-07-25 US US10/343,211 patent/US20040029855A1/en not_active Abandoned
- 2001-07-25 AT AT01984399T patent/ATE297723T1/de not_active IP Right Cessation
- 2001-07-25 ES ES01984399T patent/ES2243572T3/es not_active Expired - Lifetime
- 2001-07-25 DE DE60111539T patent/DE60111539T2/de not_active Expired - Lifetime
- 2001-07-25 AU AU2002224594A patent/AU2002224594B2/en not_active Ceased
- 2001-07-25 EP EP01984399A patent/EP1311259B1/de not_active Expired - Lifetime
- 2001-07-25 WO PCT/GB2001/003338 patent/WO2002009690A2/en not_active Ceased
- 2001-07-25 AU AU2459402A patent/AU2459402A/xx active Pending
- 2001-07-25 CA CA002417533A patent/CA2417533A1/en not_active Abandoned

Also Published As

Publication number	Publication date
WO2002009690A2 (en)	2002-02-07
DE60111539T2 (de)	2006-05-11
JP2004505040A (ja)	2004-02-19
HUP0301452A3 (en)	2005-05-30
AU2002224594B2 (en)	2006-03-09
ES2243572T3 (es)	2005-12-01
DE60111539D1 (de)	2005-07-21
ATE297723T1 (de)	2005-07-15
AU2459402A (en)	2002-02-13
RU2003105461A (ru)	2004-06-27
CA2417533A1 (en)	2002-02-07
HUP0301452A2 (hu)	2003-08-28
CN1633285A (zh)	2005-06-29
EP1311259B1 (de)	2005-06-15
EP1311259A2 (de)	2003-05-21
WO2002009690A8 (en)	2004-04-15
US20040029855A1 (en)	2004-02-12
GB0018527D0 (en)	2000-09-13
WO2002009690A3 (en)	2002-08-08
KR20030046394A (ko)	2003-06-12

Publication	Publication Date	Title
AU2002224594B2 (en)	2006-03-09	Pharmaceutical composition comprising a photochemotherapeutic agent and a mucoadhesive agent
AU2002224594A1 (en)	2002-05-09	Pharmaceutical composition comprising a photochemotherapeutic agent and a mucoadhesive agent
JP5686603B2 (ja)	2015-03-18	使用
CN1137087C (zh)	2004-02-04	用作光化学疗法中的光致敏剂的5-氨基酮戊酸的酯
JP4740524B2 (ja)	2011-08-03	熱応答粘膜接着性医薬−担体組成物
US6750212B2 (en)	2004-06-15	Photochemotherapeutic compositions
US8410172B2 (en)	2013-04-02	Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy
US20110293528A1 (en)	2011-12-01	Enema preparations and their use
CN101631541A (zh)	2010-01-20	氨基酮戊酸及其衍生物的应用
HUP0401192A2 (hu)	2004-12-28	Fényérzékenyítő szer alkalmazása sebek kezelésére adható gyógyászati készítmény előállítására
JP2007500227A (ja)	2007-01-11	光増感剤及び音増感剤と関連してのニトロキシドの使用方法
US20110223105A1 (en)	2011-09-15	New 5-aminolevulinic acid prodrugs for use in photodynamic therapy and photodynamic diagnosis
JP2001518498A (ja)	2001-10-16	空洞器官内腫瘍の全体的診断および／または治療用局所医薬製造のためのδ−アミノレブリン酸の利用
JP2002538201A (ja)	2002-11-12	癌を診断および治療する手段
CZ244799A3 (cs)	2000-02-16	Farmaceutický prostředek