CZ297975B6 - Farmaceutická kombinace antagonisty receptoru proangiotensin II a epoxymexrenonu pro lécení kardiovaskulárních poruch - Google Patents

Farmaceutická kombinace antagonisty receptoru proangiotensin II a epoxymexrenonu pro lécení kardiovaskulárních poruch Download PDF

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Publication number
CZ297975B6
CZ297975B6 CZ0385097A CZ385097A CZ297975B6 CZ 297975 B6 CZ297975 B6 CZ 297975B6 CZ 0385097 A CZ0385097 A CZ 0385097A CZ 385097 A CZ385097 A CZ 385097A CZ 297975 B6 CZ297975 B6 CZ 297975B6
Authority
CZ
Czechia
Prior art keywords
angiotensin
receptor antagonist
antagonist
epoxymexrenone
receptor
Prior art date
Application number
CZ0385097A
Other languages
Czech (cs)
English (en)
Other versions
CZ385097A3 (cs
Inventor
C. Alexander@John
R. Schuh@Joseph
J. Gorczynski@Richard
Original Assignee
G. D. Searle & Co.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by G. D. Searle & Co. filed Critical G. D. Searle & Co.
Publication of CZ385097A3 publication Critical patent/CZ385097A3/cs
Publication of CZ297975B6 publication Critical patent/CZ297975B6/cs

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Organic Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
CZ0385097A 1995-06-07 1996-06-05 Farmaceutická kombinace antagonisty receptoru proangiotensin II a epoxymexrenonu pro lécení kardiovaskulárních poruch CZ297975B6 (cs)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US48645695A 1995-06-07 1995-06-07

Publications (2)

Publication Number Publication Date
CZ385097A3 CZ385097A3 (cs) 1998-06-17
CZ297975B6 true CZ297975B6 (cs) 2007-05-09

Family

ID=23931955

Family Applications (1)

Application Number Title Priority Date Filing Date
CZ0385097A CZ297975B6 (cs) 1995-06-07 1996-06-05 Farmaceutická kombinace antagonisty receptoru proangiotensin II a epoxymexrenonu pro lécení kardiovaskulárních poruch

Country Status (21)

Country Link
US (1) US6653306B1 (2)
EP (1) EP0831910B1 (2)
JP (1) JPH11507627A (2)
KR (1) KR100618466B1 (2)
CN (2) CN1522701A (2)
AT (1) ATE209047T1 (2)
AU (1) AU725689B2 (2)
BR (1) BR9609066A (2)
CA (1) CA2224079A1 (2)
CZ (1) CZ297975B6 (2)
DE (1) DE69617235T2 (2)
DK (1) DK0831910T3 (2)
ES (1) ES2167571T3 (2)
IL (1) IL122242A (2)
NO (1) NO318184B1 (2)
NZ (1) NZ310730A (2)
PL (1) PL185150B1 (2)
PT (1) PT831910E (2)
RO (1) RO118046B1 (2)
RU (1) RU2166330C2 (2)
WO (1) WO1996040257A1 (2)

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ES2269442T3 (es) * 2000-07-27 2007-04-01 Pharmacia Corporation Terapia de combinacion de antagonista de aldosterona e inhibidor de ciclooxigenasa-2 para prevenir o tratar trastornos cardiovasculares relacionados con la inflamacion.
AU2002351412B2 (en) 2001-12-21 2010-05-20 Exelixis Patent Company Llc Modulators of LXR
US7482366B2 (en) 2001-12-21 2009-01-27 X-Ceptor Therapeutics, Inc. Modulators of LXR
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EA200870409A1 (ru) 2006-04-04 2009-04-28 Дзе Риджентс Оф Дзе Юниверсити Оф Калифорния Антагонисты киназы pi3
GB2467670B (en) 2007-10-04 2012-08-01 Intellikine Inc Chemical entities and therapeutic uses thereof
CA2711558C (en) * 2008-01-04 2016-12-13 Intellikine, Inc. Phosphatidyl inositol-3 kinase inhibiting compounds
US8193182B2 (en) 2008-01-04 2012-06-05 Intellikine, Inc. Substituted isoquinolin-1(2H)-ones, and methods of use thereof
JP5547099B2 (ja) 2008-03-14 2014-07-09 インテリカイン， エルエルシー キナーゼ阻害剤および使用方法
US8993580B2 (en) 2008-03-14 2015-03-31 Intellikine Llc Benzothiazole kinase inhibitors and methods of use
AU2009268611B2 (en) 2008-07-08 2015-04-09 Intellikine, Llc Kinase inhibitors and methods of use
WO2010006072A2 (en) 2008-07-08 2010-01-14 The Regents Of The University Of California Mtor modulators and uses thereof
JP5731978B2 (ja) 2008-09-26 2015-06-10 インテリカイン， エルエルシー 複素環キナーゼ阻害剤
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JP6027610B2 (ja) 2011-07-19 2016-11-16 インフィニティー ファーマシューティカルズ， インコーポレイテッド 複素環式化合物及びその使用
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Also Published As

Publication number Publication date
JPH11507627A (ja) 1999-07-06
RU2166330C2 (ru) 2001-05-10
KR100618466B1 (ko) 2006-12-13
CA2224079A1 (en) 1996-12-19
CZ385097A3 (cs) 1998-06-17
KR19990022548A (ko) 1999-03-25
DE69617235T2 (de) 2002-07-25
RO118046B1 (ro) 2003-01-30
DK0831910T3 (da) 2002-05-21
CN1522701A (zh) 2004-08-25
DE69617235D1 (de) 2002-01-03
PT831910E (pt) 2002-05-31
AU725689B2 (en) 2000-10-19
ATE209047T1 (de) 2001-12-15
CN1192697A (zh) 1998-09-09
NO318184B1 (no) 2005-02-14
AU6157796A (en) 1996-12-30
CN1142793C (zh) 2004-03-24
EP0831910B1 (en) 2001-11-21
BR9609066A (pt) 1999-01-26
EP0831910A1 (en) 1998-04-01
ES2167571T3 (es) 2002-05-16
IL122242A0 (en) 1998-04-05
PL324001A1 (en) 1998-04-27
NO975741D0 (no) 1997-12-05
US6653306B1 (en) 2003-11-25
NO975741L (no) 1998-01-29
NZ310730A (en) 2001-01-26
WO1996040257A1 (en) 1996-12-19
PL185150B1 (pl) 2003-03-31
IL122242A (en) 2001-07-24

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Date Code Title Description
PD00 Pending as of 2000-06-30 in czech republic
MM4A Patent lapsed due to non-payment of fee

Effective date: 20090605