BRPI0906473A8 - Certas entidades químicas, composições e métodos - Google Patents

Certas entidades químicas, composições e métodos

Info

Publication number
BRPI0906473A8
BRPI0906473A8 BRPI0906473A BRPI0906473A BRPI0906473A8 BR PI0906473 A8 BRPI0906473 A8 BR PI0906473A8 BR PI0906473 A BRPI0906473 A BR PI0906473A BR PI0906473 A BRPI0906473 A BR PI0906473A BR PI0906473 A8 BRPI0906473 A8 BR PI0906473A8
Authority
BR
Brazil
Prior art keywords
chemical entities
methods
compositions
certain chemical
kinase activity
Prior art date
Application number
BRPI0906473A
Other languages
English (en)
Inventor
Ren Pingda
Liu Yi
Troy Wilson Edward
Li Liansheng
Chan Katrina
Rommel Christian
Original Assignee
Intellikine Inc
Intellikine Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Intellikine Inc, Intellikine Llc filed Critical Intellikine Inc
Publication of BRPI0906473A2 publication Critical patent/BRPI0906473A2/pt
Publication of BRPI0906473A8 publication Critical patent/BRPI0906473A8/pt

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
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    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

CERTAS ENTIDADES QUÍMICAS, COMPOSIÇÕES E MÉTODOS se refere a entidades químicas que modulam a atividade da Pl3 quinase e entidades químicas, composições farmacêuticas e métodos de tratamento de doenças e condições associadas a atividade de PI3 quinase.
BRPI0906473A 2008-01-04 2009-01-05 Certas entidades químicas, composições e métodos BRPI0906473A8 (pt)

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