DD157614A5 - Verfahren zur herstellung von pyrimidyl-chinazolinen - Google Patents
Verfahren zur herstellung von pyrimidyl-chinazolinen Download PDFInfo
- Publication number
- DD157614A5 DD157614A5 DD81228589A DD22858981A DD157614A5 DD 157614 A5 DD157614 A5 DD 157614A5 DD 81228589 A DD81228589 A DD 81228589A DD 22858981 A DD22858981 A DD 22858981A DD 157614 A5 DD157614 A5 DD 157614A5
- Authority
- DD
- German Democratic Republic
- Prior art keywords
- formula
- compound
- atoms
- amino
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pretreatment Of Seeds And Plants (AREA)
- Catching Or Destruction (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19803011809 DE3011809A1 (de) | 1980-03-27 | 1980-03-27 | Pyrimidyl-chinazoline, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und ihre verwendung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DD157614A5 true DD157614A5 (de) | 1982-11-24 |
Family
ID=6098481
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DD81228589A DD157614A5 (de) | 1980-03-27 | 1981-03-25 | Verfahren zur herstellung von pyrimidyl-chinazolinen |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP0037495A1 (da) |
| JP (1) | JPS56150088A (da) |
| AR (1) | AR227542A1 (da) |
| AU (1) | AU6877481A (da) |
| CA (1) | CA1156656A (da) |
| CS (1) | CS219898B2 (da) |
| DD (1) | DD157614A5 (da) |
| DE (1) | DE3011809A1 (da) |
| DK (1) | DK115581A (da) |
| ES (1) | ES8202000A1 (da) |
| FI (1) | FI810778A7 (da) |
| GR (1) | GR71870B (da) |
| IL (1) | IL62495A0 (da) |
| NO (1) | NO810870L (da) |
| PL (2) | PL230320A1 (da) |
| PT (1) | PT72724B (da) |
| SU (1) | SU1052158A3 (da) |
| ZA (1) | ZA812034B (da) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS61140568A (ja) * | 1984-12-14 | 1986-06-27 | Mitsui Petrochem Ind Ltd | キナゾリン誘導体及びそれを有効成分とする血圧降下剤 |
| JPS6267077A (ja) * | 1985-09-18 | 1987-03-26 | Mitsui Petrochem Ind Ltd | キナゾリン誘導体及び医薬 |
| CN102079743B (zh) * | 2004-03-15 | 2020-08-25 | 武田药品工业株式会社 | 二肽基肽酶抑制剂 |
| US7576076B2 (en) * | 2004-07-02 | 2009-08-18 | Corcept Therapeutics, Inc. | Modified pyrimidine glucocorticoid receptor modulators |
| CN103596431B (zh) | 2011-03-18 | 2016-06-22 | 科赛普特治疗公司 | 嘧啶环己基糖皮质激素受体调节剂 |
| CA3102099C (en) | 2018-06-04 | 2023-09-26 | Corcept Therapeutics Incorporated | Pyrimidine cyclohexenyl glucocorticoid receptor modulators |
| JP7569492B2 (ja) | 2019-12-11 | 2024-10-18 | コーセプト セラピューティクス， インコーポレイテッド | 抗精神病薬誘発性体重増加のミリコリラントによる治療方法 |
| KR102911885B1 (ko) | 2020-05-06 | 2026-01-12 | 코어셉트 쎄라퓨틱스 인코포레이티드 | 피리미딘 사이클로헥실 글루코코르티코이드 수용체 조절제의 다형체 |
| AU2021266739B2 (en) | 2020-05-06 | 2024-11-28 | Corcept Therapeutics Incorporated | Formulations of pyrimidine cyclohexyl glucocorticoid receptor modulators |
| JP7853982B2 (ja) | 2020-12-21 | 2026-04-30 | コーセプト セラピューティクス， インコーポレイテッド | ピリミジンシクロヘキシルグルココルチコイド受容体調節因子を調製する方法 |
| US12616698B2 (en) | 2021-05-05 | 2026-05-05 | Corcept Therapeutics Incorporated | Methods for reducing liver fat and for treating fatty liver disorders |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2007656B (en) * | 1977-11-05 | 1982-05-19 | Pfizer Ltd | Therapeutic agents |
-
1980
- 1980-03-27 DE DE19803011809 patent/DE3011809A1/de not_active Withdrawn
- 1980-12-15 GR GR64485A patent/GR71870B/el unknown
-
1981
- 1981-03-13 FI FI810778A patent/FI810778A7/fi not_active Application Discontinuation
- 1981-03-13 NO NO810870A patent/NO810870L/no unknown
- 1981-03-13 DK DK115581A patent/DK115581A/da not_active Application Discontinuation
- 1981-03-20 EP EP81102088A patent/EP0037495A1/de not_active Ceased
- 1981-03-24 PT PT72724A patent/PT72724B/pt unknown
- 1981-03-25 PL PL23032081A patent/PL230320A1/xx unknown
- 1981-03-25 DD DD81228589A patent/DD157614A5/de unknown
- 1981-03-25 CS CS812182A patent/CS219898B2/cs unknown
- 1981-03-25 PL PL23388281A patent/PL233882A1/xx unknown
- 1981-03-25 SU SU813261941A patent/SU1052158A3/ru active
- 1981-03-25 JP JP4257181A patent/JPS56150088A/ja active Pending
- 1981-03-26 ES ES500738A patent/ES8202000A1/es not_active Expired
- 1981-03-26 AR AR284752A patent/AR227542A1/es active
- 1981-03-26 IL IL62495A patent/IL62495A0/xx unknown
- 1981-03-26 CA CA000373945A patent/CA1156656A/en not_active Expired
- 1981-03-26 ZA ZA00812034A patent/ZA812034B/xx unknown
- 1981-03-26 AU AU68774/81A patent/AU6877481A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| SU1052158A3 (ru) | 1983-10-30 |
| PT72724B (de) | 1982-03-24 |
| ZA812034B (en) | 1982-05-26 |
| IL62495A0 (en) | 1981-05-20 |
| CS219898B2 (en) | 1983-03-25 |
| AU6877481A (en) | 1981-10-01 |
| PL233882A1 (da) | 1982-05-10 |
| DK115581A (da) | 1981-09-28 |
| FI810778L (fi) | 1981-09-28 |
| FI810778A7 (fi) | 1981-09-28 |
| EP0037495A1 (de) | 1981-10-14 |
| JPS56150088A (en) | 1981-11-20 |
| DE3011809A1 (de) | 1981-10-01 |
| ES500738A0 (es) | 1982-01-16 |
| PL230320A1 (da) | 1982-03-29 |
| ES8202000A1 (es) | 1982-01-16 |
| GR71870B (da) | 1983-07-08 |
| NO810870L (no) | 1981-09-28 |
| AR227542A1 (es) | 1982-11-15 |
| CA1156656A (en) | 1983-11-08 |
| PT72724A (de) | 1981-04-01 |
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