DK0476935T3 - Nye indol- og indolinforbindelser - Google Patents

Nye indol- og indolinforbindelser

Info

Publication number: DK0476935T3
Authority: DK; Denmark
Prior art keywords: alkyl; indoline compounds; new indole; compounds; phenyl
Prior art date: 1990-09-18

Application number

DK91308365.5T

Other languages

Danish (da)

English (en)

Inventor

Jeremy Gilmore

Original Assignee

Lilly Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-09-18

Filing date

1991-09-12

Publication date

1995-09-11

1991-09-12 Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd

1995-09-11 Application granted granted Critical

1995-09-11 Publication of DK0476935T3 publication Critical patent/DK0476935T3/da

Links

SIKJAQJRHWYJAI-UHFFFAOYSA-N Indole Chemical compound C1=CC=C2NC=CC2=C1 SIKJAQJRHWYJAI-UHFFFAOYSA-N 0.000 title 2
PZOUSPYUWWUPPK-UHFFFAOYSA-N indole Natural products CC1=CC=CC2=C1C=CN2 PZOUSPYUWWUPPK-UHFFFAOYSA-N 0.000 title 1
RKJUIXBNRJVNHR-UHFFFAOYSA-N indolenine Natural products C1=CC=C2CC=NC2=C1 RKJUIXBNRJVNHR-UHFFFAOYSA-N 0.000 title 1
125000003387 indolinyl group Chemical class N1(CCC2=CC=CC=C12)* 0.000 title 1
125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
125000000008 (C1-C10) alkyl group Chemical class 0.000 abstract 1
125000006374 C2-C10 alkenyl group Chemical class 0.000 abstract 1
239000003199 leukotriene receptor blocking agent Substances 0.000 abstract 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Pulmonology (AREA)
Immunology (AREA)
Vascular Medicine (AREA)
Diabetes (AREA)
Hematology (AREA)
Dermatology (AREA)
Indole Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK91308365.5T 1990-09-18 1991-09-12 Nye indol- og indolinforbindelser DK0476935T3 (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB909020338A GB9020338D0 (en)	1990-09-18	1990-09-18	Pharmaceutical compounds

Publications (1)

Publication Number	Publication Date
DK0476935T3 true DK0476935T3 (da)	1995-09-11

Family

ID=10682362

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK91308365.5T DK0476935T3 (da)	1990-09-18	1991-09-12	Nye indol- og indolinforbindelser

Country Status (10)

Country	Link
US (1)	US5185361A (fr)
EP (1)	EP0476935B1 (fr)
JP (1)	JP3046861B2 (fr)
AT (1)	ATE125530T1 (fr)
CA (1)	CA2051460C (fr)
DE (1)	DE69111541T2 (fr)
DK (1)	DK0476935T3 (fr)
ES (1)	ES2076477T3 (fr)
GB (1)	GB9020338D0 (fr)
GR (1)	GR3017390T3 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1998015530A1 (fr) *	1996-10-08	1998-04-16	Fujisawa Pharmaceutical Co., Ltd.	Derives d'indol
WO1999000372A1 (fr) *	1997-06-27	1999-01-07	Fujisawa Pharmaceutical Co., Ltd.	Sulfamides et leur utilisation medicale
EP1283199A4 (fr) *	2000-05-16	2003-12-17	Takeda Chemical Industries Ltd	Antagoniste de l'hormone de concentration de la melanine
KR20050059294A (ko) *	2002-10-24	2005-06-17	스테릭스 리미티드	11-베타-하이드록시 스테로이드 데하이드로게나제 형태 1및 형태 2의 억제제
GB0224830D0 (en) *	2002-10-24	2002-12-04	Sterix Ltd	Compound

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4448784A (en) *	1982-04-12	1984-05-15	Hoechst-Roussel Pharmaceuticals, Inc.	1-(Aminoalkylphenyl and aminoalkylbenzyl)-indoles and indolines and analgesic method of use thereof
GB8524157D0 (en) *	1984-10-19	1985-11-06	Ici America Inc	Heterocyclic amides
GB8707051D0 (en) *	1986-04-15	1987-04-29	Ici America Inc	Heterocyclic carboxamides
GB8927981D0 (en) *	1989-12-11	1990-02-14	Ici Plc	Carbamoyl derivative

1990
- 1990-09-18 GB GB909020338A patent/GB9020338D0/en active Pending
1991
- 1991-09-12 AT AT91308365T patent/ATE125530T1/de not_active IP Right Cessation
- 1991-09-12 DE DE69111541T patent/DE69111541T2/de not_active Expired - Fee Related
- 1991-09-12 EP EP91308365A patent/EP0476935B1/fr not_active Expired - Lifetime
- 1991-09-12 DK DK91308365.5T patent/DK0476935T3/da active
- 1991-09-12 ES ES91308365T patent/ES2076477T3/es not_active Expired - Lifetime
- 1991-09-16 CA CA002051460A patent/CA2051460C/fr not_active Expired - Fee Related
- 1991-09-17 JP JP3236530A patent/JP3046861B2/ja not_active Expired - Lifetime
- 1991-09-18 US US07/761,587 patent/US5185361A/en not_active Expired - Lifetime
1995
- 1995-09-13 GR GR950402508T patent/GR3017390T3/el unknown

Also Published As

Publication number	Publication date
ES2076477T3 (es)	1995-11-01
ATE125530T1 (de)	1995-08-15
EP0476935B1 (fr)	1995-07-26
JPH04230661A (ja)	1992-08-19
CA2051460A1 (fr)	1992-03-19
DE69111541T2 (de)	1996-01-18
EP0476935A1 (fr)	1992-03-25
CA2051460C (fr)	2002-01-22
GR3017390T3 (en)	1995-12-31
US5185361A (en)	1993-02-09
JP3046861B2 (ja)	2000-05-29
DE69111541D1 (de)	1995-08-31
GB9020338D0 (en)	1990-10-31

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