DK0719779T3 - Substituerede thiazolo[3,2-alpha]azepinderivater - Google Patents

Substituerede thiazolo[3,2-alpha]azepinderivater

Info

Publication number: DK0719779T3
Authority: DK; Denmark
Prior art keywords: group; hydrogen atom; lower alkyl; alpha; substituted
Prior art date: 1994-07-18

Application number

DK95921127T

Other languages

Danish (da)

English (en)

Inventor

Hideyuki Adachi

Hitoshi Oinuma

Kazutoshi Miyake

Mamoru Saito

Takeshi Sudo

Shinji Suda

Naoki Yoneda

Makoto Kotake

Masanori Mizuno

Tomohiro Matsushima

Yoshio Fukuda

Toshiyuki Matsuoka

Masayuki Namiki

Makoto Okita

Original Assignee

Eisai Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-07-18

Filing date

1995-06-07

Publication date

2004-03-22

1994-07-18 Priority claimed from JP6165481A external-priority patent/JPH0827156A/ja

1994-08-24 Priority claimed from JP19918094A external-priority patent/JP3444666B2/ja

1994-12-09 Priority claimed from JP6306468A external-priority patent/JPH08165293A/ja

1995-06-07 Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd

2004-03-22 Application granted granted Critical

2004-03-22 Publication of DK0719779T3 publication Critical patent/DK0719779T3/da

Links

150000001538 azepines Chemical class 0.000 title 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 6
125000000217 alkyl group Chemical group 0.000 abstract 3
125000003545 alkoxy group Chemical group 0.000 abstract 2
125000004414 alkyl thio group Chemical group 0.000 abstract 2
125000006239 protecting group Chemical group 0.000 abstract 2
125000001424 substituent group Chemical group 0.000 abstract 2
102000004270 Peptidyl-Dipeptidase A Human genes 0.000 abstract 1
108090000882 Peptidyl-Dipeptidase A Proteins 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
230000002401 inhibitory effect Effects 0.000 abstract 1
230000007935 neutral effect Effects 0.000 abstract 1
125000003396 thiol group Chemical group [H]S* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Immunology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Thiazole And Isothizaole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK95921127T 1994-07-18 1995-06-07 Substituerede thiazolo[3,2-alpha]azepinderivater DK0719779T3 (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
JP6165481A JPH0827156A (ja)	1994-07-18	1994-07-18	アミノ酸誘導体の製造方法
JP19918094A JP3444666B2 (ja)	1994-08-24	1994-08-24	（２ｓ，３ｓ）−３− メチル−２− チオペンタン酸誘導体の製造方法
JP6306468A JPH08165293A (ja)	1994-12-09	1994-12-09	置換チアゾロ［３，２−ａ］アゼピン誘導体
PCT/JP1995/001139 WO1996002549A1 (en)	1994-07-18	1995-06-07	SUBSTITUTED THIAZOLO[3,2-α]AZEPINE DERIVATIVE

Publications (1)

Publication Number	Publication Date
DK0719779T3 true DK0719779T3 (da)	2004-03-22

Family

ID=27322514

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK95921127T DK0719779T3 (da)	1994-07-18	1995-06-07	Substituerede thiazolo[3,2-alpha]azepinderivater

Country Status (17)

Country	Link
US (2)	US5789403A (de)
EP (1)	EP0719779B1 (de)
KR (1)	KR100284247B1 (de)
CN (2)	CN1053908C (de)
AT (1)	ATE254622T1 (de)
AU (1)	AU694233B2 (de)
CA (1)	CA2171334C (de)
DE (1)	DE69532155T2 (de)
DK (1)	DK0719779T3 (de)
ES (1)	ES2210292T3 (de)
FI (2)	FI110001B (de)
HU (1)	HU225916B1 (de)
MX (1)	MX9601017A (de)
NO (1)	NO308077B1 (de)
NZ (1)	NZ287557A (de)
PT (1)	PT719779E (de)
WO (1)	WO1996002549A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5650408A (en) *	1995-06-07	1997-07-22	Karanewsky; Donald S.	Thiazolo benzazepine containing dual action inhibitors
AU738269B2 (en) *	1997-02-05	2001-09-13	Asubio Pharma Co., Ltd.	Pharmaceutical composition for treatment of heart disease based on cardiac hypertrophy
US9823092B2 (en)	2014-10-31	2017-11-21	Allegro Microsystems, Llc	Magnetic field sensor providing a movement detector

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA821904B (en) *	1981-03-23	1983-01-26	Merck & Co Inc	Bicyclic lactams as anthihypertensives
US4415496A (en) *	1981-03-23	1983-11-15	Merck & Co., Inc.	Bicyclic lactams
US4617301A (en) *	1983-06-22	1986-10-14	Merck & Co., Inc.	Sulfoxide and sulfone derivatives of bicyclic lactams as antihypertensives
JPS6056790A (ja) *	1983-09-03	1985-04-02	山陽科学株式会社	荷役用マット
RU2124503C1 (ru) *	1992-05-18	1999-01-10	И.Р.Сквибб энд Санз, Инк.	Гетероциклические азотсодержащие производные карбоновой кислоты, способ их получения и фармацевтическая композиция
PT669936E (pt) *	1992-10-30	2001-04-30	Merrell Pharma Inc	Derivados de lactama biciclica de mercaptoacetilamida uteis como inibidores de encefalinase e de ace
US5650408A (en) *	1995-06-07	1997-07-22	Karanewsky; Donald S.	Thiazolo benzazepine containing dual action inhibitors

1995
- 1995-06-07 US US08/612,864 patent/US5789403A/en not_active Expired - Lifetime
- 1995-06-07 ES ES95921127T patent/ES2210292T3/es not_active Expired - Lifetime
- 1995-06-07 MX MX9601017A patent/MX9601017A/es not_active IP Right Cessation
- 1995-06-07 CN CN95190779A patent/CN1053908C/zh not_active Expired - Fee Related
- 1995-06-07 DE DE69532155T patent/DE69532155T2/de not_active Expired - Fee Related
- 1995-06-07 WO PCT/JP1995/001139 patent/WO1996002549A1/ja not_active Ceased
- 1995-06-07 AU AU26301/95A patent/AU694233B2/en not_active Ceased
- 1995-06-07 AT AT95921127T patent/ATE254622T1/de not_active IP Right Cessation
- 1995-06-07 NZ NZ287557A patent/NZ287557A/en not_active IP Right Cessation
- 1995-06-07 CA CA002171334A patent/CA2171334C/en not_active Expired - Fee Related
- 1995-06-07 PT PT95921127T patent/PT719779E/pt unknown
- 1995-06-07 HU HU9600679A patent/HU225916B1/hu not_active IP Right Cessation
- 1995-06-07 EP EP95921127A patent/EP0719779B1/de not_active Expired - Lifetime
- 1995-06-07 KR KR1019960701358A patent/KR100284247B1/ko not_active Expired - Fee Related
- 1995-06-07 DK DK95921127T patent/DK0719779T3/da active
1996
- 1996-03-14 NO NO19961051A patent/NO308077B1/no not_active IP Right Cessation
- 1996-03-14 FI FI961199A patent/FI110001B/fi active
1998
- 1998-05-27 US US09/085,729 patent/US6051705A/en not_active Expired - Fee Related
1999
- 1999-10-28 CN CNB991236092A patent/CN1170832C/zh not_active Expired - Fee Related
2001
- 2001-06-01 FI FI20011154A patent/FI113656B/fi not_active IP Right Cessation

Also Published As

Publication number	Publication date
ES2210292T3 (es)	2004-07-01
CN1262275A (zh)	2000-08-09
EP0719779B1 (de)	2003-11-19
NO961051D0 (no)	1996-03-14
US5789403A (en)	1998-08-04
PT719779E (pt)	2004-04-30
CN1053908C (zh)	2000-06-28
CN1170832C (zh)	2004-10-13
HU225916B1 (en)	2007-12-28
EP0719779A4 (de)	1996-12-18
NO308077B1 (no)	2000-07-17
DE69532155T2 (de)	2004-08-19
FI110001B (fi)	2002-11-15
WO1996002549A1 (en)	1996-02-01
ATE254622T1 (de)	2003-12-15
CA2171334A1 (en)	1996-02-01
KR100284247B1 (ko)	2001-10-24
HU9600679D0 (en)	1996-05-28
FI113656B (fi)	2004-05-31
FI961199A7 (fi)	1996-05-13
NO961051L (no)	1996-05-10
DE69532155D1 (de)	2003-12-24
MX9601017A (es)	1997-10-31
NZ287557A (en)	1997-04-24
HUT76477A (en)	1997-09-29
KR960704898A (ko)	1996-10-09
US6051705A (en)	2000-04-18
FI20011154L (fi)	2001-06-01
FI961199A0 (fi)	1996-03-14
CN1134152A (zh)	1996-10-23
AU2630195A (en)	1996-02-16
EP0719779A1 (de)	1996-07-03
AU694233B2 (en)	1998-07-16
CA2171334C (en)	2008-10-21

Publication	Publication Date	Title
NO994582D0 (no)	1999-09-21	Fremgangsmaate for fremstilling av piperidinderivater
NO923528L (no)	1992-11-12	3-benzyliden-1-karbamoyl-2-pyrrolidonanaloger
DE69609325D1 (de)	2000-08-17	Derivate des radicicols
TW264476B (de)	1995-12-01
NZ304438A (en)	1999-04-29	Substituted triazole derivatives and antifungal compositions
DK0806413T3 (da)	2002-01-28	2-substituerede viatmin D3-derivater
DE69532155D1 (de)	2003-12-24	Substituierte thiazolo [3,2-alpha]azepinderivate
DE69930383D1 (de)	2006-05-11	Naphthimidobenzamid-derivate
DE69416683D1 (de)	1999-04-01	Benzolactam-derivate
DE69714841D1 (de)	2002-09-26	Ein 1-methylcarbapenem-derivat
DE69629152D1 (de)	2003-08-28	Penem-derivate und sie enthaltende anti-mikrobische mittel
NO20004477L (no)	2001-03-12	Anvendelse av organiske karbonater for vasking av metalloverflater