DK0770615T3 - Fremgangsmåde til fremstilling af dihalogenazolopyrimidiner - Google Patents

Fremgangsmåde til fremstilling af dihalogenazolopyrimidiner

Info

Publication number: DK0770615T3
Authority: DK; Denmark
Prior art keywords: dihalogenazolopyrimidines; preparation
Prior art date: 1995-10-27

Application number

DK96307528T

Other languages

Danish (da)

English (en)

Inventor

Guenther Krummel

Karl-Otto Stumm

Klaus-Juergen Pees

Peter Heinz Rudi Liers

Original Assignee

Basf Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-10-27

Filing date

1996-10-16

Publication date

2003-07-14

1996-10-16 Application filed by Basf Ag filed Critical Basf Ag

2003-07-14 Application granted granted Critical

2003-07-14 Publication of DK0770615T3 publication Critical patent/DK0770615T3/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK96307528T 1995-10-27 1996-10-16 Fremgangsmåde til fremstilling af dihalogenazolopyrimidiner DK0770615T3 (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US802295P	1995-10-27	1995-10-27

Publications (1)

Publication Number	Publication Date
DK0770615T3 true DK0770615T3 (da)	2003-07-14

Family

ID=21729405

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK96307528T DK0770615T3 (da)	1995-10-27	1996-10-16	Fremgangsmåde til fremstilling af dihalogenazolopyrimidiner

Country Status (22)

Country	Link
US (1)	US5808066A (fr)
EP (1)	EP0770615B1 (fr)
JP (1)	JP4018182B2 (fr)
KR (1)	KR100443182B1 (fr)
AR (1)	AR004122A1 (fr)
AT (1)	ATE243211T1 (fr)
BR (1)	BR9605258A (fr)
CA (1)	CA2188905C (fr)
DE (1)	DE69628712T2 (fr)
DK (1)	DK0770615T3 (fr)
ES (1)	ES2202419T3 (fr)
HU (1)	HU217773B (fr)
IL (1)	IL119496A (fr)
MX (1)	MX9604882A (fr)
PT (1)	PT770615E (fr)
RU (1)	RU2147584C1 (fr)
SG (1)	SG55239A1 (fr)
SI (1)	SI0770615T1 (fr)
SK (1)	SK284071B6 (fr)
TR (1)	TR199600792A2 (fr)
UA (1)	UA48132C2 (fr)
ZA (1)	ZA968957B (fr)

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US6117876A (en)	1997-04-14	2000-09-12	American Cyanamid Company	Fungicidal trifluorophenyl-triazolopyrimidines
HUP0100885A3 (en) *	1998-02-11	2002-12-28	American Cyanamid Company Madi	Fungicidal 7-alkyl-triazolopyrimidines
US6117865A (en) *	1998-09-10	2000-09-12	American Cyanamid Company	Fungicidal trifluorophenyl-triazolopyrimidines
US6156925A (en) *	1998-09-25	2000-12-05	American Cyanamid Company	Process for the preparation of halogenated phenylmaloates
US6242451B1 (en) *	1998-09-25	2001-06-05	Klaus-Juergen Pees	Fungicidal trihalophenyl-triazolopyrimidines
US6380202B1 (en) *	1998-09-25	2002-04-30	Basf Aktiengesellschaft	Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines
US6559151B2 (en)	2000-05-08	2003-05-06	Basf Aktiengesellschaft	6-(2-trifluoromethyl-phenyl)-triazolopyrimidines
US6756379B2 (en)	2001-07-26	2004-06-29	Taro Pharmaceutical Industries Ltd.	Non-sedating barbiturate compounds as neuroprotective agents
US7683071B2 (en) *	2000-07-26	2010-03-23	Taro Pharmaceuticals Industries Ltd.	Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
US6939873B2 (en) *	2000-07-26	2005-09-06	Taro Pharmaceuticals Industries Limited	Non-sedating barbituric acid derivatives
DE10063115A1 (de) *	2000-12-18	2002-06-27	Bayer Ag	Triazolopyrimidine
JP2002249492A (ja) *	2000-12-22	2002-09-06	Nippon Bayer Agrochem Co Ltd	トリアゾロピリミジン類
DE10121101A1 (de) *	2001-04-27	2002-10-31	Bayer Ag	Triazolopyrimidine
KR100619216B1 (ko)	2001-07-05	2006-09-08	바스프 악티엔게젤샤프트	살진균성 트리아졸로피리미딘, 이의 제조방법 및 유해진균 방제를 위한 이의 용도 및 상기 화합물을 포함하는조성물
US7038047B2 (en)	2001-07-18	2006-05-02	Basf Aktiengesellschaft	Substituted 6-(2-methoxyphenyl) triazolopyrimides as fungicides
HUP0401488A2 (hu)	2001-07-26	2004-12-28	Basf Aktiengesellschaft	Fungicid hatású 7-amino-triazolopirimidinek, előállításuk, alkalmazásuk és ilyeneket tartalmazó készítmények
ES2287312T3 (es)	2001-09-04	2007-12-16	Sumitomo Chemical Company, Limited	Imidazo(1,2-a)pirimidinas y composiciones fungicidas que las contienen.
CA2479766A1 (fr)	2002-03-21	2003-10-02	Basf Aktiengesellschaft	Triazolopyrimidines fongicides, leur procede de production et leur utilisation pour lutter contre des champignons nuisibles, et agents les contenant
WO2004052350A2 (fr) *	2002-12-11	2004-06-24	Taro Pharmaceutical Industries Limited	Methode de traitement de troubles moteurs a l'aide de derives de l'acide barbiturique
US7419982B2 (en) *	2003-09-24	2008-09-02	Wyeth Holdings Corporation	Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
SI1680425T1 (sl) *	2003-09-24	2007-04-30	Wyeth Corp	6-((substituirani)fenil)triazolopirimidini kot sredstva proti raku
ES2308256T3 (es) *	2003-09-24	2008-12-01	Wyeth Holdings Corporation	6-aril-7-halo-imidazo(1,2-a)pirimidinas como agentes anticancerosos.
MY179926A (en) *	2003-12-08	2020-11-19	Wyeth Corp	Process for the preparation of tubulin inhibitors
TW200533670A (en) *	2003-12-19	2005-10-16	Basf Ag	6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
DE102004007076A1 (de) *	2004-02-13	2005-08-25	Bayer Cropscience Ag	Imidazolopyrimidine
DE502005009862D1 (de) *	2004-03-10	2010-08-19	Basf Se	5,6-dialkyl-7-aminotriazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
EP1725560B1 (fr) *	2004-03-10	2010-07-07	Basf Se	5,6-dialkyl-7-amino-triazolopyrimidines, procedes pour leur production, leur utilisation pour lutter contre des champignons nuisibles, ainsi qu'agents les contenant
PE20060020A1 (es) *	2004-03-30	2006-03-10	Basf Ag	5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion
WO2006003651A2 (fr) *	2004-07-02	2006-01-12	Taro Pharmaceutical Industries, Ltd	Procede de preparation d'acide 1-methoxymethyl-5,5-diphenylbarbiturique
JP2008536806A (ja) *	2005-03-01	2008-09-11	ビーエーエスエフソシエタス・ヨーロピア	５，６−ジアルキル−７−アミノアゾロピリミジン、それらの製造方法、植物病原性菌類を防除するためのそれらの使用、および該化合物を含む薬剤
JP2008532944A (ja) *	2005-03-01	2008-08-21	ビーエーエスエフソシエタス・ヨーロピア	５，６−ジアルキル−７−アミノアゾロピリミジン、それらの製造方法、有害な菌類を防除するためのそれらの使用、およびそれらの化合物を含む物質
JP2008531653A (ja) *	2005-03-01	2008-08-14	ビーエーエスエフソシエタス・ヨーロピア	５，６−ジアルキル−７−アミノアゾロピリミジン類、その調製法および有害菌類を防除するためのその使用、ならびにこれらの化合物を含む組成物
US20080139581A1 (en) *	2005-03-02	2008-06-12	Basf Aktiengesellschaft	2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds
US20080176744A1 (en) *	2005-03-10	2008-07-24	Basf Aktiengesellschaft	Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them
US20080146839A1 (en) *	2005-03-18	2008-06-19	Basf Aktiengesellschaft	Method for Producing 5-Halo-2,4,6-Trifluoroisophthalic Acid
CN101208289A (zh) *	2005-06-27	2008-06-25	巴斯福股份公司	生产取代的苯基丙二酸酯中间体化合物的方法及其在生产5,7-二羟基-6-(2,4,6-三氟苯基)[1,2,4]三唑并[1,5-a]嘧啶中的用途
CN101208287A (zh) *	2005-06-27	2008-06-25	巴斯福股份公司	生产取代的苯基丙二酸酯的方法，新的苯基丙二酸酯及其用途
EP2081576A4 (fr) *	2006-11-14	2010-06-30	Taro Pharmaceuticals North Ame	Procédé d'amélioration de la biodisponibilité pour les barbituriques non sédatifs
WO2008084082A1 (fr) *	2007-01-11	2008-07-17	Basf Se	Procédé de production de pyrimidines annelées, substituées par aryle
US8343977B2 (en) *	2009-12-30	2013-01-01	Arqule, Inc.	Substituted triazolo-pyrimidine compounds

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AU557300B2 (en) *	1982-03-16	1986-12-18	Farmitalia Carlo Erba S.P.A.	Substituted 1h-pyrazolo(1,5-alpha)pyrimidines and processes for their preparation
JPS5962593A (ja) *	1982-09-30	1984-04-10	Ss Pharmaceut Co Ltd	３―置換―５，７―ジクロルトリアゾロピリミジン誘導体
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US4910306A (en) *	1987-11-09	1990-03-20	The Dow Chemical Company	Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US4892945A (en) *	1987-12-21	1990-01-09	Ciba-Geigy Corporation	Isoindoline pigments containing at least one triazolopyrimidone radical
US5006656A (en) *	1990-02-26	1991-04-09	Dowelanco	Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
KR100191774B1 (ko) *	1991-04-22	1999-06-15	오스카 아끼히꼬	피라졸로[1,5-알파] 피리미딘 유도체 및 이것을 함유하는 항염증제
US5356897A (en) *	1991-09-09	1994-10-18	Fujisawa Pharmaceutical Co., Ltd.	3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines
US5177206A (en) *	1991-10-08	1993-01-05	Dowelanco	Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides
TW224044B (fr) *	1991-12-30	1994-05-21	Shell Internat Res Schappej B V
IL108731A (en) *	1993-03-04	1997-03-18	Shell Int Research	6, N-DISUBSTITUTED-£1, 2, 4\| TRIAZOLO-£1, 5-a\| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
RU2066295C1 (ru) *	1993-05-19	1996-09-10	Институт структурной макрокинетики РАН	Способ получения порошкового материала на основе карбида титана
EP0628559B1 (fr) *	1993-06-10	2002-04-03	Beiersdorf-Lilly GmbH	Composés de pyrimidine et leur application comme agents pharmaceutiques
DE69429728T2 (de) *	1993-10-18	2002-10-31	Dow Agrosciences Llc, Indianapolis	Verfahren zur herstellung von n-(2,6-dichloro-3-methylphenyl)-5-7-dihalo[1,2,4]triazolo[1,5a]pyrimidin-2-sulfonamid durch cyclisierung und halo-dehydroxylierung

1996
- 1996-09-30 RU RU96120421A patent/RU2147584C1/ru not_active IP Right Cessation
- 1996-10-03 TR TR96/00792A patent/TR199600792A2/xx unknown
- 1996-10-15 US US08/729,204 patent/US5808066A/en not_active Expired - Lifetime
- 1996-10-16 MX MX9604882A patent/MX9604882A/es not_active IP Right Cessation
- 1996-10-16 DK DK96307528T patent/DK0770615T3/da active
- 1996-10-16 AT AT96307528T patent/ATE243211T1/de not_active IP Right Cessation
- 1996-10-16 DE DE69628712T patent/DE69628712T2/de not_active Expired - Lifetime
- 1996-10-16 SI SI9630630T patent/SI0770615T1/xx unknown
- 1996-10-16 PT PT96307528T patent/PT770615E/pt unknown
- 1996-10-16 ES ES96307528T patent/ES2202419T3/es not_active Expired - Lifetime
- 1996-10-16 EP EP96307528A patent/EP0770615B1/fr not_active Expired - Lifetime
- 1996-10-18 SG SG1996010896A patent/SG55239A1/en unknown
- 1996-10-23 UA UA96104029A patent/UA48132C2/uk unknown
- 1996-10-23 JP JP29790396A patent/JP4018182B2/ja not_active Expired - Fee Related
- 1996-10-24 ZA ZA9608957A patent/ZA968957B/xx unknown
- 1996-10-25 SK SK1377-96A patent/SK284071B6/sk unknown
- 1996-10-25 BR BR9605258A patent/BR9605258A/pt not_active IP Right Cessation
- 1996-10-25 CA CA002188905A patent/CA2188905C/fr not_active Expired - Fee Related
- 1996-10-25 AR ARP960104928A patent/AR004122A1/es active IP Right Grant
- 1996-10-25 HU HU9602957A patent/HU217773B/hu not_active IP Right Cessation
- 1996-10-26 KR KR1019960048877A patent/KR100443182B1/ko not_active Expired - Fee Related
- 1996-10-27 IL IL11949696A patent/IL119496A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
JP4018182B2 (ja)	2007-12-05
SK284071B6 (sk)	2004-09-08
SG55239A1 (en)	1998-12-21
HUP9602957A3 (en)	1998-01-28
KR970021081A (ko)	1997-05-28
ATE243211T1 (de)	2003-07-15
HU217773B (hu)	2000-04-28
US5808066A (en)	1998-09-15
SI0770615T1 (en)	2003-12-31
EP0770615B1 (fr)	2003-06-18
JPH09124651A (ja)	1997-05-13
ZA968957B (en)	1998-04-24
SK137796A3 (en)	1997-05-07
AR004122A1 (es)	1998-09-30
BR9605258A (pt)	1998-07-21
IL119496A (en)	2001-07-24
IL119496A0 (en)	1997-01-10
CA2188905C (fr)	2005-12-06
TR199600792A2 (tr)	1997-05-21
EP0770615A1 (fr)	1997-05-02
HU9602957D0 (en)	1996-12-30
UA48132C2 (uk)	2002-08-15
DE69628712D1 (de)	2003-07-24
KR100443182B1 (ko)	2005-04-19
PT770615E (pt)	2003-10-31
HUP9602957A2 (en)	1997-06-30
DE69628712T2 (de)	2004-04-29
ES2202419T3 (es)	2004-04-01
RU2147584C1 (ru)	2000-04-20
CA2188905A1 (fr)	1997-04-28
MX9604882A (es)	1997-04-30

Publication	Publication Date	Title
DK0770615T3 (da)	2003-07-14	Fremgangsmåde til fremstilling af dihalogenazolopyrimidiner
DK0747116T3 (da)	2001-11-26	Fremgangsmåde til fremstilling af mikrokapselsammensætninger
DK0812357T3 (da)	2007-05-14	Fremgangsmåde til fremstilling af heteromultimere polypeptider
FI973281L (fi)	1997-08-08	Menetelmä tiettyjen atsasykloheksapeptidien valmistamiseksi
DK1032566T3 (da)	2003-06-10	Fremgangsmåde til fremstilling af citalopram
DK0797542T3 (da)	2002-05-27	Fremgangsmåde til fremstilling af aluminosilikatderivater
DK0775100T3 (da)	2000-11-27	Fremgangsmåde til fremstilling af trifluorethylen
DK0937055T3 (da)	2002-07-29	Fremgangsmåde til fremstilling af d,I-alfa-tocopherol
DK0839138T3 (da)	2004-09-27	Fremgangsmåde til fremstilling af N-substituerede 3-hydroxypyrazoler
DK0768310T3 (da)	2000-04-17	Fremgangsmåde til fremstilling af imidazo-benzodiazepin-derivater
DK0756597T3 (da)	2001-08-20	Fremgangsmåde til fremstilling af puriner
DK0824517T3 (da)	2002-11-18	Fremgangsmåde til fremstilling af lercanidipinhydrochlorid
DK0877738T3 (da)	2003-09-08	Fremgangsmåde til fremstilling af phenylimidazolidinderivater
DK1027315T3 (da)	2003-09-29	Fremgangsmåde til fremstilling af n-butanol
DK0996642T3 (da)	2006-05-08	Fremgangsmåde til fremstilling af heparin
DK0873326T3 (da)	2006-03-27	Fremgangsmåde til fremstilling af 2-chlorthiazolforbindelser
DK0721453T3 (da)	2003-03-17	Fremgangsmåde til fremstilling af N-methyl-3-(1-methyl-4-piperidinyl)-14-indol-5-ethansulfonamid
DK0946514T3 (da)	2003-08-25	Fremgangsmåde til fremstilling af n-substituerede 3-hydroxypyrazoler
DK0815092T3 (da)	1999-12-06	Fremgangsmåde til fremstilling af 1,2-benzisothiazolin-3-oner
DK0648738T3 (da)	1997-06-16	Fremgangsmåde til fremstilling af acetoacetarylamider
DK0735043T3 (da)	1998-10-07	Fremgangsmåde til fremstilling af 2-substitueret 3,3-difluorfuran
NO996432D0 (no)	1999-12-23	Fremgangsmåte for fremstilling av 4-substituert-1H-indol-3- glykosamider
DK0721929T3 (da)	2000-03-27	Fremgangsmåde til fremstilling af hydroxyalkoxybenzophenoner
DK1012152T3 (da)	2003-02-10	Fremgangsmåde til fremstilling af oxazaphosphorin-2-aminer
DK0648748T3 (da)	1997-10-13	Fremgangsmåde til fremstilling af 5-acetoacetylaminobenzimidazolon-2