ATE243211T1 - Verfahren zur herstellung von dihalogenazolopyrimidinen - Google Patents

Verfahren zur herstellung von dihalogenazolopyrimidinen

Info

Publication number: ATE243211T1
Authority: AT; Austria
Prior art keywords: dihalogenazolopyrimidines; producing; producing dihalogenazolopyrimidines
Prior art date: 1995-10-27

Application number

AT96307528T

Other languages

English (en)

Inventor

Guenther Krummel

Karl-Otto Stumm

Klaus-Juergen Pees

Peter Heinz Rudi Liers

Original Assignee

Basf Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-10-27

Filing date

1996-10-16

Publication date

2003-07-15

1996-10-16 Application filed by Basf Ag filed Critical Basf Ag

2003-07-15 Application granted granted Critical

2003-07-15 Publication of ATE243211T1 publication Critical patent/ATE243211T1/de

Links

238000004519 manufacturing process Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT96307528T 1995-10-27 1996-10-16 Verfahren zur herstellung von dihalogenazolopyrimidinen ATE243211T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US802295P	1995-10-27	1995-10-27

Publications (1)

Publication Number	Publication Date
ATE243211T1 true ATE243211T1 (de)	2003-07-15

Family

ID=21729405

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT96307528T ATE243211T1 (de)	1995-10-27	1996-10-16	Verfahren zur herstellung von dihalogenazolopyrimidinen

Country Status (22)

Country	Link
US (1)	US5808066A (de)
EP (1)	EP0770615B1 (de)
JP (1)	JP4018182B2 (de)
KR (1)	KR100443182B1 (de)
AR (1)	AR004122A1 (de)
AT (1)	ATE243211T1 (de)
BR (1)	BR9605258A (de)
CA (1)	CA2188905C (de)
DE (1)	DE69628712T2 (de)
DK (1)	DK0770615T3 (de)
ES (1)	ES2202419T3 (de)
HU (1)	HU217773B (de)
IL (1)	IL119496A (de)
MX (1)	MX9604882A (de)
PT (1)	PT770615E (de)
RU (1)	RU2147584C1 (de)
SG (1)	SG55239A1 (de)
SI (1)	SI0770615T1 (de)
SK (1)	SK284071B6 (de)
TR (1)	TR199600792A2 (de)
UA (1)	UA48132C2 (de)
ZA (1)	ZA968957B (de)

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KR100368102B1 (ko) *	1998-02-11	2003-03-17	아메리칸사이아나미드컴파니	살진균성 7-알킬-트리아졸로피리미딘
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US6242451B1 (en) *	1998-09-25	2001-06-05	Klaus-Juergen Pees	Fungicidal trihalophenyl-triazolopyrimidines
US6559151B2 (en)	2000-05-08	2003-05-06	Basf Aktiengesellschaft	6-(2-trifluoromethyl-phenyl)-triazolopyrimidines
US7683071B2 (en) *	2000-07-26	2010-03-23	Taro Pharmaceuticals Industries Ltd.	Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
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US6756379B2 (en)	2001-07-26	2004-06-29	Taro Pharmaceutical Industries Ltd.	Non-sedating barbiturate compounds as neuroprotective agents
DE10063115A1 (de) *	2000-12-18	2002-06-27	Bayer Ag	Triazolopyrimidine
JP2002249492A (ja) *	2000-12-22	2002-09-06	Nippon Bayer Agrochem Co Ltd	トリアゾロピリミジン類
DE10121101A1 (de) *	2001-04-27	2002-10-31	Bayer Ag	Triazolopyrimidine
DE50209496D1 (de)	2001-07-05	2007-03-29	Basf Ag	Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
EP1412356A1 (de)	2001-07-18	2004-04-28	Basf Aktiengesellschaft	Substituierte 6-(2-methoxyphenyl)triazolopyrimidine als fungizide
UA76486C2 (en)	2001-07-26	2006-08-15	Basf Ag	7-amino triazolopyrimidines, a process of praparation, a fungicidal preparations based thereon and a method to control phytopathogenic fungi
EP1431299B1 (de)	2001-09-04	2007-05-23	Sumitomo Chemical Company, Limited	IMIDAZO(1,2-a)PYRIMIDINE UND DIESE ENTHALTENDE FUNGIZIDZUSAMMENSETZUNGEN
PL372978A1 (en)	2002-03-21	2005-08-08	Basf Aktiengesellschaft	Fungicidal triazolopyrimidines, methods for producing the same, use thereof for combating harmful fungi and agents containing said substances
JP4739760B2 (ja)	2002-12-11	2011-08-03	タロー・ファーマシューティカル・インダストリーズ・リミテッド	バルビツール酸誘導体を使用する運動障害の治療方法
US7419982B2 (en) *	2003-09-24	2008-09-02	Wyeth Holdings Corporation	Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
ES2279452T3 (es) *	2003-09-24	2007-08-16	Wyeth Holdings Corporation	6-((sustituido)fenil)triazolopirimidinas como agentes antineoplasicos.
WO2005030218A1 (en) *	2003-09-24	2005-04-07	Wyeth Holdings Corporation	6-aryl-7-halo-imidazo[1,2-a]pyrimidines as anticancer agent
MY179926A (en) *	2003-12-08	2020-11-19	Wyeth Corp	Process for the preparation of tubulin inhibitors
TW200533670A (en) *	2003-12-19	2005-10-16	Basf Ag	6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
DE102004007076A1 (de) *	2004-02-13	2005-08-25	Bayer Cropscience Ag	Imidazolopyrimidine
CN1930165A (zh) *	2004-03-10	2007-03-14	巴斯福股份公司	5,6－二烷基－7－氨基三唑并嘧啶、其制备方法、在防治致病性真菌中的用途以及包含所述化合物的试剂
JP5005528B2 (ja)	2004-03-10	2012-08-22	ビーエーエスエフソシエタス・ヨーロピア	５，６−ジアルキル−７−アミノトリアゾロピリミジン、その調製、および有害真菌を防除するためのその使用、ならびにそれらの化合物を含む組成物
PE20060020A1 (es) *	2004-03-30	2006-03-10	Basf Ag	5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion
WO2006003651A2 (en) *	2004-07-02	2006-01-12	Taro Pharmaceutical Industries, Ltd	A process for preparing 1-methoxymethyl-5,5-diphenylbarbituric acid
EP1856118A1 (de) *	2005-03-01	2007-11-21	Basf Aktiengesellschaft	5,6-dialkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
CN101128465A (zh) *	2005-03-01	2008-02-20	巴斯福股份公司	5,6-二烷基-7-氨基唑并嘧啶、其制备方法及其在防治病原性真菌中的用途以及包含这些化合物的组合物
EP1856121A1 (de) *	2005-03-01	2007-11-21	Basf Aktiengesellschaft	5,6-dialkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
WO2006092428A2 (de) *	2005-03-02	2006-09-08	Basf Aktiengesellschaft	2-substituierte 7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
BRPI0608411A2 (pt) *	2005-03-10	2009-12-29	Basf Ag	uso de um composto, composto, processo para preparar compostos, agente, semente, e, processo para combater fungos nocivos fitopatogênicos
EP1863752A1 (de) *	2005-03-18	2007-12-12	Basf Aktiengesellschaft	Verfahren zur herstellung von 5-halo-2,4,6-trifluorisophthalsäure
CN101208289A (zh) *	2005-06-27	2008-06-25	巴斯福股份公司	生产取代的苯基丙二酸酯中间体化合物的方法及其在生产5,7-二羟基-6-(2,4,6-三氟苯基)[1,2,4]三唑并[1,5-a]嘧啶中的用途
BRPI0612673A2 (pt) *	2005-06-27	2016-11-29	Basf Ag	processo para preparar compostos, compostos, e, uso de compostos
EP2081576A4 (de) *	2006-11-14	2010-06-30	Taro Pharmaceuticals North Ame	Verfahren zur verbesserung der bioverfügbarkeit für nichtsedierende barbiturate
EP2111404A1 (de) *	2007-01-11	2009-10-28	Basf Se	Verfahren zur herstellung arylsubstituierter anellierter pyrimidine
US8343977B2 (en) *	2009-12-30	2013-01-01	Arqule, Inc.	Substituted triazolo-pyrimidine compounds

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AU557300B2 (en) *	1982-03-16	1986-12-18	Farmitalia Carlo Erba S.P.A.	Substituted 1h-pyrazolo(1,5-alpha)pyrimidines and processes for their preparation
JPS5962593A (ja) *	1982-09-30	1984-04-10	Ss Pharmaceut Co Ltd	３―置換―５，７―ジクロルトリアゾロピリミジン誘導体
DE3522463A1 (de) *	1985-06-22	1987-01-02	Bayer Ag	Herbizide mittel
US4910306A (en) *	1987-11-09	1990-03-20	The Dow Chemical Company	Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US4892945A (en) *	1987-12-21	1990-01-09	Ciba-Geigy Corporation	Isoindoline pigments containing at least one triazolopyrimidone radical
US5006656A (en) *	1990-02-26	1991-04-09	Dowelanco	Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
DE69130683T2 (de) *	1991-04-22	1999-05-06	Otsuka Pharmaceutical Factory, Inc., Naruto, Tokushima	PYRAZOLO[1,5-a]PYRIMIDINDERIVATE UND SIE ENTHALTENDE ANTIINFLAMMATORISCHE MITTEL
US5356897A (en) *	1991-09-09	1994-10-18	Fujisawa Pharmaceutical Co., Ltd.	3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines
US5177206A (en) *	1991-10-08	1993-01-05	Dowelanco	Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides
TW224044B (de) *	1991-12-30	1994-05-21	Shell Internat Res Schappej B V
IL108731A (en) *	1993-03-04	1997-03-18	Shell Int Research	6, N-DISUBSTITUTED-£1, 2, 4\| TRIAZOLO-£1, 5-a\| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
RU2066295C1 (ru) *	1993-05-19	1996-09-10	Институт структурной макрокинетики РАН	Способ получения порошкового материала на основе карбида титана
EP0628559B1 (de) *	1993-06-10	2002-04-03	Beiersdorf-Lilly GmbH	Pyrimidinverbindungen und ihre Verwendung als Pharmazeutika
WO1995011246A1 (en) *	1993-10-18	1995-04-27	Dowelanco	Process for preparing n-(2,6-dichloro-3-methylphenyl)-5-7-dihalo[1,2,4]triazolo[1,5a]pyrimidine-2-sulfonamide by cyclization and halo-dehydroxylation

1996
- 1996-09-30 RU RU96120421A patent/RU2147584C1/ru not_active IP Right Cessation
- 1996-10-03 TR TR96/00792A patent/TR199600792A2/xx unknown
- 1996-10-15 US US08/729,204 patent/US5808066A/en not_active Expired - Lifetime
- 1996-10-16 MX MX9604882A patent/MX9604882A/es not_active IP Right Cessation
- 1996-10-16 ES ES96307528T patent/ES2202419T3/es not_active Expired - Lifetime
- 1996-10-16 AT AT96307528T patent/ATE243211T1/de not_active IP Right Cessation
- 1996-10-16 DE DE69628712T patent/DE69628712T2/de not_active Expired - Lifetime
- 1996-10-16 SI SI9630630T patent/SI0770615T1/xx unknown
- 1996-10-16 DK DK96307528T patent/DK0770615T3/da active
- 1996-10-16 EP EP96307528A patent/EP0770615B1/de not_active Expired - Lifetime
- 1996-10-16 PT PT96307528T patent/PT770615E/pt unknown
- 1996-10-18 SG SG1996010896A patent/SG55239A1/en unknown
- 1996-10-23 JP JP29790396A patent/JP4018182B2/ja not_active Expired - Fee Related
- 1996-10-23 UA UA96104029A patent/UA48132C2/uk unknown
- 1996-10-24 ZA ZA9608957A patent/ZA968957B/xx unknown
- 1996-10-25 SK SK1377-96A patent/SK284071B6/sk unknown
- 1996-10-25 CA CA002188905A patent/CA2188905C/en not_active Expired - Fee Related
- 1996-10-25 BR BR9605258A patent/BR9605258A/pt not_active IP Right Cessation
- 1996-10-25 HU HU9602957A patent/HU217773B/hu not_active IP Right Cessation
- 1996-10-25 AR ARP960104928A patent/AR004122A1/es active IP Right Grant
- 1996-10-26 KR KR1019960048877A patent/KR100443182B1/ko not_active Expired - Fee Related
- 1996-10-27 IL IL11949696A patent/IL119496A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
SI0770615T1 (en)	2003-12-31
UA48132C2 (uk)	2002-08-15
CA2188905C (en)	2005-12-06
IL119496A (en)	2001-07-24
BR9605258A (pt)	1998-07-21
SK284071B6 (sk)	2004-09-08
HU217773B (hu)	2000-04-28
ZA968957B (en)	1998-04-24
HUP9602957A2 (en)	1997-06-30
RU2147584C1 (ru)	2000-04-20
DK0770615T3 (da)	2003-07-14
HU9602957D0 (en)	1996-12-30
EP0770615A1 (de)	1997-05-02
JPH09124651A (ja)	1997-05-13
CA2188905A1 (en)	1997-04-28
IL119496A0 (en)	1997-01-10
SK137796A3 (en)	1997-05-07
TR199600792A2 (tr)	1997-05-21
JP4018182B2 (ja)	2007-12-05
MX9604882A (es)	1997-04-30
DE69628712D1 (de)	2003-07-24
HUP9602957A3 (en)	1998-01-28
DE69628712T2 (de)	2004-04-29
SG55239A1 (en)	1998-12-21
ES2202419T3 (es)	2004-04-01
KR100443182B1 (ko)	2005-04-19
PT770615E (pt)	2003-10-31
EP0770615B1 (de)	2003-06-18
US5808066A (en)	1998-09-15
AR004122A1 (es)	1998-09-30
KR970021081A (ko)	1997-05-28

Legal Events

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2004-01-15

UEP

Publication of translation of european patent specification

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2009-07-15

REN

Ceased due to non-payment of the annual fee

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