ATE243211T1 - Verfahren zur herstellung von dihalogenazolopyrimidinen - Google Patents
Verfahren zur herstellung von dihalogenazolopyrimidinenInfo
- Publication number
- ATE243211T1 ATE243211T1 AT96307528T AT96307528T ATE243211T1 AT E243211 T1 ATE243211 T1 AT E243211T1 AT 96307528 T AT96307528 T AT 96307528T AT 96307528 T AT96307528 T AT 96307528T AT E243211 T1 ATE243211 T1 AT E243211T1
- Authority
- AT
- Austria
- Prior art keywords
- dihalogenazolopyrimidines
- producing
- producing dihalogenazolopyrimidines
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US802295P | 1995-10-27 | 1995-10-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE243211T1 true ATE243211T1 (de) | 2003-07-15 |
Family
ID=21729405
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT96307528T ATE243211T1 (de) | 1995-10-27 | 1996-10-16 | Verfahren zur herstellung von dihalogenazolopyrimidinen |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US5808066A (de) |
| EP (1) | EP0770615B1 (de) |
| JP (1) | JP4018182B2 (de) |
| KR (1) | KR100443182B1 (de) |
| AR (1) | AR004122A1 (de) |
| AT (1) | ATE243211T1 (de) |
| BR (1) | BR9605258A (de) |
| CA (1) | CA2188905C (de) |
| DE (1) | DE69628712T2 (de) |
| DK (1) | DK0770615T3 (de) |
| ES (1) | ES2202419T3 (de) |
| HU (1) | HU217773B (de) |
| IL (1) | IL119496A (de) |
| MX (1) | MX9604882A (de) |
| PT (1) | PT770615E (de) |
| RU (1) | RU2147584C1 (de) |
| SG (1) | SG55239A1 (de) |
| SI (1) | SI0770615T1 (de) |
| SK (1) | SK284071B6 (de) |
| TR (1) | TR199600792A2 (de) |
| UA (1) | UA48132C2 (de) |
| ZA (1) | ZA968957B (de) |
Families Citing this family (40)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6117876A (en) * | 1997-04-14 | 2000-09-12 | American Cyanamid Company | Fungicidal trifluorophenyl-triazolopyrimidines |
| NZ506247A (en) * | 1998-02-11 | 2003-03-28 | American Cyanamid Co | Fungicidal 7-(alkyl, alkenyl, alkadienyl, cycloalkyl, cycloalkenyl or aryl)-[1,2,4]triazolo[1,5-a]pyrimidines |
| US6117865A (en) * | 1998-09-10 | 2000-09-12 | American Cyanamid Company | Fungicidal trifluorophenyl-triazolopyrimidines |
| US6242451B1 (en) * | 1998-09-25 | 2001-06-05 | Klaus-Juergen Pees | Fungicidal trihalophenyl-triazolopyrimidines |
| US6380202B1 (en) * | 1998-09-25 | 2002-04-30 | Basf Aktiengesellschaft | Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines |
| US6156925A (en) * | 1998-09-25 | 2000-12-05 | American Cyanamid Company | Process for the preparation of halogenated phenylmaloates |
| US6559151B2 (en) | 2000-05-08 | 2003-05-06 | Basf Aktiengesellschaft | 6-(2-trifluoromethyl-phenyl)-triazolopyrimidines |
| US6756379B2 (en) * | 2001-07-26 | 2004-06-29 | Taro Pharmaceutical Industries Ltd. | Non-sedating barbiturate compounds as neuroprotective agents |
| US7683071B2 (en) * | 2000-07-26 | 2010-03-23 | Taro Pharmaceuticals Industries Ltd. | Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid |
| US6939873B2 (en) * | 2000-07-26 | 2005-09-06 | Taro Pharmaceuticals Industries Limited | Non-sedating barbituric acid derivatives |
| DE10063115A1 (de) * | 2000-12-18 | 2002-06-27 | Bayer Ag | Triazolopyrimidine |
| JP2002249492A (ja) * | 2000-12-22 | 2002-09-06 | Nippon Bayer Agrochem Co Ltd | トリアゾロピリミジン類 |
| DE10121101A1 (de) * | 2001-04-27 | 2002-10-31 | Bayer Ag | Triazolopyrimidine |
| EA007164B1 (ru) | 2001-07-05 | 2006-08-25 | Басф Акциенгезельшафт | Фунгицидные триазолопиримидины, способ их получения и их применение для борьбы с фитопатогенными грибами, а также содержащие их средства |
| WO2003008416A1 (en) | 2001-07-18 | 2003-01-30 | Basf Aktiengesellschaft | Substituted 6-(2-methoxyphenyl) triazolopyrimides as fungicides |
| DK1414302T3 (da) | 2001-07-26 | 2007-06-18 | Basf Ag | 7-aminotriazolopyrimidiner til bekæmpelse af skadelige svampe |
| ES2287312T3 (es) | 2001-09-04 | 2007-12-16 | Sumitomo Chemical Company, Limited | Imidazo(1,2-a)pirimidinas y composiciones fungicidas que las contienen. |
| IL163709A0 (en) | 2002-03-21 | 2005-12-18 | Basf Ag | Fungicidal triazolopyrimidines, methods for producing the same, use thereof for combating harmful fungiand agents containing said substances |
| ES2315569T3 (es) * | 2002-12-11 | 2009-04-01 | Taro Pharmaceutical Industries Ltd. | Procedimiento de tratamiento de trastornos del movimiento usando derivados de acido barbiturico. |
| US7419982B2 (en) * | 2003-09-24 | 2008-09-02 | Wyeth Holdings Corporation | Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts |
| CN100486580C (zh) * | 2003-09-24 | 2009-05-13 | 惠氏控股公司 | 作为抗癌剂的6-芳基-7-卤基-咪唑并[1,2-a]嘧啶 |
| ES2279452T3 (es) * | 2003-09-24 | 2007-08-16 | Wyeth Holdings Corporation | 6-((sustituido)fenil)triazolopirimidinas como agentes antineoplasicos. |
| MY179926A (en) * | 2003-12-08 | 2020-11-19 | Wyeth Corp | Process for the preparation of tubulin inhibitors |
| TW200533670A (en) * | 2003-12-19 | 2005-10-16 | Basf Ag | 6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds |
| DE102004007076A1 (de) * | 2004-02-13 | 2005-08-25 | Bayer Cropscience Ag | Imidazolopyrimidine |
| US9487519B2 (en) * | 2004-03-10 | 2016-11-08 | Basf Se | 5,6-Dialkyl-7-aminotriazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds |
| EA009883B1 (ru) * | 2004-03-10 | 2008-04-28 | Басф Акциенгезельшафт | 5, 6-диалкил-7-амино-триазолопиримидины, способ их получения и их применение для борьбы с патогенными растениями, а также содержащие их средства |
| PE20060020A1 (es) * | 2004-03-30 | 2006-03-10 | Basf Ag | 5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion |
| CA2572797A1 (en) * | 2004-07-02 | 2006-01-12 | Daniella Gutman | A process for preparing 1-methoxymethyl-5,5-diphenylbarbituric acid |
| TW200640928A (en) * | 2005-03-01 | 2006-12-01 | Basf Ag | 5,6-Dialkyl-7-aminoazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds |
| JP2008532944A (ja) * | 2005-03-01 | 2008-08-21 | ビーエーエスエフ ソシエタス・ヨーロピア | ５，６−ジアルキル−７−アミノアゾロピリミジン、それらの製造方法、有害な菌類を防除するためのそれらの使用、およびそれらの化合物を含む物質 |
| CN101133059A (zh) * | 2005-03-01 | 2008-02-27 | 巴斯福股份公司 | 5,6-二烷基-7-氨基唑并嘧啶、其制备方法及其在防治病原性真菌中的用途以及包含这些化合物的组合物 |
| WO2006092428A2 (de) * | 2005-03-02 | 2006-09-08 | Basf Aktiengesellschaft | 2-substituierte 7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| BRPI0608411A2 (pt) * | 2005-03-10 | 2009-12-29 | Basf Ag | uso de um composto, composto, processo para preparar compostos, agente, semente, e, processo para combater fungos nocivos fitopatogênicos |
| BRPI0608712A2 (pt) * | 2005-03-18 | 2010-12-07 | Basf Ag | processo para a preparação de composto, e, uso do composto |
| WO2007000412A1 (de) * | 2005-06-27 | 2007-01-04 | Basf Aktiengesellschaft | Verfahren zur herstellung von substituierten phenylmalonestern, zwischenverbindungen sowie deren verwendung zur herstellung von 5 , 7-dihydr0xy-6- (2,4, 6-trifluorphenyl) -(1,2 , 4) triazolo (1 , 5-a) pyrimidinen |
| US20080200675A1 (en) * | 2005-06-27 | 2008-08-21 | Basf Aktiengesellschaft | Method for Production of Substituted Phenylmalonate Esters, Novel Phenylmalonate Esters and Use Thereof |
| EP2081576A4 (de) * | 2006-11-14 | 2010-06-30 | Taro Pharmaceuticals North Ame | Verfahren zur verbesserung der bioverfügbarkeit für nichtsedierende barbiturate |
| US20100087640A1 (en) * | 2007-01-11 | 2010-04-08 | Basf Se | Method for production of aryl-substituted annelated pyrimidines |
| US8343977B2 (en) * | 2009-12-30 | 2013-01-01 | Arqule, Inc. | Substituted triazolo-pyrimidine compounds |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3907799A (en) * | 1971-08-16 | 1975-09-23 | Icn Pharmaceuticals | Xanthine oxidase inhibitors |
| AU557300B2 (en) * | 1982-03-16 | 1986-12-18 | Farmitalia Carlo Erba S.P.A. | Substituted 1h-pyrazolo(1,5-alpha)pyrimidines and processes for their preparation |
| JPS5962593A (ja) * | 1982-09-30 | 1984-04-10 | Ss Pharmaceut Co Ltd | ３―置換―５，７―ジクロルトリアゾロピリミジン誘導体 |
| DE3522463A1 (de) * | 1985-06-22 | 1987-01-02 | Bayer Ag | Herbizide mittel |
| US4910306A (en) * | 1987-11-09 | 1990-03-20 | The Dow Chemical Company | Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides |
| US4892945A (en) * | 1987-12-21 | 1990-01-09 | Ciba-Geigy Corporation | Isoindoline pigments containing at least one triazolopyrimidone radical |
| US5006656A (en) * | 1990-02-26 | 1991-04-09 | Dowelanco | Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides |
| AU651986B2 (en) * | 1991-04-22 | 1994-08-11 | Otsuka Pharmaceutical Factory, Inc. | Pyrazolo{1,5-a}pyrimidine derivative and anti-inflammatory containing the same |
| US5356897A (en) * | 1991-09-09 | 1994-10-18 | Fujisawa Pharmaceutical Co., Ltd. | 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines |
| US5177206A (en) * | 1991-10-08 | 1993-01-05 | Dowelanco | Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides |
| TW224044B (de) * | 1991-12-30 | 1994-05-21 | Shell Internat Res Schappej B V | |
| IL108731A (en) * | 1993-03-04 | 1997-03-18 | Shell Int Research | 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES |
| RU2066295C1 (ru) * | 1993-05-19 | 1996-09-10 | Институт структурной макрокинетики РАН | Способ получения порошкового материала на основе карбида титана |
| EP0628559B1 (de) * | 1993-06-10 | 2002-04-03 | Beiersdorf-Lilly GmbH | Pyrimidinverbindungen und ihre Verwendung als Pharmazeutika |
| DE69429728T2 (de) * | 1993-10-18 | 2002-10-31 | Dow Agrosciences Llc, Indianapolis | Verfahren zur herstellung von n-(2,6-dichloro-3-methylphenyl)-5-7-dihalo[1,2,4]triazolo[1,5a]pyrimidin-2-sulfonamid durch cyclisierung und halo-dehydroxylierung |
-
1996
- 1996-09-30 RU RU96120421A patent/RU2147584C1/ru not_active IP Right Cessation
- 1996-10-03 TR TR96/00792A patent/TR199600792A2/xx unknown
- 1996-10-15 US US08/729,204 patent/US5808066A/en not_active Expired - Lifetime
- 1996-10-16 SI SI9630630T patent/SI0770615T1/xx unknown
- 1996-10-16 ES ES96307528T patent/ES2202419T3/es not_active Expired - Lifetime
- 1996-10-16 MX MX9604882A patent/MX9604882A/es not_active IP Right Cessation
- 1996-10-16 EP EP96307528A patent/EP0770615B1/de not_active Expired - Lifetime
- 1996-10-16 PT PT96307528T patent/PT770615E/pt unknown
- 1996-10-16 DE DE69628712T patent/DE69628712T2/de not_active Expired - Lifetime
- 1996-10-16 AT AT96307528T patent/ATE243211T1/de not_active IP Right Cessation
- 1996-10-16 DK DK96307528T patent/DK0770615T3/da active
- 1996-10-18 SG SG1996010896A patent/SG55239A1/en unknown
- 1996-10-23 JP JP29790396A patent/JP4018182B2/ja not_active Expired - Fee Related
- 1996-10-23 UA UA96104029A patent/UA48132C2/uk unknown
- 1996-10-24 ZA ZA9608957A patent/ZA968957B/xx unknown
- 1996-10-25 HU HU9602957A patent/HU217773B/hu not_active IP Right Cessation
- 1996-10-25 SK SK1377-96A patent/SK284071B6/sk unknown
- 1996-10-25 BR BR9605258A patent/BR9605258A/pt not_active IP Right Cessation
- 1996-10-25 AR ARP960104928A patent/AR004122A1/es active IP Right Grant
- 1996-10-25 CA CA002188905A patent/CA2188905C/en not_active Expired - Fee Related
- 1996-10-26 KR KR1019960048877A patent/KR100443182B1/ko not_active Expired - Fee Related
- 1996-10-27 IL IL11949696A patent/IL119496A/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| SG55239A1 (en) | 1998-12-21 |
| US5808066A (en) | 1998-09-15 |
| JP4018182B2 (ja) | 2007-12-05 |
| AR004122A1 (es) | 1998-09-30 |
| ZA968957B (en) | 1998-04-24 |
| TR199600792A2 (tr) | 1997-05-21 |
| JPH09124651A (ja) | 1997-05-13 |
| ES2202419T3 (es) | 2004-04-01 |
| SK137796A3 (en) | 1997-05-07 |
| HU217773B (hu) | 2000-04-28 |
| SI0770615T1 (en) | 2003-12-31 |
| BR9605258A (pt) | 1998-07-21 |
| DE69628712T2 (de) | 2004-04-29 |
| EP0770615B1 (de) | 2003-06-18 |
| CA2188905C (en) | 2005-12-06 |
| PT770615E (pt) | 2003-10-31 |
| CA2188905A1 (en) | 1997-04-28 |
| KR970021081A (ko) | 1997-05-28 |
| HU9602957D0 (en) | 1996-12-30 |
| IL119496A0 (en) | 1997-01-10 |
| IL119496A (en) | 2001-07-24 |
| HUP9602957A2 (en) | 1997-06-30 |
| DE69628712D1 (de) | 2003-07-24 |
| EP0770615A1 (de) | 1997-05-02 |
| KR100443182B1 (ko) | 2005-04-19 |
| MX9604882A (es) | 1997-04-30 |
| RU2147584C1 (ru) | 2000-04-20 |
| DK0770615T3 (da) | 2003-07-14 |
| UA48132C2 (uk) | 2002-08-15 |
| SK284071B6 (sk) | 2004-09-08 |
| HUP9602957A3 (en) | 1998-01-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
Ref document number: 0770615 Country of ref document: EP |
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| REN | Ceased due to non-payment of the annual fee |